SI1706385T1 - Pirazolni derivati kot modulatorji protein-kinaze - Google Patents

Pirazolni derivati kot modulatorji protein-kinaze

Info

Publication number
SI1706385T1
SI1706385T1 SI200431571T SI200431571T SI1706385T1 SI 1706385 T1 SI1706385 T1 SI 1706385T1 SI 200431571 T SI200431571 T SI 200431571T SI 200431571 T SI200431571 T SI 200431571T SI 1706385 T1 SI1706385 T1 SI 1706385T1
Authority
SI
Slovenia
Prior art keywords
protein kinase
pyrazole derivatives
kinase modulators
modulators
pyrazole
Prior art date
Application number
SI200431571T
Other languages
English (en)
Inventor
Valerio Berdini
Gordon Saxty
Marinus Leendert Verdonk
Steven John Woodhead
Paul Graham Wyatt
Robert George Boyle
Hannah Fiona Sore
David Winter Walker
Ian Collins
Robert Downham
Robin Arthur Ellis Carr
Original Assignee
Astex Therapeutics Ltd
Cancer Rec Tech Ltd
Cancer Res Inst Royal
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astex Therapeutics Ltd, Cancer Rec Tech Ltd, Cancer Res Inst Royal filed Critical Astex Therapeutics Ltd
Priority claimed from EP04806258A external-priority patent/EP1706385B1/en
Publication of SI1706385T1 publication Critical patent/SI1706385T1/sl

Links

SI200431571T 2003-12-23 2004-12-23 Pirazolni derivati kot modulatorji protein-kinaze SI1706385T1 (sl)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US53219903P 2003-12-23 2003-12-23
GB0329617A GB0329617D0 (en) 2003-12-23 2003-12-23 Pharmaceutical compounds
US57784304P 2004-06-08 2004-06-08
EP04806258A EP1706385B1 (en) 2003-12-23 2004-12-23 Pyrazole derivatives as protein kinase modulators
PCT/GB2004/005464 WO2005061463A1 (en) 2003-12-23 2004-12-23 Pyrazole derivatives as protein kinase modulators

Publications (1)

Publication Number Publication Date
SI1706385T1 true SI1706385T1 (sl) 2011-01-31

Family

ID=30776233

Family Applications (1)

Application Number Title Priority Date Filing Date
SI200431571T SI1706385T1 (sl) 2003-12-23 2004-12-23 Pirazolni derivati kot modulatorji protein-kinaze

Country Status (11)

Country Link
CN (1) CN1922148B (sl)
AT (1) ATE483689T1 (sl)
DE (1) DE602004029501D1 (sl)
DK (1) DK1706385T3 (sl)
GB (1) GB0329617D0 (sl)
ME (1) ME01934B (sl)
PT (1) PT1706385E (sl)
RS (1) RS51546B (sl)
SI (1) SI1706385T1 (sl)
UA (1) UA90461C2 (sl)
ZA (1) ZA200605127B (sl)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0704932D0 (en) * 2007-03-14 2007-04-25 Astex Therapeutics Ltd Pharmaceutical compounds
CN108339121A (zh) * 2017-01-25 2018-07-31 苏州大学 蛋白激酶a抑制剂在制备治疗血小板数量增多相关疾病药物中的用途
CN111056990B (zh) * 2019-12-16 2022-06-17 爱斯特(成都)生物制药股份有限公司 一种合成1-叔丁氧羰基-4-(4-羧基苯基)哌啶的制备方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9804734D0 (en) * 1998-03-05 1998-04-29 Pfizer Ltd Compounds
KR20020091829A (ko) * 1999-07-30 2002-12-06 애보트 게엠베하 운트 콤파니 카게 2-피라졸린-5-온

Also Published As

Publication number Publication date
UA90461C2 (en) 2010-05-11
ME01934B (me) 2011-06-30
RS51546B (en) 2011-06-30
GB0329617D0 (en) 2004-01-28
PT1706385E (pt) 2010-12-22
DK1706385T3 (da) 2011-01-10
ATE483689T1 (de) 2010-10-15
CN1922148A (zh) 2007-02-28
CN1922148B (zh) 2012-03-21
ZA200605127B (en) 2010-07-28
DE602004029501D1 (de) 2010-11-18

Similar Documents

Publication Publication Date Title
HK1097543A1 (en) Pyrazole derivatives as protein kinase modulators
IL173380A0 (en) Pyridinylamino-pyrimidine derivatives as protein kinase inhibitors
EP1684762A4 (en) UREA DERIVATIVES AS MODULATORS OF KINASE
EP1670460A4 (en) PYRAZOLE DERIVATIVES AS MODULATORS OF THE CANNABINOID RECEPTOR
GB0309637D0 (en) Pyrazole compounds
PL377778A1 (pl) Pochodne pirazolu
AP2048A (en) Diazepinoindole derivatives as kinase inhibitors
AP2114A (en) Aminoheteroaryl compounds as protein kinase inhibitors
ZA200606921B (en) Fused derivatives of pyrazole
PL377844A1 (pl) Podstawione pirazole
IL172132A0 (en) Thienopyridone derivatives as kinase inhibitors
IL180044A0 (en) Pyrazole derivatives
ZA200604069B (en) AKT protein kinase inhibitors
ZA200508946B (en) Pyrazole compounds
HUP0500111A3 (en) Indolinone derivatives useful as protein kinase inhibitors
ZA200508923B (en) Substituted pyrazole compounds
IL173911A0 (en) Imidazole derivatives
ZA200800327B (en) Pyrazole derivatives as CB 1 modulators
IL174911A0 (en) N-Substituted pyrazolyl carboxanilides
IL180889A0 (en) Pyrazole derivative
SI1603570T1 (sl) Spojine aminoheteroarila kot zaviralci proteinkinaze
EP1581309A4 (en) KINASE MODULATORS
ZA200605127B (en) Pyrazole derivatives as protein kinase modulators
EG27149A (en) Pyrazole derivatives as anti-inflammatory-antimicrobial agent
AU2004228124B2 (en) Substituted pyrazole compounds