TR199902963T2 - Composition containing 5-$4-$2-(N-Methyl-N-2-Pyridyl)Amino)Ethoxy]Benzyl]Thiazolidine-2,4-Dion - Google Patents

Composition containing 5-$4-$2-(N-Methyl-N-2-Pyridyl)Amino)Ethoxy]Benzyl]Thiazolidine-2,4-Dion

Info

Publication number
TR199902963T2
TR199902963T2 TR1999/02963T TR9902963T TR199902963T2 TR 199902963 T2 TR199902963 T2 TR 199902963T2 TR 1999/02963 T TR1999/02963 T TR 1999/02963T TR 9902963 T TR9902963 T TR 9902963T TR 199902963 T2 TR199902963 T2 TR 199902963T2
Authority
TR
Turkey
Prior art keywords
dion
thiazolidine
pyridyl
ethoxy
benzyl
Prior art date
Application number
TR1999/02963T
Other languages
Turkish (tr)
Inventor
Patel Jai
Ross Hamish
Price Robin
Roger Granett Jeffrey
Nigel Wray Paul
Original Assignee
Smithkline Beecham P.L.C.
Smithkline Beecham Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9712851.6A external-priority patent/GB9712851D0/en
Application filed by Smithkline Beecham P.L.C., Smithkline Beecham Corporation filed Critical Smithkline Beecham P.L.C.
Publication of TR199902963T2 publication Critical patent/TR199902963T2/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

Terkibin farmasötik olarak kabul edilebilir formda ve farmasötik olarak kabul edilebilir bir tasiyici içinde 2 ila 12 mg Bilesik (I) içermesi ile karakterize edilen bir terkip; böyle bir terkibin ilaç yapiminda kullanilmasi; böyle bir terkibin ve böyle bir proseste faydali bir ara terkibin hazirlanmasi için prosesler.A composition characterized in that the composition contains 2 to 12 mg of Compound (I) in a pharmaceutically acceptable form and in a pharmaceutically acceptable carrier; use of such a composition in medicine; processes for the preparation of such a composition and an intermediate composition useful in such a process.

TR1999/02963T 1997-06-05 1998-06-02 Composition containing 5-$4-$2-(N-Methyl-N-2-Pyridyl)Amino)Ethoxy]Benzyl]Thiazolidine-2,4-Dion TR199902963T2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9711683.4A GB9711683D0 (en) 1997-06-05 1997-06-05 Composition
GBGB9712851.6A GB9712851D0 (en) 1997-06-18 1997-06-18 Composition

Publications (1)

Publication Number Publication Date
TR199902963T2 true TR199902963T2 (en) 2000-02-21

Family

ID=26311662

Family Applications (2)

Application Number Title Priority Date Filing Date
TR2000/02790T TR200002790T2 (en) 1997-06-05 1998-06-02 Composition containing 5- (4- (2- (N-methyl-N-2-pyridyl) amino) ethoxy) benzyl) thiazolidin-2,4-dione
TR1999/02963T TR199902963T2 (en) 1997-06-05 1998-06-02 Composition containing 5-$4-$2-(N-Methyl-N-2-Pyridyl)Amino)Ethoxy]Benzyl]Thiazolidine-2,4-Dion

Family Applications Before (1)

Application Number Title Priority Date Filing Date
TR2000/02790T TR200002790T2 (en) 1997-06-05 1998-06-02 Composition containing 5- (4- (2- (N-methyl-N-2-pyridyl) amino) ethoxy) benzyl) thiazolidin-2,4-dione

Country Status (29)

Country Link
EP (1) EP0998284A1 (en)
JP (1) JP2001521553A (en)
KR (1) KR20010013410A (en)
CN (3) CN1112926C (en)
AP (1) AP1214A (en)
AR (2) AR008198A1 (en)
AU (1) AU8215098A (en)
BG (1) BG104048A (en)
BR (1) BR9810405A (en)
CA (2) CA2333352A1 (en)
CO (1) CO4940400A1 (en)
DZ (1) DZ2510A1 (en)
EA (1) EA002384B1 (en)
GB (1) GB9711683D0 (en)
HU (1) HUP0004070A3 (en)
ID (1) ID24264A (en)
IL (1) IL133074A0 (en)
MX (1) MXPA99011322A (en)
NO (2) NO995938L (en)
NZ (2) NZ523725A (en)
OA (1) OA11306A (en)
PE (1) PE78899A1 (en)
PL (1) PL337201A1 (en)
SK (1) SK164899A3 (en)
TR (2) TR200002790T2 (en)
TW (1) TW570797B (en)
UY (1) UY25032A1 (en)
WO (1) WO1998055122A1 (en)
ZA (2) ZA984826B (en)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20040248945A1 (en) 1999-04-23 2004-12-09 Smithkline Beecham P.L.C. Thiazolidinedione derivative and its use as antidiabetic
CO5170421A1 (en) 1999-04-23 2002-06-27 Smithkline Beecham Plc NEW MALEICO PHARMACEUTICAL COMPOUND
DZ3155A1 (en) 1999-04-23 2000-11-02 Smithkline Beecham Plc New pharmaceutical composition.
GB0021978D0 (en) 2000-09-07 2000-10-25 Smithkline Beecham Plc Novel pharmaceutical
GB0127805D0 (en) * 2001-11-20 2002-01-09 Smithkline Beecham Plc Pharmaceutical composition
GB0129871D0 (en) * 2001-12-13 2002-02-06 Smithkline Beecham Plc Novel pharmaceutical
GB0129876D0 (en) * 2001-12-13 2002-02-06 Smithkline Beecham Plc Novel pharmaceutical
AU2002350965A1 (en) * 2001-12-13 2003-06-23 Smithkline Beecham Plc Toluenesulfonate hydrates of a thiazolidinedione derivative
GB0130509D0 (en) * 2001-12-20 2002-02-06 Smithkline Beecham Plc Novel pharmaceutical
DE06252444T8 (en) * 2006-05-09 2009-03-19 Teva Pharmaceutical Industries Ltd. 2-N- {5 - [[4- [2- (Methyl-2-pyridinylamino) -ethoxy] -phenyl] -methyl] -2,4-thiazolidinedione-succinic acid, method of preparation and compositions with rosiglitazone maleate
US7435741B2 (en) 2006-05-09 2008-10-14 Teva Pharmaceutical Industries, Ltd. 2-N{5-[[4-[2-(methyl-2-pyridinylamino) ethoxy] phenyl]methyl]-2,4-thiazolidinedione} butanedioic acid, methods of preparation and compositions with rosiglitazone maleate
WO2015008234A1 (en) * 2013-07-17 2015-01-22 Glenmark Pharmaceuticals S.A. Bicyclic heterocyclic compounds as ror gamma modulators

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3856378T2 (en) * 1987-09-04 2000-05-11 Beecham Group Plc Substituted thiazolidinedione derivatives
GB9218830D0 (en) * 1992-09-05 1992-10-21 Smithkline Beecham Plc Novel compounds
EP0777469A1 (en) * 1994-02-10 1997-06-11 Smithkline Beecham Plc Use of insulin sensitisers for treating renal diseases
CN1192683A (en) * 1995-08-10 1998-09-09 沃尼尔·朗伯公司 Method for reducing amount of exogenous insulin administered to a patient having noninsulin-dependent diabetes mellitus
AU7604596A (en) * 1995-11-17 1997-06-11 Warner-Lambert Company A method of treating myotonic dystrophy
NZ314406A (en) * 1996-03-18 2000-12-22 Sankyo Co Treatment or prophylaxis of pancreatitis with a medicament containing an insulin sensitiser including oxazoles and thiazoles
CN1230114A (en) * 1996-07-12 1999-09-29 史密丝克莱恩比彻姆有限公司 Novel treatment of leptine resistance

Also Published As

Publication number Publication date
OA11306A (en) 2003-10-22
IL133074A0 (en) 2001-03-19
BG104048A (en) 2000-07-31
GB9711683D0 (en) 1997-08-06
NZ513922A (en) 2001-09-28
CN1430959A (en) 2003-07-23
TW570797B (en) 2004-01-11
CN1112926C (en) 2003-07-02
BR9810405A (en) 2000-08-29
TR200002790T2 (en) 2001-11-21
KR20010013410A (en) 2001-02-26
NO995938L (en) 2000-02-02
CA2292629C (en) 2004-01-06
HUP0004070A2 (en) 2002-02-28
ZA9811572B (en) 1999-07-22
AP1214A (en) 2003-10-08
DZ2510A1 (en) 2003-01-25
NO995938D0 (en) 1999-12-03
AR008198A1 (en) 1999-12-29
JP2001521553A (en) 2001-11-06
HUP0004070A3 (en) 2002-03-28
CN1259050A (en) 2000-07-05
NO20040738L (en) 2000-02-02
UY25032A1 (en) 1998-11-26
CO4940400A1 (en) 2000-07-24
AP9901696A0 (en) 1999-12-31
AU8215098A (en) 1998-12-21
CA2292629A1 (en) 1998-12-10
NZ523725A (en) 2004-09-24
AR015120A1 (en) 2001-04-18
ZA984826B (en) 1999-08-03
EA199901116A1 (en) 2000-06-26
CN1526391A (en) 2004-09-08
PL337201A1 (en) 2000-08-14
CA2333352A1 (en) 1998-12-10
MXPA99011322A (en) 2004-12-02
ID24264A (en) 2000-07-13
EP0998284A1 (en) 2000-05-10
PE78899A1 (en) 1999-10-22
WO1998055122A1 (en) 1998-12-10
EA002384B1 (en) 2002-04-25
SK164899A3 (en) 2000-11-07

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