SK284286B6 - Farmaceutický prostriedok, obsahujúci lamivudín a zidovudín, spôsob jeho výroby a jeho použitie - Google Patents

Farmaceutický prostriedok, obsahujúci lamivudín a zidovudín, spôsob jeho výroby a jeho použitie Download PDF

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Publication number
SK284286B6
SK284286B6 SK575-99A SK57599A SK284286B6 SK 284286 B6 SK284286 B6 SK 284286B6 SK 57599 A SK57599 A SK 57599A SK 284286 B6 SK284286 B6 SK 284286B6
Authority
SK
Slovakia
Prior art keywords
pharmaceutically acceptable
lamivudine
pharmaceutical composition
zidovudine
acceptable derivative
Prior art date
Application number
SK575-99A
Other languages
English (en)
Slovak (sk)
Other versions
SK57599A3 (en
Inventor
Gary Wayne Goodson
Allen Wayne Wood
Katherine Jeannette Ford
Original Assignee
Glaxo Group Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Limited filed Critical Glaxo Group Limited
Publication of SK57599A3 publication Critical patent/SK57599A3/sk
Publication of SK284286B6 publication Critical patent/SK284286B6/sk

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A61K31/7064Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
    • A61K31/7068Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A61K31/7064Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
    • A61K31/7068Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid
    • A61K31/7072Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid having two oxo groups directly attached to the pyrimidine ring, e.g. uridine, uridylic acid, thymidine, zidovudine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/20Antivirals for DNA viruses
    • A61P31/22Antivirals for DNA viruses for herpes viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
SK575-99A 1996-10-31 1997-10-29 Farmaceutický prostriedok, obsahujúci lamivudín a zidovudín, spôsob jeho výroby a jeho použitie SK284286B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9622681.6A GB9622681D0 (en) 1996-10-31 1996-10-31 Pharmaceutical compositions
PCT/EP1997/005953 WO1998018477A2 (en) 1996-10-31 1997-10-29 Pharmaceutical compositions containing lamivudine and zidovudine

Publications (2)

Publication Number Publication Date
SK57599A3 SK57599A3 (en) 2000-06-12
SK284286B6 true SK284286B6 (sk) 2005-01-03

Family

ID=10802224

Family Applications (1)

Application Number Title Priority Date Filing Date
SK575-99A SK284286B6 (sk) 1996-10-31 1997-10-29 Farmaceutický prostriedok, obsahujúci lamivudín a zidovudín, spôsob jeho výroby a jeho použitie

Country Status (44)

Country Link
EP (1) EP0941100B1 (id)
JP (1) JP2001502718A (id)
KR (1) KR100551652B1 (id)
AP (1) AP1067A (id)
AR (1) AR009135A1 (id)
AT (1) ATE241364T1 (id)
AU (1) AU736607B2 (id)
BG (1) BG64541B1 (id)
BR (1) BR9712614A (id)
CA (1) CA2270174A1 (id)
CO (1) CO4930269A1 (id)
CY (1) CY2485B1 (id)
CZ (1) CZ296080B6 (id)
DE (1) DE69722433T2 (id)
DK (1) DK0941100T3 (id)
EA (1) EA002437B1 (id)
EE (1) EE03806B1 (id)
ES (1) ES2200204T3 (id)
GB (1) GB9622681D0 (id)
GE (1) GEP20022735B (id)
GT (1) GT199700116A (id)
HK (1) HK1020880A1 (id)
HR (1) HRP970569B1 (id)
HU (1) HU224969B1 (id)
ID (1) ID18698A (id)
IL (1) IL129422A0 (id)
IS (1) IS5024A (id)
MY (1) MY119513A (id)
NO (1) NO317163B1 (id)
NZ (1) NZ335153A (id)
OA (1) OA11038A (id)
PA (1) PA8441101A1 (id)
PE (1) PE10099A1 (id)
PL (1) PL190349B1 (id)
PT (1) PT941100E (id)
SI (1) SI0941100T1 (id)
SK (1) SK284286B6 (id)
SV (1) SV1997000090A (id)
TR (1) TR199900950T2 (id)
UA (1) UA64725C2 (id)
UY (1) UY24766A1 (id)
WO (1) WO1998018477A2 (id)
YU (1) YU19999A (id)
ZA (1) ZA979726B (id)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9622681D0 (en) * 1996-10-31 1997-01-08 Glaxo Group Ltd Pharmaceutical compositions
GB9809213D0 (en) * 1998-04-29 1998-07-01 Glaxo Group Ltd Pharmaceutical compositions
US7074417B2 (en) * 2000-10-13 2006-07-11 Advancis Pharmaceutical Corporation Multiple-delayed release anti-viral product, use and formulation thereof
SK285383B6 (sk) * 2002-04-23 2006-12-07 Lupin Limited Kompozície matrice s modifikovaným uvoľňovaním, sdlhodobým účinkom
WO2004043433A2 (en) * 2002-11-08 2004-05-27 Glaxo Group Limited Pharmaceutical antiviral compositions
ES2308136T3 (es) 2003-01-14 2008-12-01 Gilead Sciences, Inc. Composiciones y procedimientos para la politerapia antiviral.
AR045841A1 (es) * 2004-09-28 2005-11-16 Richmond Sa Com Ind Y Financie Una composicion farmaceutica solida que comprende al tiazolil metil ester del acido [5s-(5r*, 8r*, 10r*,11r*)] -10- hidroxi-2- metil-5-(1-metiletil)-1-[2-(1-metiletil)-4-tiazolil]-3,6-dioxo-8,11-bis(fenilmetil)-2,4,7,12- tetraazatridecan-13-oico y un procedimiento para prepararla.
WO2011156594A2 (en) 2010-06-09 2011-12-15 Vaccine Technologies, Incorporated Therapeutic immunization in hiv infected subjects receiving stable antiretroviral treatment
EP2822560A1 (en) 2012-03-05 2015-01-14 Cipla Limited Pharmaceutical antiretroviral combinations comprising lamivudine, festinavir and nevirapine
WO2014130553A2 (en) * 2013-02-20 2014-08-28 Abbvie Inc. Tablet dosage forms

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4950652A (en) * 1987-03-23 1990-08-21 Hem Research, Inc. dsRNAs for combination therapy in the treatment of viral diseases
DK0513917T4 (da) * 1991-05-16 2001-06-25 Glaxo Group Ltd Antivirale kombinationer indeholdende nukleosidanaloger
GB9110624D0 (en) * 1991-05-16 1991-07-03 Glaxo Group Ltd Combinations
GB9622681D0 (en) * 1996-10-31 1997-01-08 Glaxo Group Ltd Pharmaceutical compositions

Also Published As

Publication number Publication date
DE69722433D1 (de) 2003-07-03
MY119513A (en) 2005-06-30
PE10099A1 (es) 1999-03-02
JP2001502718A (ja) 2001-02-27
SI0941100T1 (en) 2003-12-31
SV1997000090A (es) 1998-10-07
CZ296080B6 (cs) 2006-01-11
UA64725C2 (uk) 2004-03-15
WO1998018477A2 (en) 1998-05-07
AP1067A (en) 2002-05-01
DK0941100T3 (da) 2003-09-01
NO317163B1 (no) 2004-08-30
EP0941100B1 (en) 2003-05-28
ZA979726B (en) 1999-04-29
KR100551652B1 (ko) 2006-02-13
CY2485B1 (en) 2005-06-03
ES2200204T3 (es) 2004-03-01
NO992091L (no) 1999-06-29
EA199900345A1 (ru) 2000-02-28
PL190349B1 (pl) 2005-11-30
WO1998018477A3 (en) 1998-06-18
HRP970569A2 (en) 1998-08-31
HU224969B1 (en) 2006-04-28
EP0941100A2 (en) 1999-09-15
PA8441101A1 (es) 2000-05-24
HUP0000344A3 (en) 2002-04-29
CO4930269A1 (es) 2000-06-27
GT199700116A (es) 1999-04-22
CZ155799A3 (cs) 1999-10-13
BG103435A (en) 2000-04-28
YU19999A (sh) 2000-10-30
GB9622681D0 (en) 1997-01-08
AP9901519A0 (en) 1999-06-30
BG64541B1 (bg) 2005-07-29
ATE241364T1 (de) 2003-06-15
AU736607B2 (en) 2001-08-02
DE69722433T2 (de) 2004-04-08
EA002437B1 (ru) 2002-04-25
BR9712614A (pt) 1999-10-26
IL129422A0 (en) 2000-02-17
NZ335153A (en) 2001-04-27
EE9900175A (et) 1999-12-15
PL333143A1 (en) 1999-11-22
UY24766A1 (es) 2000-12-29
AR009135A1 (es) 2000-03-08
NO992091D0 (no) 1999-04-29
SK57599A3 (en) 2000-06-12
AU5314298A (en) 1998-05-22
GEP20022735B (en) 2002-07-25
KR20000052893A (ko) 2000-08-25
IS5024A (is) 1999-04-09
HRP970569B1 (en) 2004-10-31
ID18698A (id) 1998-04-30
TR199900950T2 (xx) 1999-07-21
HK1020880A1 (en) 2000-05-26
PT941100E (pt) 2003-10-31
HUP0000344A2 (hu) 2001-05-28
CA2270174A1 (en) 1998-05-07
EE03806B1 (et) 2002-08-15
OA11038A (en) 2002-02-06

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