BR0206502A - Histamine Receptor Antagonists - Google Patents
Histamine Receptor AntagonistsInfo
- Publication number
- BR0206502A BR0206502A BR0206502-9A BR0206502A BR0206502A BR 0206502 A BR0206502 A BR 0206502A BR 0206502 A BR0206502 A BR 0206502A BR 0206502 A BR0206502 A BR 0206502A
- Authority
- BR
- Brazil
- Prior art keywords
- histamine
- receptor antagonists
- receptor
- histamine receptor
- antagonist
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pulmonology (AREA)
- Epidemiology (AREA)
- Immunology (AREA)
- Otolaryngology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
"ANTAGONISTAS DO RECEPTOR DE HISTAMINA". A presente invenção fornece uma combinação de (a) um antagonista do receptor de histamina H, e (b) um antagonista que é pelo menos dez vezes mais seletivo para o receptor de histamina H~ 4~ quando comparado com o receptor de histamina H~ 3~ e um antagonista que é pelo menos dez vezes mais seletivo para o receptor de histamina H~ 4~ quando comparado com o receptor de histamina H~ 3~, e suas composições."HISTAMIN RECEPTOR ANTAGONISTS". The present invention provides a combination of (a) a histamine H receptor antagonist, and (b) an antagonist that is at least ten times more selective for the histamine H 4 -receptor compared to the histamine H-4receptor. 3? Is an antagonist that is at least ten times more selective for the H? 4? Histamine receptor as compared to the H? 3? Histamine receptor, and compositions thereof.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0101223.6A GB0101223D0 (en) | 2001-01-17 | 2001-01-17 | Histamine receptor antagonists |
| PCT/IB2002/000042 WO2002056871A2 (en) | 2001-01-17 | 2002-01-10 | Histamine receptor antagonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR0206502A true BR0206502A (en) | 2003-10-21 |
Family
ID=9906993
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0206502-9A BR0206502A (en) | 2001-01-17 | 2002-01-10 | Histamine Receptor Antagonists |
Country Status (31)
| Country | Link |
|---|---|
| EP (1) | EP1353657A1 (en) |
| JP (1) | JP2004517883A (en) |
| KR (1) | KR20030069216A (en) |
| CN (1) | CN1486178A (en) |
| AP (1) | AP2002002401A0 (en) |
| AR (1) | AR032101A1 (en) |
| BG (1) | BG107834A (en) |
| BR (1) | BR0206502A (en) |
| CA (1) | CA2435121A1 (en) |
| CR (1) | CR6983A (en) |
| CZ (1) | CZ20031853A3 (en) |
| DO (1) | DOP2002000325A (en) |
| EA (1) | EA200300537A1 (en) |
| EC (1) | ECSP034692A (en) |
| EE (1) | EE200300335A (en) |
| GB (1) | GB0101223D0 (en) |
| GT (1) | GT200200003A (en) |
| HU (1) | HUP0302767A2 (en) |
| IL (1) | IL156087A0 (en) |
| IS (1) | IS6818A (en) |
| MA (1) | MA26980A1 (en) |
| MX (1) | MXPA03006408A (en) |
| NO (1) | NO20033223L (en) |
| OA (1) | OA12440A (en) |
| PA (1) | PA8537101A1 (en) |
| PL (1) | PL362793A1 (en) |
| SK (1) | SK8572003A3 (en) |
| SV (1) | SV2003000849A (en) |
| TN (1) | TNSN02003A1 (en) |
| WO (1) | WO2002056871A2 (en) |
| ZA (1) | ZA200304180B (en) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20030133931A1 (en) * | 2001-12-21 | 2003-07-17 | Robin Thurmond | Use of histamine H4 receptor antagonist for the treatment of inflammatory responses |
| WO2004021999A2 (en) * | 2002-09-06 | 2004-03-18 | Janssen Pharmaceutica, N.V. | Use of histamine h4 receptor modulators for the treatment of allergy and asthma |
| US20050090527A1 (en) * | 2003-01-28 | 2005-04-28 | Schering Corporation | Combination of H1, H3 and H4 receptor antagonists for treatment of allergic and non-allergic pulmonary inflammation, congestion and allergic rhinitis |
| US8236786B2 (en) * | 2008-08-07 | 2012-08-07 | Pulmagen Therapeutics (Inflammation) Limited | Respiratory disease treatment |
| WO2013151982A1 (en) | 2012-04-03 | 2013-10-10 | Arena Pharmaceuticals, Inc. | Methods and compounds useful in treating pruritus, and methods for identifying such compounds |
| EP3378476A1 (en) | 2012-06-08 | 2018-09-26 | Sensorion | H4 receptor inhibitors for treating tinnitus |
-
2001
- 2001-01-17 GB GBGB0101223.6A patent/GB0101223D0/en not_active Ceased
-
2002
- 2002-01-10 OA OA1200300174A patent/OA12440A/en unknown
- 2002-01-10 SK SK857-2003A patent/SK8572003A3/en unknown
- 2002-01-10 EE EEP200300335A patent/EE200300335A/en unknown
- 2002-01-10 CN CNA028036840A patent/CN1486178A/en active Pending
- 2002-01-10 IL IL15608702A patent/IL156087A0/en unknown
- 2002-01-10 MX MXPA03006408A patent/MXPA03006408A/en unknown
- 2002-01-10 PL PL02362793A patent/PL362793A1/en not_active Application Discontinuation
- 2002-01-10 EA EA200300537A patent/EA200300537A1/en unknown
- 2002-01-10 CZ CZ20031853A patent/CZ20031853A3/en unknown
- 2002-01-10 BR BR0206502-9A patent/BR0206502A/en not_active IP Right Cessation
- 2002-01-10 WO PCT/IB2002/000042 patent/WO2002056871A2/en not_active Application Discontinuation
- 2002-01-10 CA CA002435121A patent/CA2435121A1/en not_active Abandoned
- 2002-01-10 EP EP02732099A patent/EP1353657A1/en not_active Withdrawn
- 2002-01-10 HU HU0302767A patent/HUP0302767A2/en unknown
- 2002-01-10 KR KR10-2003-7009493A patent/KR20030069216A/en not_active Application Discontinuation
- 2002-01-10 JP JP2002557379A patent/JP2004517883A/en not_active Withdrawn
- 2002-01-11 DO DO2002000325A patent/DOP2002000325A/en unknown
- 2002-01-14 PA PA20028537101A patent/PA8537101A1/en unknown
- 2002-01-16 TN TNTNSN02003A patent/TNSN02003A1/en unknown
- 2002-01-16 SV SV2002000849A patent/SV2003000849A/en not_active Application Discontinuation
- 2002-01-16 AR ARP020100145A patent/AR032101A1/en not_active Application Discontinuation
- 2002-01-16 GT GT200200003A patent/GT200200003A/en unknown
- 2002-01-17 AP APAP/P/2002/002401A patent/AP2002002401A0/en unknown
-
2003
- 2003-05-15 IS IS6818A patent/IS6818A/en unknown
- 2003-05-21 BG BG107834A patent/BG107834A/en unknown
- 2003-05-22 CR CR6983A patent/CR6983A/en not_active Application Discontinuation
- 2003-05-29 ZA ZA200304180A patent/ZA200304180B/en unknown
- 2003-07-11 MA MA27233A patent/MA26980A1/en unknown
- 2003-07-16 NO NO20033223A patent/NO20033223L/en not_active Application Discontinuation
- 2003-07-17 EC EC2003004692A patent/ECSP034692A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| SV2003000849A (en) | 2003-01-13 |
| NO20033223D0 (en) | 2003-07-16 |
| TNSN02003A1 (en) | 2005-12-23 |
| PL362793A1 (en) | 2004-11-02 |
| HUP0302767A2 (en) | 2003-11-28 |
| OA12440A (en) | 2006-05-22 |
| EA200300537A1 (en) | 2004-02-26 |
| EP1353657A1 (en) | 2003-10-22 |
| ECSP034692A (en) | 2003-08-29 |
| EE200300335A (en) | 2003-12-15 |
| GB0101223D0 (en) | 2001-02-28 |
| MXPA03006408A (en) | 2003-10-15 |
| PA8537101A1 (en) | 2002-08-29 |
| CR6983A (en) | 2003-11-25 |
| ZA200304180B (en) | 2004-06-15 |
| CN1486178A (en) | 2004-03-31 |
| JP2004517883A (en) | 2004-06-17 |
| NO20033223L (en) | 2003-07-16 |
| IL156087A0 (en) | 2003-12-23 |
| BG107834A (en) | 2004-01-30 |
| GT200200003A (en) | 2002-08-19 |
| CA2435121A1 (en) | 2002-07-25 |
| AP2002002401A0 (en) | 2002-03-31 |
| IS6818A (en) | 2003-05-15 |
| KR20030069216A (en) | 2003-08-25 |
| AR032101A1 (en) | 2003-10-22 |
| SK8572003A3 (en) | 2004-07-07 |
| CZ20031853A3 (en) | 2004-07-14 |
| DOP2002000325A (en) | 2003-01-31 |
| WO2002056871A2 (en) | 2002-07-25 |
| MA26980A1 (en) | 2004-12-20 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 5A,6A,7A E 8A ANUIDADES. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 DA RPI 2025 DE 27/10/2009. |