SI2699581T1 - Derivati 2-okso-1-imidazolidinil imidazotiadiazola - Google Patents

Derivati 2-okso-1-imidazolidinil imidazotiadiazola

Info

Publication number
SI2699581T1
SI2699581T1 SI201230413T SI201230413T SI2699581T1 SI 2699581 T1 SI2699581 T1 SI 2699581T1 SI 201230413 T SI201230413 T SI 201230413T SI 201230413 T SI201230413 T SI 201230413T SI 2699581 T1 SI2699581 T1 SI 2699581T1
Authority
SI
Slovenia
Prior art keywords
oxo
imidazothiadiazole derivatives
imidazolidinyl
imidazolidinyl imidazothiadiazole
derivatives
Prior art date
Application number
SI201230413T
Other languages
English (en)
Inventor
Laurent Provins
Yannick Quesnel
Original Assignee
Ucb Biopharma Sprl
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ucb Biopharma Sprl filed Critical Ucb Biopharma Sprl
Publication of SI2699581T1 publication Critical patent/SI2699581T1/sl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/433Thidiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
SI201230413T 2011-04-18 2012-04-17 Derivati 2-okso-1-imidazolidinil imidazotiadiazola SI2699581T1 (sl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP11162853 2011-04-18
US201161480134P 2011-04-28 2011-04-28
PCT/EP2012/001658 WO2012143117A1 (en) 2011-04-18 2012-04-17 2-oxo-1-imidazolidinyl imidazothiadiazole derivatives
EP12714587.8A EP2699581B1 (en) 2011-04-18 2012-04-17 2-oxo-1-imidazolidinyl imidazothiadiazole derivatives

Publications (1)

Publication Number Publication Date
SI2699581T1 true SI2699581T1 (sl) 2016-02-29

Family

ID=44072751

Family Applications (1)

Application Number Title Priority Date Filing Date
SI201230413T SI2699581T1 (sl) 2011-04-18 2012-04-17 Derivati 2-okso-1-imidazolidinil imidazotiadiazola

Country Status (16)

Country Link
US (1) US8957218B2 (sl)
EP (1) EP2699581B1 (sl)
JP (1) JP5969003B2 (sl)
CA (1) CA2831830C (sl)
CY (1) CY1117210T1 (sl)
DK (1) DK2699581T3 (sl)
ES (1) ES2559288T3 (sl)
HR (1) HRP20151419T1 (sl)
HU (1) HUE026889T2 (sl)
ME (1) ME02351B (sl)
PL (1) PL2699581T3 (sl)
PT (1) PT2699581E (sl)
RS (1) RS54487B1 (sl)
SI (1) SI2699581T1 (sl)
SM (1) SMT201600024B (sl)
WO (1) WO2012143117A1 (sl)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA127921C2 (uk) 2014-01-21 2024-02-14 Янссен Фармацевтика Нв Комбінації, які містять позитивні алостеричні модулятори або ортостеричні агоністи метаботропного глутаматергічного рецептора 2 підтипу, та їх застосування
DK3096790T3 (da) 2014-01-21 2019-10-07 Janssen Pharmaceutica Nv Kombinationer omfattende positive allosteriske modulatorer eller orthosteriske agonister af metabotrop glutamaterg subtype 2-receptor og anvendelse af disse
MA49558A (fr) * 2017-07-10 2021-05-05 UCB Biopharma SRL Dérivativés de 2-oxo-1-imidazolidinyl imidazothiadiazole
RU2020104753A (ru) * 2017-07-10 2021-08-10 Юсб Байофарма Срл Производные 2-оксо-1, 3-оксазолидинилимидазотиазола
MA51126A (fr) 2017-12-12 2020-10-21 UCB Biopharma SRL Dérivés de 2-oxo-1-pyrrolidinyl imidazothiadiazole
JP7340542B2 (ja) * 2018-05-08 2023-09-07 ユーシービー バイオファルマ エスアールエル 1-イミダゾチアジアゾロ-2h-ピロール-5-オン誘導体

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1464259A (en) * 1975-10-03 1977-02-09 Pfizer Ltd Imidazo-thiazole and -thiadiazole sulphonamides and their use as therapeutic agents
GB8412357D0 (en) 1984-05-15 1984-06-20 Ucb Sa Pharmaceutical composition
GB8412358D0 (en) 1984-05-15 1984-06-20 Ucb Sa Pharmaceutical composition
GB0004297D0 (en) 2000-02-23 2000-04-12 Ucb Sa 2-oxo-1 pyrrolidine derivatives process for preparing them and their uses
EP1706376B1 (en) 2003-12-02 2009-03-04 UCB Pharma, S.A. Imidazole derivatives, processes for preparing them and their uses
JP2008542322A (ja) 2005-06-01 2008-11-27 ユセベ ファルマ ソシエテ アノニム 2−オキソ−1−ピロリジン誘導体
WO2008132139A2 (en) 2007-04-27 2008-11-06 Ucb Pharma S.A. New heterocyclic derivatives useful for the treatment of cns disorders
CN102574869A (zh) * 2009-10-23 2012-07-11 Ucb医药有限公司 2-氧代-1-吡咯烷基咪唑并噻二唑衍生物

Also Published As

Publication number Publication date
CA2831830C (en) 2017-12-12
ME02351B (me) 2016-06-20
HUE026889T2 (en) 2016-07-28
DK2699581T3 (en) 2016-01-11
CA2831830A1 (en) 2012-10-26
SMT201600024B (sl) 2016-02-25
RS54487B1 (en) 2016-06-30
HRP20151419T1 (hr) 2016-01-29
WO2012143117A1 (en) 2012-10-26
JP5969003B2 (ja) 2016-08-10
AU2012244614A1 (en) 2013-10-31
US8957218B2 (en) 2015-02-17
PL2699581T3 (pl) 2016-05-31
US20140148489A1 (en) 2014-05-29
JP2014511883A (ja) 2014-05-19
EP2699581A1 (en) 2014-02-26
ES2559288T3 (es) 2016-02-11
PT2699581E (pt) 2016-03-22
CY1117210T1 (el) 2017-04-05
EP2699581B1 (en) 2015-11-25

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