TR200000952A2 - Synthesis of 1,1-dioxopenicillaniloxymethyl 6- [D-alpha- (benzylideneamino-phenylacetamido)] penicillanate and the like. New intermediates suitable for the synthesis of sultamicillin. - Google Patents
Synthesis of 1,1-dioxopenicillaniloxymethyl 6- [D-alpha- (benzylideneamino-phenylacetamido)] penicillanate and the like. New intermediates suitable for the synthesis of sultamicillin.Info
- Publication number
- TR200000952A2 TR200000952A2 TR2000/00952A TR200000952A TR200000952A2 TR 200000952 A2 TR200000952 A2 TR 200000952A2 TR 2000/00952 A TR2000/00952 A TR 2000/00952A TR 200000952 A TR200000952 A TR 200000952A TR 200000952 A2 TR200000952 A2 TR 200000952A2
- Authority
- TR
- Turkey
- Prior art keywords
- synthesis
- dioxopenicillaniloxymethyl
- sultamicillin
- alpha
- penicillanate
- Prior art date
Links
Abstract
Bu bulus, 1,1-dioksopenisilanoiloksimetil 6-[D-alfa-(aminofenilasetamido)]penisilanat ve benzerlerinin sentezini tanimlamaktadir. Bu yeni ürünler, ya serbest baz ya da tosilat tuzu olarak sültamisilinin orta ve yüksek verimde hazirlanmasinda etkin ara ürünler olduklarini göstermistir.This invention describes the synthesis of 1,1-dioxopenicillaniloxymethyl 6- [D-alpha- (aminophenylacetamido)] peniculanate and the like. These new products have shown that they are effective intermediates in the preparation of sultamicillin as a free base or tosylate salt in medium and high yields.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ES9900717A ES2161602B1 (en) | 1999-04-08 | 1999-04-08 | SYNTHESIS OF 6- (D-ALPHA- (BENCILIDENAMINOPHENYLACETAMIDE)) PENICILANATE 1,1-DIOXOPENICILANLANILOXIMETILO AND ANALOGS. NEW INTERMEDIATES FOR SYNTHESIS OF SULTAMICILLIN. |
Publications (2)
Publication Number | Publication Date |
---|---|
TR200000952A3 TR200000952A3 (en) | 2000-11-21 |
TR200000952A2 true TR200000952A2 (en) | 2000-11-21 |
Family
ID=8307946
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TR2000/00952A TR200000952A2 (en) | 1999-04-08 | 2000-04-10 | Synthesis of 1,1-dioxopenicillaniloxymethyl 6- [D-alpha- (benzylideneamino-phenylacetamido)] penicillanate and the like. New intermediates suitable for the synthesis of sultamicillin. |
Country Status (3)
Country | Link |
---|---|
JP (1) | JP2000344783A (en) |
ES (1) | ES2161602B1 (en) |
TR (1) | TR200000952A2 (en) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2007004239A1 (en) * | 2005-07-06 | 2007-01-11 | Morepen Laboratories Limited | New polymorphic form of sultamicillin tosylate and a process therefor |
CN100336816C (en) * | 2005-12-14 | 2007-09-12 | 广州大学 | Preparation method of sulbactam |
Citations (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2052992A1 (en) * | 1969-06-20 | 1971-04-16 | Clin Midy | Alpha aldimino benzyl penicillins |
FR2230649A1 (en) * | 1973-05-23 | 1974-12-20 | Aries Robert | Alkanoyloxymethyl esters of penicillins - with alpha-(methyleneimino)phenylacetamido side-chain with long duration of action |
GB1461860A (en) * | 1974-10-22 | 1977-01-19 | Prodotti Antibiotici Spa | Semi-synthetic penicillin |
EP0112087A1 (en) * | 1982-12-06 | 1984-06-27 | Pfizer Inc. | Process and intermediates for sultamicillin and analogs |
EP0405316A2 (en) * | 1989-06-20 | 1991-01-02 | Yeong Sul Kim | 1,1-dioxopenicillanoyloxymethyl D-6-[alpha(methyleneamino)-phenyl-acetamidol]-penicillanate and a process for the preparation thereof |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IE49881B1 (en) * | 1979-02-13 | 1986-01-08 | Leo Pharm Prod Ltd | B-lactam intermediates |
IL64009A (en) * | 1980-10-31 | 1984-09-30 | Rech Applications Therap | Crystalline 1,1-dioxopenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate tosylate hydrates,their production and pharmaceutical compositions containing them |
US4381263A (en) * | 1981-03-23 | 1983-04-26 | Pfizer Inc. | Process for the preparation of penicillanic acid esters |
ES2100125B1 (en) * | 1995-06-02 | 1998-04-01 | Asturpharma S A | PROCEDURE FOR THE PREPARATION OF METHANODIOL ESTERS OF DIOXOPENICILANIC ACID. |
-
1999
- 1999-04-08 ES ES9900717A patent/ES2161602B1/en not_active Expired - Lifetime
-
2000
- 2000-04-10 TR TR2000/00952A patent/TR200000952A2/en unknown
- 2000-04-10 JP JP2000108544A patent/JP2000344783A/en active Pending
Patent Citations (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2052992A1 (en) * | 1969-06-20 | 1971-04-16 | Clin Midy | Alpha aldimino benzyl penicillins |
FR2230649A1 (en) * | 1973-05-23 | 1974-12-20 | Aries Robert | Alkanoyloxymethyl esters of penicillins - with alpha-(methyleneimino)phenylacetamido side-chain with long duration of action |
GB1461860A (en) * | 1974-10-22 | 1977-01-19 | Prodotti Antibiotici Spa | Semi-synthetic penicillin |
EP0112087A1 (en) * | 1982-12-06 | 1984-06-27 | Pfizer Inc. | Process and intermediates for sultamicillin and analogs |
EP0405316A2 (en) * | 1989-06-20 | 1991-01-02 | Yeong Sul Kim | 1,1-dioxopenicillanoyloxymethyl D-6-[alpha(methyleneamino)-phenyl-acetamidol]-penicillanate and a process for the preparation thereof |
Also Published As
Publication number | Publication date |
---|---|
TR200000952A3 (en) | 2000-11-21 |
ES2161602A1 (en) | 2001-12-01 |
ES2161602B1 (en) | 2003-02-16 |
JP2000344783A (en) | 2000-12-12 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ES2173480T3 (en) | PREPARATION OF CICLOHEXENO CARBOXYLATE DERIVATIVES. | |
BR0115273A (en) | Methods for preparing a plurality of agglomerated abrasive grains, and an abrasive article | |
AU3877500A (en) | Methods for preparing 3-aryloxy-3-arylpropylamines and intermediates thereof | |
IL130260A0 (en) | 3-thiocarbamoylpyrazole derivatives as pesticides | |
SE9901875D0 (en) | Novel compounds | |
MX9709240A (en) | Phenylpyridazinones. | |
HK1030218A1 (en) | Novel 2-(iminomethyl)amino-phenyl derivatives, preparation, application as medicines and compositions containing same. | |
FI973475A0 (en) | Composition and product are obtained | |
CY1112871T1 (en) | METHOD AND INTERMEDIATE UNIONS | |
NO990789L (en) | Cytotoxic amino sugar and related sugar derivatives of indolopyrrolocarbazoles | |
DK1083903T3 (en) | Bridged Indopyrrolocarbazoles | |
DK0681574T3 (en) | C7 taxane derivatives and pharmaceutical compositions containing them | |
TR200000952A2 (en) | Synthesis of 1,1-dioxopenicillaniloxymethyl 6- [D-alpha- (benzylideneamino-phenylacetamido)] penicillanate and the like. New intermediates suitable for the synthesis of sultamicillin. | |
DE60141654D1 (en) | PROCESS FOR THE PREPARATION OF HETERORYLAMINE DERIVATIVES | |
DK0864255T3 (en) | Water-continuously spreadable product | |
DK1017681T3 (en) | Hydrazone-benzazulin derivatives, pharmaceuticals and intermediates | |
DE60111614D1 (en) | TAXAN DERIVATIVES FOR THE TREATMENT OF CANCER | |
PT1011329E (en) | 7-METHYLTHYOXXYETHYL AND 7-METHYLTHYDROXYETHYL PACLITAXES | |
ID27656A (en) | AZABISIKLOHEPTANA N-SUBSTITUTIONAL DERIVES, THE PRODUCTION AND USE OF IT | |
DE60044804D1 (en) | ACYL DERIVATIVES OF THE 4-DEMETHYLENE CLOMEDINE, USE AND PREPARATION THEREOF | |
IT1306207B1 (en) | PRODUCTION OF HETEROLOGICAL PROTEINS FROM ZYGOSACCHAROMYCES BAILII. | |
IT1290444B1 (en) | CONJUGATES OF BIS-PHOSPHONATES WITH ALKYLANTS FUNCTIONALITY HAVING ANTI-TUMOR ACTIVITIES | |
IT243461Y1 (en) | EXHIBITOR OF JEWELS, PARTICULARLY FOR SHOWCASES. | |
TW200505413A (en) | Intermediates useful in the synthesis of hiv-protease inhibitors and methods for preparing the same | |
Conlon | Increase booth traffic with demonstrations. |