SI3510031T1 - Postopek za pripravo 2-(6-nitropiridin-3-il)-9H-dipirido(2,3-b;3',4'-d)pirola - Google Patents

Postopek za pripravo 2-(6-nitropiridin-3-il)-9H-dipirido(2,3-b;3',4'-d)pirola

Info

Publication number
SI3510031T1
SI3510031T1 SI201730610T SI201730610T SI3510031T1 SI 3510031 T1 SI3510031 T1 SI 3510031T1 SI 201730610 T SI201730610 T SI 201730610T SI 201730610 T SI201730610 T SI 201730610T SI 3510031 T1 SI3510031 T1 SI 3510031T1
Authority
SI
Slovenia
Prior art keywords
dipyrido
nitropyridin
pyrrole
preparation
Prior art date
Application number
SI201730610T
Other languages
English (en)
Inventor
Bjoern Bartels
Philipp Cueni
Matthias Koerner
Dieter Muri
Original Assignee
F. Hoffmann-La Roche Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F. Hoffmann-La Roche Ag filed Critical F. Hoffmann-La Roche Ag
Publication of SI3510031T1 publication Critical patent/SI3510031T1/sl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs
SI201730610T 2016-09-09 2017-09-04 Postopek za pripravo 2-(6-nitropiridin-3-il)-9H-dipirido(2,3-b;3',4'-d)pirola SI3510031T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP16187960 2016-09-09
EP17768700.1A EP3510031B1 (en) 2016-09-09 2017-09-04 Process for preparation of 2-(6-nitropyridin-3-yl)-9h-dipyrido[2,3-b;3',4'-d]pyrrole
PCT/EP2017/072062 WO2018046428A1 (en) 2016-09-09 2017-09-04 Process for preparation of 2-(6-nitropyridin-3-yl)-9h-dipyrido[2,3-b;3',4'-d]pyrrole

Publications (1)

Publication Number Publication Date
SI3510031T1 true SI3510031T1 (sl) 2021-03-31

Family

ID=56936288

Family Applications (1)

Application Number Title Priority Date Filing Date
SI201730610T SI3510031T1 (sl) 2016-09-09 2017-09-04 Postopek za pripravo 2-(6-nitropiridin-3-il)-9H-dipirido(2,3-b;3',4'-d)pirola

Country Status (18)

Country Link
US (1) US11306093B2 (sl)
EP (1) EP3510031B1 (sl)
JP (1) JP6997769B2 (sl)
KR (1) KR102502701B1 (sl)
CN (1) CN109689653B (sl)
AR (1) AR109586A1 (sl)
AU (1) AU2017324297B2 (sl)
BR (1) BR112019004091B1 (sl)
CA (1) CA3035624A1 (sl)
ES (1) ES2847903T3 (sl)
HR (1) HRP20210145T1 (sl)
IL (1) IL265013B (sl)
MX (1) MX2019002362A (sl)
PL (1) PL3510031T3 (sl)
SG (1) SG11201901983PA (sl)
SI (1) SI3510031T1 (sl)
TW (1) TWI753009B (sl)
WO (1) WO2018046428A1 (sl)

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR044152A1 (es) * 2003-05-09 2005-08-24 Bayer Corp Derivados de alquilarilo, metodo de preparacion y uso para el tratamiento de la obesidad
FR2876377B1 (fr) 2004-10-11 2007-03-16 Univ Claude Bernard Lyon Nouveaux derives de 9h-pyrido[2,3-b]indole, leur procede de preparation, ainsi que les compositions pharmaceutiques contenant de tels composes
US8932557B2 (en) 2008-02-14 2015-01-13 Eli Lilly And Company Imaging agents for detecting neurological dysfunction
WO2009102498A1 (en) 2008-02-14 2009-08-20 Siemens Medical Solutions Usa, Inc. Novel imaging agents for detecting neurological dysfunction
WO2009151589A1 (en) 2008-06-11 2009-12-17 Genentech, Inc. Diazacarbazoles and methods of use
EP2323697A2 (en) 2008-07-24 2011-05-25 Siemens Medical Solutions USA, Inc. Imaging agents useful for identifying ad pathology
US20100056491A1 (en) * 2008-08-29 2010-03-04 Memory Pharmaceuticals Corporation 4'-amino cyclic compounds having 5-ht6 receptor affinity
EP2411057B1 (en) 2009-03-23 2020-05-06 Eli Lilly and Company Imaging agents for detecting neurological disorders
US8691187B2 (en) 2009-03-23 2014-04-08 Eli Lilly And Company Imaging agents for detecting neurological disorders
US20110183938A1 (en) 2009-12-16 2011-07-28 Genentech, Inc. 1,7-diazacarbazoles and methods of use
US20150368244A1 (en) 2011-01-31 2015-12-24 Genentech, Inc. Diazacarbazoles and methods of use
RU2014103806A (ru) 2011-07-05 2015-08-10 Вертекс Фармасьютикалз Инкорпорейтед Способы и промежуточные соединения для получения азаиндолов
JP6034005B2 (ja) 2011-08-03 2016-11-30 出光興産株式会社 ビスカルバゾール誘導体およびこれを用いた有機エレクトロルミネッセンス素子
EP3055308B1 (en) 2013-10-08 2017-11-22 F.Hoffmann-La Roche Ag Diazacarbazole derivatives as tau-pet-ligands
MY191590A (en) 2015-02-02 2022-06-30 Ucb Biopharma Sprl 9h-pyrrolo-dipyridine derivatives
JP6831372B2 (ja) 2015-09-09 2021-02-17 エフ.ホフマン−ラ ロシュ アーゲーF. Hoffmann−La Roche Aktiengesellschaft 架橋ピペリジン誘導体

Also Published As

Publication number Publication date
JP2019529401A (ja) 2019-10-17
EP3510031A1 (en) 2019-07-17
MX2019002362A (es) 2019-06-17
JP6997769B2 (ja) 2022-02-10
CN109689653A (zh) 2019-04-26
US11306093B2 (en) 2022-04-19
SG11201901983PA (en) 2019-04-29
BR112019004091B1 (pt) 2023-02-14
ES2847903T3 (es) 2021-08-04
US20190300529A1 (en) 2019-10-03
TWI753009B (zh) 2022-01-21
KR20190044648A (ko) 2019-04-30
AU2017324297A1 (en) 2019-03-14
WO2018046428A1 (en) 2018-03-15
TW201811787A (zh) 2018-04-01
CN109689653B (zh) 2022-04-12
BR112019004091A2 (pt) 2019-05-28
PL3510031T3 (pl) 2021-05-31
HRP20210145T1 (hr) 2021-03-05
CA3035624A1 (en) 2018-03-15
AU2017324297B2 (en) 2021-08-05
KR102502701B1 (ko) 2023-02-23
AR109586A1 (es) 2018-12-26
IL265013B (en) 2021-09-30
EP3510031B1 (en) 2020-12-02

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SI3510031T1 (sl) Postopek za pripravo 2-(6-nitropiridin-3-il)-9H-dipirido(2,3-b;3',4'-d)pirola