TN2012000147A1 - 2-oxo-1-pyrrolidinyl imidazothiadiazole derivatives - Google Patents

2-oxo-1-pyrrolidinyl imidazothiadiazole derivatives

Info

Publication number
TN2012000147A1
TN2012000147A1 TNP2012000147A TN2012000147A TN2012000147A1 TN 2012000147 A1 TN2012000147 A1 TN 2012000147A1 TN P2012000147 A TNP2012000147 A TN P2012000147A TN 2012000147 A TN2012000147 A TN 2012000147A TN 2012000147 A1 TN2012000147 A1 TN 2012000147A1
Authority
TN
Tunisia
Prior art keywords
oxo
imidazothiadiazole derivatives
pyrrolidinyl
derivatives
pyrrolidinyl imidazothiadiazole
Prior art date
Application number
TNP2012000147A
Other languages
English (en)
Inventor
Yannick Quesnel
Laurent Turet
Jo? Mercier
Original Assignee
Ucb Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42034570&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TN2012000147(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ucb Pharma Sa filed Critical Ucb Pharma Sa
Publication of TN2012000147A1 publication Critical patent/TN2012000147A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/433Thidiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
TNP2012000147A 2009-10-23 2012-03-29 2-oxo-1-pyrrolidinyl imidazothiadiazole derivatives TN2012000147A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP09173912 2009-10-23
PCT/EP2010/006434 WO2011047860A1 (en) 2009-10-23 2010-10-21 2-oxo-1-pyrrolidinyl imidazothiadiazole derivatives

Publications (1)

Publication Number Publication Date
TN2012000147A1 true TN2012000147A1 (en) 2013-09-19

Family

ID=42034570

Family Applications (1)

Application Number Title Priority Date Filing Date
TNP2012000147A TN2012000147A1 (en) 2009-10-23 2012-03-29 2-oxo-1-pyrrolidinyl imidazothiadiazole derivatives

Country Status (30)

Country Link
US (1) US8822508B2 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
EP (1) EP2491045B1 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
JP (1) JP5808020B2 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
KR (1) KR20120102058A (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
CN (1) CN102574869A (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
AR (1) AR078722A1 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
AU (1) AU2010310100B2 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
BR (1) BR112012009310B8 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
CA (1) CA2778194C (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
CL (1) CL2012001031A1 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
CY (1) CY1117288T1 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
DK (1) DK2491045T3 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
EA (1) EA201200616A1 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
ES (1) ES2565515T3 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
HR (1) HRP20160263T1 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
HU (1) HUE028668T2 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
IL (1) IL218696A0 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
IN (1) IN2012DN02793A (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
MA (1) MA33679B1 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
ME (1) ME02355B (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
MX (1) MX347070B (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
PE (1) PE20121562A1 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
PH (1) PH12012500570A1 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
PL (1) PL2491045T3 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
RS (1) RS54595B1 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
SI (1) SI2491045T1 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
SM (1) SMT201600076B (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
TN (1) TN2012000147A1 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
TW (1) TW201118103A (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)
WO (1) WO2011047860A1 (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2699581B1 (en) * 2011-04-18 2015-11-25 UCB Biopharma SPRL 2-oxo-1-imidazolidinyl imidazothiadiazole derivatives
US9581654B2 (en) 2013-02-12 2017-02-28 Johnson Controls Technology Company Vehicle battery monitoring system
SI3096790T1 (sl) 2014-01-21 2019-11-29 Janssen Pharmaceutica Nv Kombinacije, ki vsebujejo pozitivne aleostrične modulatorje ali ortosterične agoniste metabotropnega glutamatergičnega receptorja podtipa 2 in njihova uporaba
DK3096790T3 (da) 2014-01-21 2019-10-07 Janssen Pharmaceutica Nv Kombinationer omfattende positive allosteriske modulatorer eller orthosteriske agonister af metabotrop glutamaterg subtype 2-receptor og anvendelse af disse
US11155565B2 (en) 2017-07-10 2021-10-26 UCB Biopharma SRL 2-oxo-1,3-oxazolidinyl imidazothiadiazole derivatives
CA3069172A1 (en) 2017-07-10 2019-01-17 UCB Biopharma SRL 2-oxo-1-imidazolidinyl imidazothiadiazole derivatives
CN107827870B (zh) * 2017-10-24 2019-11-08 江苏仁明生物科技有限公司 一种正电子药物[18f]fpmmp及其制备方法与中间体
WO2019115292A1 (en) 2017-12-12 2019-06-20 Ucb Biopharma Sprl 2-oxo-1-pyrrolidinyl imidazothiadiazole derivatives
WO2019215062A1 (en) 2018-05-08 2019-11-14 Ucb Biopharma Sprl 1-imidazothiadiazolo-2h-pyrrol-5-one derivatives
CN113549052B (zh) * 2021-07-09 2022-09-02 首都医科大学脑重大疾病研究中心(北京脑重大疾病研究院) 4-苯基-1-(吡啶-4-基甲基)吡咯烷-2-酮衍生物及其制备方法和应用
WO2025132331A1 (en) 2023-12-21 2025-06-26 UCB Biopharma SRL Compounds for treatment of a hyperkinetic movement disorder
CN119606962B (zh) * 2025-02-17 2025-05-02 中国人民解放军总医院第三医学中心 padsevonil在制备治疗TFE3重排性肾细胞癌的药物中的应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8412358D0 (en) 1984-05-15 1984-06-20 Ucb Sa Pharmaceutical composition
GB8412357D0 (en) 1984-05-15 1984-06-20 Ucb Sa Pharmaceutical composition
GB0004297D0 (en) * 2000-02-23 2000-04-12 Ucb Sa 2-oxo-1 pyrrolidine derivatives process for preparing them and their uses
EP2050736A1 (en) 2003-12-02 2009-04-22 UCB Pharma, S.A. Imidazole derivatives, processes for preparing them and their uses
CA2610695A1 (en) * 2005-06-01 2006-12-07 Ucb Pharma, S.A. 2-oxo-1-pyrrolidine derivatives and their therapeutic use on the central nervous system

Also Published As

Publication number Publication date
CA2778194A1 (en) 2011-04-28
US20120245208A1 (en) 2012-09-27
IL218696A0 (en) 2012-05-31
EA201200616A1 (ru) 2012-12-28
PH12012500570A1 (en) 2012-10-22
MA33679B1 (fr) 2012-10-01
ME02355B (me) 2016-06-20
AU2010310100A1 (en) 2012-05-17
TW201118103A (en) 2011-06-01
EP2491045A1 (en) 2012-08-29
EP2491045B1 (en) 2015-12-23
SI2491045T1 (sl) 2016-04-29
AR078722A1 (es) 2011-11-30
BR112012009310B8 (pt) 2021-05-25
SMT201600076B (it) 2016-04-29
ES2565515T3 (es) 2016-04-05
BR112012009310B1 (pt) 2021-01-12
KR20120102058A (ko) 2012-09-17
CY1117288T1 (el) 2017-04-26
WO2011047860A1 (en) 2011-04-28
US8822508B2 (en) 2014-09-02
BR112012009310A2 (pt) 2016-06-07
PE20121562A1 (es) 2012-11-30
IN2012DN02793A (c_deeref_Disk_and_Scratch_Disk_Pools_and_Their_Defaults.html) 2015-07-24
MX2012003839A (es) 2012-05-08
JP2013508321A (ja) 2013-03-07
PL2491045T3 (pl) 2016-06-30
CN102574869A (zh) 2012-07-11
HUE028668T2 (en) 2016-12-28
CL2012001031A1 (es) 2012-09-14
DK2491045T3 (en) 2016-03-14
HRP20160263T1 (hr) 2016-04-08
CA2778194C (en) 2016-07-12
AU2010310100B2 (en) 2015-09-10
JP5808020B2 (ja) 2015-11-10
MX347070B (es) 2017-04-11
RS54595B1 (en) 2016-08-31

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