SI1082314T1 - New dipeptidyl peptidase iv effectors - Google Patents

New dipeptidyl peptidase iv effectors

Info

Publication number
SI1082314T1
SI1082314T1 SI9930209T SI9930209T SI1082314T1 SI 1082314 T1 SI1082314 T1 SI 1082314T1 SI 9930209 T SI9930209 T SI 9930209T SI 9930209 T SI9930209 T SI 9930209T SI 1082314 T1 SI1082314 T1 SI 1082314T1
Authority
SI
Slovenia
Prior art keywords
dipeptidyl peptidase
peptidase iv
iv effectors
new dipeptidyl
new
Prior art date
Application number
SI9930209T
Other languages
Slovenian (sl)
Inventor
Hans-Ulrich Demuth
Konrad Glund
Dagmar Schlenzig
Susanne Kruber
Original Assignee
Probiodrug Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to DE1998123831 priority Critical patent/DE19823831A1/en
Application filed by Probiodrug Ag filed Critical Probiodrug Ag
Priority to PCT/EP1999/003712 priority patent/WO1999061431A1/en
Priority to EP19990926464 priority patent/EP1082314B1/en
Publication of SI1082314T1 publication Critical patent/SI1082314T1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2.] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2.] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2.] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182Radicals derived from carboxylic acids
    • C07D295/185Radicals derived from carboxylic acids from aliphatic carboxylic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/4261,3-Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/427Thiazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/04Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
SI9930209T 1998-05-28 1999-05-28 New dipeptidyl peptidase iv effectors SI1082314T1 (en)

Priority Applications (3)

Application Number Priority Date Filing Date Title
DE1998123831 DE19823831A1 (en) 1998-05-28 1998-05-28 New pharmaceutical use of isoleucyl thiazolidide and its salts
PCT/EP1999/003712 WO1999061431A1 (en) 1998-05-28 1999-05-28 New dipeptidyl peptidase iv effectors
EP19990926464 EP1082314B1 (en) 1998-05-28 1999-05-28 New dipeptidyl peptidase iv effectors

Publications (1)

Publication Number Publication Date
SI1082314T1 true SI1082314T1 (en) 2003-08-31

Family

ID=7869159

Family Applications (2)

Application Number Title Priority Date Filing Date
SI9930209T SI1082314T1 (en) 1998-05-28 1999-05-28 New dipeptidyl peptidase iv effectors
SI9930771T SI1304327T1 (en) 1998-05-28 1999-05-28

Family Applications After (1)

Application Number Title Priority Date Filing Date
SI9930771T SI1304327T1 (en) 1998-05-28 1999-05-28

Country Status (23)

Country Link
US (4) US6548481B1 (en)
EP (6) EP1398030B1 (en)
JP (1) JP2002516318A (en)
KR (1) KR100630258B1 (en)
CN (4) CN1332954C (en)
AT (6) AT338546T (en)
AU (1) AU764262B2 (en)
BR (1) BR9910758A (en)
CA (1) CA2333603C (en)
DE (10) DE19823831A1 (en)
DK (2) DK1304327T3 (en)
ES (5) ES2271458T3 (en)
HK (3) HK1033316A1 (en)
HU (1) HU0102001A3 (en)
IL (3) IL139862D0 (en)
IS (3) IS5728A (en)
NO (1) NO317989B1 (en)
NZ (2) NZ525799A (en)
PL (1) PL344403A1 (en)
PT (2) PT1304327E (en)
RU (3) RU2227800C2 (en)
SI (2) SI1082314T1 (en)
WO (1) WO1999061431A1 (en)

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AU4370999A (en) 1999-12-13
CN101095675A (en) 2008-01-02
EP1215207A2 (en) 2002-06-19
DE29909210U1 (en) 1999-09-09
AT231497T (en) 2003-02-15
NO20005994L (en) 2001-01-25
HU0102001A3 (en) 2001-12-28
CN1637018A (en) 2005-07-13
ES2193709T3 (en) 2003-11-01
US20030134802A1 (en) 2003-07-17
DE59911670D1 (en) 2005-03-31
EP1214936A2 (en) 2002-06-19
EP1082314A1 (en) 2001-03-14
NZ508260A (en) 2003-06-30
RU2003121766A (en) 2005-02-10
HK1033316A1 (en) 2003-08-15
JP2002516318A (en) 2002-06-04
IS7763A (en) 2005-03-21
EP1304327A2 (en) 2003-04-23
AT272059T (en) 2004-08-15
US20050203030A1 (en) 2005-09-15
DE59910084D1 (en) 2004-09-02
IS2130B (en) 2006-07-14
EP1214936A3 (en) 2002-07-03
DE29909208U1 (en) 1999-09-09
EP1398030B1 (en) 2006-09-06
HU0102001A2 (en) 2001-11-28
DE59910083D1 (en) 2004-09-02
KR20040063979A (en) 2004-07-15
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EP1428533A3 (en) 2004-06-23
US20080182798A1 (en) 2008-07-31

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