CR6983A - HISTAMINE RECEIVER ANTAGONISTS - Google Patents
HISTAMINE RECEIVER ANTAGONISTSInfo
- Publication number
- CR6983A CR6983A CR6983A CR6983A CR6983A CR 6983 A CR6983 A CR 6983A CR 6983 A CR6983 A CR 6983A CR 6983 A CR6983 A CR 6983A CR 6983 A CR6983 A CR 6983A
- Authority
- CR
- Costa Rica
- Prior art keywords
- histamine
- receiver
- histamine receiver
- receiver antagonists
- antagonists
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pulmonology (AREA)
- Epidemiology (AREA)
- Immunology (AREA)
- Otolaryngology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
LA PRESENTE INVENCION PROPORCIONA UNA COMBINACION DE (A) UN ANTAGONISTA DE RECEPTOR H1 DE HISTAMINA Y (B) UN ANTAGONISTA QUE ES AL MENOS 10 VECES MAS SELECTIVO PARA EL RECEPTOR H4 DE HISTAMINA EN COMPARACION CON EL RECEPTOR H3 DE HISTAMINA, Y UN ANTAGONISTA QUE ES AL MENOS 10 VECES MAS SELECTIVO PARA EL RECEPTOR H4 DE HISTAMINA EN COMPARACION CON EL RECEPTOR H3 DE HISTAMINA Y SUS COMPOSICIONES Y USOS.THIS INVENTION PROVIDES A COMBINATION OF (A) AN HISTAMINE RECEIVER ANTAGONIST AND (B) AN ANTAGONIST THAT IS AT LEAST 10 TIMES MORE SELECTIVE FOR HISTAMINE RECEIVER H4, COMPARED TO HISTAMINE RECEIVER, AND AN ANTAGON IT IS AT LEAST 10 TIMES MORE SELECTIVE FOR THE H4 HISTAMINE RECEIVER COMPARED TO THE HISTAMINE H3 RECEIVER AND ITS COMPOSITIONS AND USES.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0101223.6A GB0101223D0 (en) | 2001-01-17 | 2001-01-17 | Histamine receptor antagonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CR6983A true CR6983A (en) | 2003-11-25 |
Family
ID=9906993
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CR6983A CR6983A (en) | 2001-01-17 | 2003-05-22 | HISTAMINE RECEIVER ANTAGONISTS |
Country Status (31)
| Country | Link |
|---|---|
| EP (1) | EP1353657A1 (en) |
| JP (1) | JP2004517883A (en) |
| KR (1) | KR20030069216A (en) |
| CN (1) | CN1486178A (en) |
| AP (1) | AP2002002401A0 (en) |
| AR (1) | AR032101A1 (en) |
| BG (1) | BG107834A (en) |
| BR (1) | BR0206502A (en) |
| CA (1) | CA2435121A1 (en) |
| CR (1) | CR6983A (en) |
| CZ (1) | CZ20031853A3 (en) |
| DO (1) | DOP2002000325A (en) |
| EA (1) | EA200300537A1 (en) |
| EC (1) | ECSP034692A (en) |
| EE (1) | EE200300335A (en) |
| GB (1) | GB0101223D0 (en) |
| GT (1) | GT200200003A (en) |
| HU (1) | HUP0302767A2 (en) |
| IL (1) | IL156087A0 (en) |
| IS (1) | IS6818A (en) |
| MA (1) | MA26980A1 (en) |
| MX (1) | MXPA03006408A (en) |
| NO (1) | NO20033223L (en) |
| OA (1) | OA12440A (en) |
| PA (1) | PA8537101A1 (en) |
| PL (1) | PL362793A1 (en) |
| SK (1) | SK8572003A3 (en) |
| SV (1) | SV2003000849A (en) |
| TN (1) | TNSN02003A1 (en) |
| WO (1) | WO2002056871A2 (en) |
| ZA (1) | ZA200304180B (en) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20030133931A1 (en) * | 2001-12-21 | 2003-07-17 | Robin Thurmond | Use of histamine H4 receptor antagonist for the treatment of inflammatory responses |
| WO2004021999A2 (en) * | 2002-09-06 | 2004-03-18 | Janssen Pharmaceutica, N.V. | Use of histamine h4 receptor modulators for the treatment of allergy and asthma |
| US20050090527A1 (en) * | 2003-01-28 | 2005-04-28 | Schering Corporation | Combination of H1, H3 and H4 receptor antagonists for treatment of allergic and non-allergic pulmonary inflammation, congestion and allergic rhinitis |
| US8236786B2 (en) * | 2008-08-07 | 2012-08-07 | Pulmagen Therapeutics (Inflammation) Limited | Respiratory disease treatment |
| WO2013151982A1 (en) | 2012-04-03 | 2013-10-10 | Arena Pharmaceuticals, Inc. | Methods and compounds useful in treating pruritus, and methods for identifying such compounds |
| EP3378476A1 (en) | 2012-06-08 | 2018-09-26 | Sensorion | H4 receptor inhibitors for treating tinnitus |
-
2001
- 2001-01-17 GB GBGB0101223.6A patent/GB0101223D0/en not_active Ceased
-
2002
- 2002-01-10 OA OA1200300174A patent/OA12440A/en unknown
- 2002-01-10 SK SK857-2003A patent/SK8572003A3/en unknown
- 2002-01-10 EE EEP200300335A patent/EE200300335A/en unknown
- 2002-01-10 CN CNA028036840A patent/CN1486178A/en active Pending
- 2002-01-10 IL IL15608702A patent/IL156087A0/en unknown
- 2002-01-10 MX MXPA03006408A patent/MXPA03006408A/en unknown
- 2002-01-10 PL PL02362793A patent/PL362793A1/en not_active Application Discontinuation
- 2002-01-10 EA EA200300537A patent/EA200300537A1/en unknown
- 2002-01-10 CZ CZ20031853A patent/CZ20031853A3/en unknown
- 2002-01-10 BR BR0206502-9A patent/BR0206502A/en not_active IP Right Cessation
- 2002-01-10 WO PCT/IB2002/000042 patent/WO2002056871A2/en not_active Application Discontinuation
- 2002-01-10 CA CA002435121A patent/CA2435121A1/en not_active Abandoned
- 2002-01-10 EP EP02732099A patent/EP1353657A1/en not_active Withdrawn
- 2002-01-10 HU HU0302767A patent/HUP0302767A2/en unknown
- 2002-01-10 KR KR10-2003-7009493A patent/KR20030069216A/en not_active Application Discontinuation
- 2002-01-10 JP JP2002557379A patent/JP2004517883A/en not_active Withdrawn
- 2002-01-11 DO DO2002000325A patent/DOP2002000325A/en unknown
- 2002-01-14 PA PA20028537101A patent/PA8537101A1/en unknown
- 2002-01-16 TN TNTNSN02003A patent/TNSN02003A1/en unknown
- 2002-01-16 SV SV2002000849A patent/SV2003000849A/en not_active Application Discontinuation
- 2002-01-16 AR ARP020100145A patent/AR032101A1/en not_active Application Discontinuation
- 2002-01-16 GT GT200200003A patent/GT200200003A/en unknown
- 2002-01-17 AP APAP/P/2002/002401A patent/AP2002002401A0/en unknown
-
2003
- 2003-05-15 IS IS6818A patent/IS6818A/en unknown
- 2003-05-21 BG BG107834A patent/BG107834A/en unknown
- 2003-05-22 CR CR6983A patent/CR6983A/en not_active Application Discontinuation
- 2003-05-29 ZA ZA200304180A patent/ZA200304180B/en unknown
- 2003-07-11 MA MA27233A patent/MA26980A1/en unknown
- 2003-07-16 NO NO20033223A patent/NO20033223L/en not_active Application Discontinuation
- 2003-07-17 EC EC2003004692A patent/ECSP034692A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| BR0206502A (en) | 2003-10-21 |
| SV2003000849A (en) | 2003-01-13 |
| NO20033223D0 (en) | 2003-07-16 |
| TNSN02003A1 (en) | 2005-12-23 |
| PL362793A1 (en) | 2004-11-02 |
| HUP0302767A2 (en) | 2003-11-28 |
| OA12440A (en) | 2006-05-22 |
| EA200300537A1 (en) | 2004-02-26 |
| EP1353657A1 (en) | 2003-10-22 |
| ECSP034692A (en) | 2003-08-29 |
| EE200300335A (en) | 2003-12-15 |
| GB0101223D0 (en) | 2001-02-28 |
| MXPA03006408A (en) | 2003-10-15 |
| PA8537101A1 (en) | 2002-08-29 |
| ZA200304180B (en) | 2004-06-15 |
| CN1486178A (en) | 2004-03-31 |
| JP2004517883A (en) | 2004-06-17 |
| NO20033223L (en) | 2003-07-16 |
| IL156087A0 (en) | 2003-12-23 |
| BG107834A (en) | 2004-01-30 |
| GT200200003A (en) | 2002-08-19 |
| CA2435121A1 (en) | 2002-07-25 |
| AP2002002401A0 (en) | 2002-03-31 |
| IS6818A (en) | 2003-05-15 |
| KR20030069216A (en) | 2003-08-25 |
| AR032101A1 (en) | 2003-10-22 |
| SK8572003A3 (en) | 2004-07-07 |
| CZ20031853A3 (en) | 2004-07-14 |
| DOP2002000325A (en) | 2003-01-31 |
| WO2002056871A2 (en) | 2002-07-25 |
| MA26980A1 (en) | 2004-12-20 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal (granting procedure) |