TNSN02003A1 - COMBINATION OF A HISTAMINE H1 RECEPTOR ANTAGONIST AND A SELECTIVE HISTAMINE H4 ANTAGONIST, AND COMPOSITION CONTAINING THE SAME. - Google Patents

COMBINATION OF A HISTAMINE H1 RECEPTOR ANTAGONIST AND A SELECTIVE HISTAMINE H4 ANTAGONIST, AND COMPOSITION CONTAINING THE SAME.

Info

Publication number
TNSN02003A1
TNSN02003A1 TNTNSN02003A TNSN02003A TNSN02003A1 TN SN02003 A1 TNSN02003 A1 TN SN02003A1 TN TNSN02003 A TNTNSN02003 A TN TNSN02003A TN SN02003 A TNSN02003 A TN SN02003A TN SN02003 A1 TNSN02003 A1 TN SN02003A1
Authority
TN
Tunisia
Prior art keywords
histamine
antagonist
combination
composition containing
same
Prior art date
Application number
TNTNSN02003A
Other languages
French (fr)
Inventor
Jenkinson Stephen
Anthony O'reilly Mark
Andrew Trevethick Michael
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of TNSN02003A1 publication Critical patent/TNSN02003A1/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/02Nasal agents, e.g. decongestants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/16Otologicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents

Abstract

L'INVENTION PROPOSE UNE ASSOCIATION (a) D'UN ANTAGONISTE DES RECEPTEURS D'HISTAMINE H1 ET (b) D'UN ANTAGONISTE QUI EST AU MOINS 10 FOIS PLUS SELECTIF POUR LE RECEPTEUR D'HISTAMINE H4 QUE POUR LE RECEPTEUR D'HISTAMINE H3. ELLE CONCERNE EGALEMENT UNE COMPOSITION PHARMACEUTIQUE LA CONTENANT. APPLICATION : UTILISATION DE CETTE ASSOCIATION OU COMPOSITION POUR LE TRAITEMENT DE DIVERSES MALADIES, TELLES QUE LA RHINITE ALLERGIQUE OU L'ASTHME.THE INVENTION PROPOSES A COMBINATION (a) OF AN ANTAGONIST OF HISTAMINE H1 RECEPTORS AND (b) OF AN ANTAGONIST THAT IS AT LEAST 10 TIMES MORE SELECTIVE FOR THE HISTAMINE H4 RECEPTOR THAN FOR THE HISTAMINE H3 RECEPTOR . IT ALSO CONCERNS A PHARMACEUTICAL COMPOSITION CONTAINING IT. APPLICATION: USE OF THIS ASSOCIATION OR COMPOSITION FOR THE TREATMENT OF VARIOUS ILLNESSES, SUCH AS ALLERGIC RHINITIS OR ASTHMA.

TNTNSN02003A 2001-01-17 2002-01-16 COMBINATION OF A HISTAMINE H1 RECEPTOR ANTAGONIST AND A SELECTIVE HISTAMINE H4 ANTAGONIST, AND COMPOSITION CONTAINING THE SAME. TNSN02003A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0101223.6A GB0101223D0 (en) 2001-01-17 2001-01-17 Histamine receptor antagonists

Publications (1)

Publication Number Publication Date
TNSN02003A1 true TNSN02003A1 (en) 2005-12-23

Family

ID=9906993

Family Applications (1)

Application Number Title Priority Date Filing Date
TNTNSN02003A TNSN02003A1 (en) 2001-01-17 2002-01-16 COMBINATION OF A HISTAMINE H1 RECEPTOR ANTAGONIST AND A SELECTIVE HISTAMINE H4 ANTAGONIST, AND COMPOSITION CONTAINING THE SAME.

Country Status (31)

Country Link
EP (1) EP1353657A1 (en)
JP (1) JP2004517883A (en)
KR (1) KR20030069216A (en)
CN (1) CN1486178A (en)
AP (1) AP2002002401A0 (en)
AR (1) AR032101A1 (en)
BG (1) BG107834A (en)
BR (1) BR0206502A (en)
CA (1) CA2435121A1 (en)
CR (1) CR6983A (en)
CZ (1) CZ20031853A3 (en)
DO (1) DOP2002000325A (en)
EA (1) EA200300537A1 (en)
EC (1) ECSP034692A (en)
EE (1) EE200300335A (en)
GB (1) GB0101223D0 (en)
GT (1) GT200200003A (en)
HU (1) HUP0302767A2 (en)
IL (1) IL156087A0 (en)
IS (1) IS6818A (en)
MA (1) MA26980A1 (en)
MX (1) MXPA03006408A (en)
NO (1) NO20033223L (en)
OA (1) OA12440A (en)
PA (1) PA8537101A1 (en)
PL (1) PL362793A1 (en)
SK (1) SK8572003A3 (en)
SV (1) SV2003000849A (en)
TN (1) TNSN02003A1 (en)
WO (1) WO2002056871A2 (en)
ZA (1) ZA200304180B (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20030133931A1 (en) * 2001-12-21 2003-07-17 Robin Thurmond Use of histamine H4 receptor antagonist for the treatment of inflammatory responses
CA2497788A1 (en) * 2002-09-06 2004-03-18 Janssen Pharmaceutica, N.V. Use of histamine h4 receptor modulators for the treatment of allergy and asthma
WO2004066960A2 (en) * 2003-01-28 2004-08-12 Schering Corporation Combination of h1, h3 and h4 receptor antagonists for treatment of allergic and non-allergic pulmonary inflammation, congestion and allergic rhinitis
US8236786B2 (en) 2008-08-07 2012-08-07 Pulmagen Therapeutics (Inflammation) Limited Respiratory disease treatment
WO2013151982A1 (en) 2012-04-03 2013-10-10 Arena Pharmaceuticals, Inc. Methods and compounds useful in treating pruritus, and methods for identifying such compounds
EP2858647B1 (en) 2012-06-08 2018-05-23 Sensorion H4 receptor inhibitors for treating tinnitus

Also Published As

Publication number Publication date
SK8572003A3 (en) 2004-07-07
EP1353657A1 (en) 2003-10-22
DOP2002000325A (en) 2003-01-31
MXPA03006408A (en) 2003-10-15
KR20030069216A (en) 2003-08-25
MA26980A1 (en) 2004-12-20
CR6983A (en) 2003-11-25
PA8537101A1 (en) 2002-08-29
ZA200304180B (en) 2004-06-15
IL156087A0 (en) 2003-12-23
SV2003000849A (en) 2003-01-13
JP2004517883A (en) 2004-06-17
IS6818A (en) 2003-05-15
GB0101223D0 (en) 2001-02-28
AP2002002401A0 (en) 2002-03-31
AR032101A1 (en) 2003-10-22
GT200200003A (en) 2002-08-19
PL362793A1 (en) 2004-11-02
NO20033223D0 (en) 2003-07-16
NO20033223L (en) 2003-07-16
CN1486178A (en) 2004-03-31
BR0206502A (en) 2003-10-21
CZ20031853A3 (en) 2004-07-14
WO2002056871A2 (en) 2002-07-25
EA200300537A1 (en) 2004-02-26
ECSP034692A (en) 2003-08-29
BG107834A (en) 2004-01-30
EE200300335A (en) 2003-12-15
CA2435121A1 (en) 2002-07-25
HUP0302767A2 (en) 2003-11-28
OA12440A (en) 2006-05-22

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