TH94288B - 1,1-dioxo-thymorpholinyl indoleyl methanone derivatives - Google Patents
1,1-dioxo-thymorpholinyl indoleyl methanone derivativesInfo
- Publication number
- TH94288B TH94288B TH601005925A TH0601005925A TH94288B TH 94288 B TH94288 B TH 94288B TH 601005925 A TH601005925 A TH 601005925A TH 0601005925 A TH0601005925 A TH 0601005925A TH 94288 B TH94288 B TH 94288B
- Authority
- TH
- Thailand
- Prior art keywords
- alkyl
- thymorpholinyl
- indoleyl
- dioxo
- methanone derivatives
- Prior art date
Links
- SBNOTUDDIXOFSN-UHFFFAOYSA-N 1H-indole-2-carbaldehyde Chemical class C1=CC=C2NC(C=O)=CC2=C1 SBNOTUDDIXOFSN-UHFFFAOYSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 claims abstract 3
- 239000000126 substance Substances 0.000 claims abstract 2
- 125000004183 alkoxy alkyl group Chemical group 0.000 claims 1
- 125000000217 alkyl group Chemical group 0.000 claims 1
- 125000004390 alkyl sulfonyl group Chemical group 0.000 claims 1
- 125000002915 carbonyl group Chemical group [*:2]C([*:1])=O 0.000 claims 1
- 125000004966 cyanoalkyl group Chemical group 0.000 claims 1
- 125000001316 cycloalkyl alkyl group Chemical group 0.000 claims 1
- 125000001188 haloalkyl group Chemical group 0.000 claims 1
- 229910052739 hydrogen Inorganic materials 0.000 claims 1
- 239000001257 hydrogen Substances 0.000 claims 1
- 125000004435 hydrogen atoms Chemical class [H]* 0.000 claims 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 1
- 201000010099 disease Diseases 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000011780 sodium chloride Substances 0.000 abstract 1
Abstract
การประดิษฐ์นี้จะเกี่ยวข้องกับสารประกอบที่สูตร I (สูตรเคมี) I ที่ซึ่ง R1 , R2 และ G คือ ดังที่ถูกนิยามในการบรรยาย และข้อถือสิทธิ และเกลือของสิ่งเหล่านี้ ที่ยอมรับได้ทางเภสัชกรรม สารประกอบจะเป็นประโยชน์สำหรับการบำบัดรักษา และ/หรือ การป้องกันของโรค ซึ่งเกี่ยวเนื่องกับการปรับของ H3 รีเซพเตอร์ This invention involves compounds with formula I (chemical formula) I, where R1, R2 and G are, as defined in the description. And the claim And the salt of these Acceptable pharmaceutical Compounds are useful for treatment and / or prevention of disease. Which is related to the adjustment of the H3 receptor
Claims (1)
Publications (2)
| Publication Number | Publication Date |
|---|---|
| TH94288A TH94288A (en) | 2009-03-13 |
| TH94288B true TH94288B (en) | 2009-03-13 |
Family
ID=
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