PE78899A1 - COMPOSITION OF 5- [4- [2- (N-METHYL-N- (2-PIRIDIL) AMINO) ETOXI] BENCIL] THIAZOLIDIN-2,4-DIONA - Google Patents
COMPOSITION OF 5- [4- [2- (N-METHYL-N- (2-PIRIDIL) AMINO) ETOXI] BENCIL] THIAZOLIDIN-2,4-DIONAInfo
- Publication number
- PE78899A1 PE78899A1 PE1998000466A PE00046698A PE78899A1 PE 78899 A1 PE78899 A1 PE 78899A1 PE 1998000466 A PE1998000466 A PE 1998000466A PE 00046698 A PE00046698 A PE 00046698A PE 78899 A1 PE78899 A1 PE 78899A1
- Authority
- PE
- Peru
- Prior art keywords
- piridil
- etoxi
- bencil
- diona
- thiazolidin
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
Abstract
CARACTERIZADA PORQUE COMPRENDE UN COMPUESTO 5-[4-[2-(N-METIL-N-(2-PIRIDIL)AMINO)ETOXI]BENCIL]TIAZOLIDIN-2,4-DIONA DE 2 A 12 mg O COMO UNA SAL DE MALEATO. TAMBIEN SE REFIERE A UN PROCEDIMIENTO PARA LA PREPARACION QUE COMPRENDE LA MEZCLA DEL COMPUESTO CON UN PRIMER VEHICULO, LUEGO MEZCLAR CON UN SEGUNDO VEHICULO. TAMBIEN SE REFIERE A UNA COMPOSICION QUE COMPRENDE EL COMPUESTO, SAL SODICA DE GLICOLATO DE ALMIDON, HIDROXIPROPILMETILCELULOSA 2910, CELULOSA MICRO-CRISTALINA Y LACTOSA MONOHIDRATADACHARACTERIZED BECAUSE IT INCLUDES A COMPOUND 5- [4- [2- (N-METHYL-N- (2-PIRIDIL) AMINO) ETOXI] BENCIL] THIAZOLIDIN-2,4-DIONA FROM 2 TO 12 mg OR AS A MALEATE SALT. IT ALSO REFERS TO A PREPARATION PROCEDURE WHICH INCLUDES THE MIXTURE OF THE COMPOUND WITH A FIRST VEHICLE, THEN MIX WITH A SECOND VEHICLE. ALSO REFERS TO A COMPOSITION THAT INCLUDES THE COMPOUND, SODIUM SALT OF STARCH GLYCOLATE, HYDROXYPROPYL METHYL CELLULOSE 2910, MICRO-CRYSTALLINE CELLULOSE AND MONOHYDRATED LACTOSE
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB9711683.4A GB9711683D0 (en) | 1997-06-05 | 1997-06-05 | Composition |
GBGB9712851.6A GB9712851D0 (en) | 1997-06-18 | 1997-06-18 | Composition |
Publications (1)
Publication Number | Publication Date |
---|---|
PE78899A1 true PE78899A1 (en) | 1999-10-22 |
Family
ID=26311662
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PE1998000466A PE78899A1 (en) | 1997-06-05 | 1998-06-05 | COMPOSITION OF 5- [4- [2- (N-METHYL-N- (2-PIRIDIL) AMINO) ETOXI] BENCIL] THIAZOLIDIN-2,4-DIONA |
Country Status (29)
Country | Link |
---|---|
EP (1) | EP0998284A1 (en) |
JP (1) | JP2001521553A (en) |
KR (1) | KR20010013410A (en) |
CN (3) | CN1112926C (en) |
AP (1) | AP1214A (en) |
AR (2) | AR008198A1 (en) |
AU (1) | AU8215098A (en) |
BG (1) | BG104048A (en) |
BR (1) | BR9810405A (en) |
CA (2) | CA2333352A1 (en) |
CO (1) | CO4940400A1 (en) |
DZ (1) | DZ2510A1 (en) |
EA (1) | EA002384B1 (en) |
GB (1) | GB9711683D0 (en) |
HU (1) | HUP0004070A3 (en) |
ID (1) | ID24264A (en) |
IL (1) | IL133074A0 (en) |
MX (1) | MXPA99011322A (en) |
NO (2) | NO995938L (en) |
NZ (2) | NZ523725A (en) |
OA (1) | OA11306A (en) |
PE (1) | PE78899A1 (en) |
PL (1) | PL337201A1 (en) |
SK (1) | SK164899A3 (en) |
TR (2) | TR200002790T2 (en) |
TW (1) | TW570797B (en) |
UY (1) | UY25032A1 (en) |
WO (1) | WO1998055122A1 (en) |
ZA (2) | ZA984826B (en) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20040248945A1 (en) | 1999-04-23 | 2004-12-09 | Smithkline Beecham P.L.C. | Thiazolidinedione derivative and its use as antidiabetic |
PL351684A1 (en) * | 1999-04-23 | 2003-06-02 | Smithkline Beecham Plc | Polymorph of 5−[4−[2− (n−methyl−n−( 2−pyridyl)amino) ethoxy]benzyl] thiazolidine−2,4−dione, maleic acid salt |
WO2000064892A2 (en) | 1999-04-23 | 2000-11-02 | Smithkline Beecham P.L.C. | Thiazolidinedione derivative and its use as antidiabetic |
GB0021978D0 (en) | 2000-09-07 | 2000-10-25 | Smithkline Beecham Plc | Novel pharmaceutical |
GB0127805D0 (en) * | 2001-11-20 | 2002-01-09 | Smithkline Beecham Plc | Pharmaceutical composition |
AU2002350965A1 (en) * | 2001-12-13 | 2003-06-23 | Smithkline Beecham Plc | Toluenesulfonate hydrates of a thiazolidinedione derivative |
GB0129871D0 (en) * | 2001-12-13 | 2002-02-06 | Smithkline Beecham Plc | Novel pharmaceutical |
GB0129876D0 (en) * | 2001-12-13 | 2002-02-06 | Smithkline Beecham Plc | Novel pharmaceutical |
GB0130509D0 (en) * | 2001-12-20 | 2002-02-06 | Smithkline Beecham Plc | Novel pharmaceutical |
ES2294980T1 (en) * | 2006-05-09 | 2008-04-16 | Teva Pharmaceutical Industries Ltd. | ACID 2-N- (5 - ((4- (2- (METHYL-2-PYRIDINYLAMINE) ETHOXY) PHENYL) METHYL) -2,4-THIAZOLIDINDIONA) -BUTANODIOIC, PREPARATION PROCEDURES AND COMPOSITIONS WITH ROSIGLITAZONA MALEATE. |
US7435741B2 (en) | 2006-05-09 | 2008-10-14 | Teva Pharmaceutical Industries, Ltd. | 2-N{5-[[4-[2-(methyl-2-pyridinylamino) ethoxy] phenyl]methyl]-2,4-thiazolidinedione} butanedioic acid, methods of preparation and compositions with rosiglitazone maleate |
WO2015008234A1 (en) * | 2013-07-17 | 2015-01-22 | Glenmark Pharmaceuticals S.A. | Bicyclic heterocyclic compounds as ror gamma modulators |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3856378T2 (en) * | 1987-09-04 | 2000-05-11 | Beecham Group Plc | Substituted thiazolidinedione derivatives |
GB9218830D0 (en) * | 1992-09-05 | 1992-10-21 | Smithkline Beecham Plc | Novel compounds |
WO1995021608A1 (en) * | 1994-02-10 | 1995-08-17 | Smithkline Beecham Plc | Use of insulin sensitisers for treating renal diseases |
NZ313874A (en) * | 1995-08-10 | 2000-09-29 | Warner Lambert Co | Compounds used as medicaments useful in eliminating the amount of exogenous insulin administered to a patient having noninsulin-dependent diabetes mellitus |
AU7604596A (en) * | 1995-11-17 | 1997-06-11 | Warner-Lambert Company | A method of treating myotonic dystrophy |
NZ314406A (en) * | 1996-03-18 | 2000-12-22 | Sankyo Co | Treatment or prophylaxis of pancreatitis with a medicament containing an insulin sensitiser including oxazoles and thiazoles |
CA2260044A1 (en) * | 1996-07-12 | 1998-01-22 | Stephen Alistair Smith | Novel treatment of leptine resistance |
-
1997
- 1997-06-05 GB GBGB9711683.4A patent/GB9711683D0/en active Pending
-
1998
- 1998-06-02 WO PCT/EP1998/003478 patent/WO1998055122A1/en not_active Application Discontinuation
- 1998-06-02 NZ NZ523725A patent/NZ523725A/en unknown
- 1998-06-02 IL IL13307498A patent/IL133074A0/en unknown
- 1998-06-02 BR BR9810405-5A patent/BR9810405A/en not_active IP Right Cessation
- 1998-06-02 CA CA002333352A patent/CA2333352A1/en not_active Abandoned
- 1998-06-02 CN CN98805686A patent/CN1112926C/en not_active Expired - Lifetime
- 1998-06-02 TR TR2000/02790T patent/TR200002790T2/en unknown
- 1998-06-02 CA CA002292629A patent/CA2292629C/en not_active Expired - Fee Related
- 1998-06-02 HU HU0004070A patent/HUP0004070A3/en unknown
- 1998-06-02 CN CNA2003101199090A patent/CN1526391A/en active Pending
- 1998-06-02 JP JP50158799A patent/JP2001521553A/en not_active Ceased
- 1998-06-02 MX MXPA99011322A patent/MXPA99011322A/en unknown
- 1998-06-02 EP EP98932144A patent/EP0998284A1/en not_active Withdrawn
- 1998-06-02 ID IDW991520A patent/ID24264A/en unknown
- 1998-06-02 TR TR1999/02963T patent/TR199902963T2/en unknown
- 1998-06-02 KR KR19997011411A patent/KR20010013410A/en not_active Application Discontinuation
- 1998-06-02 SK SK1648-99A patent/SK164899A3/en unknown
- 1998-06-02 PL PL98337201A patent/PL337201A1/en unknown
- 1998-06-02 EA EA199901116A patent/EA002384B1/en not_active IP Right Cessation
- 1998-06-02 AU AU82150/98A patent/AU8215098A/en not_active Abandoned
- 1998-06-02 AP APAP/P/1999/001696A patent/AP1214A/en active
- 1998-06-03 DZ DZ980120A patent/DZ2510A1/en active
- 1998-06-04 AR ARP980102649A patent/AR008198A1/en not_active Application Discontinuation
- 1998-06-04 CO CO98031614A patent/CO4940400A1/en unknown
- 1998-06-04 ZA ZA9804826A patent/ZA984826B/en unknown
- 1998-06-04 UY UY25032A patent/UY25032A1/en not_active IP Right Cessation
- 1998-06-04 ZA ZA9811572A patent/ZA9811572B/en unknown
- 1998-06-04 AR ARP980102650A patent/AR015120A1/en not_active Application Discontinuation
- 1998-06-05 PE PE1998000466A patent/PE78899A1/en not_active Application Discontinuation
- 1998-10-23 TW TW087117536A patent/TW570797B/en not_active IP Right Cessation
-
1999
- 1999-12-02 OA OA9900267A patent/OA11306A/en unknown
- 1999-12-03 NO NO995938A patent/NO995938L/en not_active Application Discontinuation
- 1999-12-27 BG BG104048A patent/BG104048A/en unknown
-
2001
- 2001-09-03 NZ NZ513922A patent/NZ513922A/en unknown
-
2002
- 2002-11-05 CN CN02149972A patent/CN1430959A/en active Pending
-
2004
- 2004-02-20 NO NO20040738A patent/NO20040738L/en not_active Application Discontinuation
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
PE78899A1 (en) | COMPOSITION OF 5- [4- [2- (N-METHYL-N- (2-PIRIDIL) AMINO) ETOXI] BENCIL] THIAZOLIDIN-2,4-DIONA | |
EA200601145A1 (en) | TABLET OF SLOW-DIVISION OF INSULIN SENSITIZER AND OTHER ANTI-DIABETIC AGENTS | |
TR200001880T2 (en) | The compound and method of an oral preparation of itraconazole. | |
PE20000550A1 (en) | COMPOSITION OF A BENZIMIDAZOLE DERIVATIVE USEFUL AS ANTI-VIRAL AND ANTI-HIV | |
MA30598B1 (en) | PHARMACEUTICAL COMPOSITION CONTAINING TETRAHYDROFOLIC ACID. | |
AR057970A2 (en) | PHARMACEUTICAL COMPOSITIONS FOR THE TREATMENT OF MELLITUS DIABETES AND CONDITIONS ASSOCIATED WITH MELLITUS DIABETES AND PROCEDURES TO PREPARE SUCH COMPOSITIONS | |
ES2165833T1 (en) | ENTERIC COVERED PHARMACEUTICAL COMPOSITION AND MANUFACTURING PROCEDURE. | |
EP1106210A3 (en) | Combination of aldose reductase inhibitors and antihypertensive agents for the treatment of diabetic complications | |
EA199901100A1 (en) | PHARMACEUTICAL COMPOSITIONS CONTAINING ELETRIPTAN HEMISULPHATE AND CAFFEINE | |
DE69803750T2 (en) | THIAZOLIDINEDIONE AND OXAZOLIDINEDIONE DERIVATIVES WITH ANTIDIABETIC, HYPOLIPIDEMIC AND ANTI-HYPERTENSIVE PROPERTIES | |
JO2239B1 (en) | Process for the preparation of benzothiophene derivatives | |
PE20061373A1 (en) | PHARMACEUTICAL COMPOSITION CONTAINING 'N- (2-CHLORO-6-METHYLPHENIL) -2 - [[6- [4- (2-HYDROXYETHYL) -1-PIPERAZINYL] -2-METHYL-4-PYRIMIDINYL] AMINO] -5- THIAZOLCARBOXAMIDE | |
BR0111868A (en) | Pharmaceutical Compositions | |
ES2188766T3 (en) | PHARMACEUTICAL COMPOSITION CONTAINING LAMOTRIGINE. | |
EA200702648A1 (en) | PHARMACEUTICAL COMPOSITION, SUITABLE FOR INTRODUCTION ONCE A DAY | |
TR200002543T2 (en) | Pharmaceutical compositions containing phospholipase inhibitor sodium [[3- (2-amino-1,2-dioxyethyl-1-phenylmethyl) -2-ethyl-1-phenylmethyl) - 1H-indol-4-yl] oxy] acetate | |
DK0842165T3 (en) | Thiazolidine-4-carboxylic acid derivatives as cytoprotective agents | |
ID27649A (en) | PAPER MAKING PROCESS | |
DE69819742D1 (en) | INDOLDER DERIVATIVES AS 5-HT1B AND 5-HT1D AGONISTS | |
PE61699A1 (en) | PHARMACEUTICAL COMPOSITION OF LAMIVUDINE | |
PE108199A1 (en) | PHARMACEUTICAL COMPOSITION OF TIAZOLIDINDIONA AND SULFONILUREA | |
AR051727A1 (en) | ORAL IMMEDIATE RELEASE FORMULATION OF A LOW SOLUBLE ACTIVE SUBSTANCE IN WATER | |
UY25051A1 (en) | COMPOSITIONS FOR THE TREATMENT OF DIABETES MELLITUS | |
TR200002293T2 (en) | Pharmaceutical compositions. | |
HK1047228A1 (en) | Endoparasiticidal agents |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC | Refusal |