TH107679B - Indole derivatives - Google Patents
Indole derivativesInfo
- Publication number
- TH107679B TH107679B TH501002826A TH0501002826A TH107679B TH 107679 B TH107679 B TH 107679B TH 501002826 A TH501002826 A TH 501002826A TH 0501002826 A TH0501002826 A TH 0501002826A TH 107679 B TH107679 B TH 107679B
- Authority
- TH
- Thailand
- Prior art keywords
- alkyl
- indole derivatives
- lower molecular
- compound
- mass
- Prior art date
Links
- 229940054051 antipsychotic Indole derivatives Drugs 0.000 title 1
- 150000002475 indoles Chemical class 0.000 title 1
- 150000001875 compounds Chemical class 0.000 claims abstract 4
- 239000000126 substance Substances 0.000 claims abstract 2
- 125000000217 alkyl group Chemical group 0.000 claims 3
- 125000001316 cycloalkyl alkyl group Chemical group 0.000 claims 1
- 125000000753 cycloalkyl group Chemical group 0.000 claims 1
- 229910052739 hydrogen Inorganic materials 0.000 claims 1
- 239000001257 hydrogen Substances 0.000 claims 1
- 125000004435 hydrogen atoms Chemical group [H]* 0.000 claims 1
- 125000002768 hydroxyalkyl group Chemical group 0.000 claims 1
- 102000004384 Histamine H3 Receptors Human genes 0.000 abstract 1
- 108090000981 Histamine H3 Receptors Proteins 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000011780 sodium chloride Substances 0.000 abstract 1
Abstract
การประดิษฐ์นี้เกี่ยวข้องกับสารประกอบของสูตร I (สูตรเคมี) I โดยที่ X, R2, R2, R3, R4 และ R5 คือตามที่ถูกนิยามในการอธิบายและข้อถือสิทธิ, และ เกลือที่สามารถยอมรับได้ทางเภสัชกรรมของสิ่งเหล่านี้, เพื่อเตรียมของสารประกอบดังกล่าวและ สารผสมทางเภสัชกรรมที่มีสิ่งเหล่านี้ สารประกอบเป็นประโยชน์สำหรับการทรีทเมนท์และ/หรือการ ป้องกันของโรคซึ่งเกี่ยวข้องกับการควบคุมของ H3 รีเซพเตอร์ This invention involves compounds of formula I (chemical formula) I, where X, R2, R2, R3, R4 and R5 are, as defined in the description and claim, and the pharmacologically acceptable salts of them. This, to prepare the compound and Pharmaceutical mixtures that contain these The compound is useful for treatment and / or Prevention of disease, which is related to the control of H3 receptors.
Claims (1)
Publications (2)
Publication Number | Publication Date |
---|---|
TH107679A TH107679A (en) | 2011-05-12 |
TH107679B true TH107679B (en) | 2011-05-12 |
Family
ID=
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