SI1038875T1 - Imidazopyridine derivatives and process for making them - Google Patents

Imidazopyridine derivatives and process for making them

Info

Publication number
SI1038875T1
SI1038875T1 SI9930383T SI9930383T SI1038875T1 SI 1038875 T1 SI1038875 T1 SI 1038875T1 SI 9930383 T SI9930383 T SI 9930383T SI 9930383 T SI9930383 T SI 9930383T SI 1038875 T1 SI1038875 T1 SI 1038875T1
Authority
SI
Slovenia
Prior art keywords
making
imidazopyridine derivatives
chem
compound
formula
Prior art date
Application number
SI9930383T
Other languages
English (en)
Slovenian (sl)
Inventor
Gerrit Jan Bouke Ettema
Jacobus Maria Lemmens
Theodorus Hendricus Antonius Peters
Frantisek Picha
Original Assignee
Synthon B.V.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthon B.V. filed Critical Synthon B.V.
Publication of SI1038875T1 publication Critical patent/SI1038875T1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Inert Electrodes (AREA)
SI9930383T 1999-03-25 1999-10-22 Imidazopyridine derivatives and process for making them SI1038875T1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US12649499P 1999-03-25 1999-03-25
EP99203478A EP1038875B1 (en) 1999-03-25 1999-10-22 Imidazopyridine derivatives and process for making them

Publications (1)

Publication Number Publication Date
SI1038875T1 true SI1038875T1 (en) 2003-12-31

Family

ID=22425138

Family Applications (1)

Application Number Title Priority Date Filing Date
SI9930383T SI1038875T1 (en) 1999-03-25 1999-10-22 Imidazopyridine derivatives and process for making them

Country Status (8)

Country Link
US (2) US6242460B1 (xx)
EP (1) EP1038875B1 (xx)
AT (1) ATE242241T1 (xx)
DE (1) DE69908546T2 (xx)
DK (1) DK1038875T3 (xx)
ES (1) ES2195510T3 (xx)
PT (1) PT1038875E (xx)
SI (1) SI1038875T1 (xx)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1272181A2 (en) 2000-04-13 2003-01-08 Synthon B.V. Modified release formulations containing a hypnotic agent
DE60125429T2 (de) * 2000-04-24 2007-09-27 Teva Pharmaceutical Industries Ltd. Zolpidem hemitartrat solvat
EP1600159A1 (en) * 2000-04-24 2005-11-30 Teva Pharmaceutical Industries Ltd A method for synthesizing different Zolpidem hemitartrate derivatives
US20030165566A1 (en) * 2002-01-10 2003-09-04 O'toole Edel Sedative non-benzodiazepine formulations
ES2320758T3 (es) * 2002-12-18 2009-05-28 Mallinckrodt Inc. Sintesis de heteroaril acetamidas.
GB0329918D0 (en) * 2003-12-24 2004-01-28 West Pharm Serv Drug Res Ltd Intranasal compositions
EP1715853A4 (en) * 2004-02-17 2012-07-18 Transcept Pharmaceuticals Inc COMPOSITIONS FOR THE DISTRIBUTION OF HYPNOTICS IN THE FIELD OF MUNICHCHLEIMHÄUTE AND USE METHOD THEREOF
US20080262025A1 (en) * 2004-07-16 2008-10-23 Yatendra Kumar Processes for the Preparation of Zolpidem and its Hemitartrate
NZ563979A (en) * 2005-05-25 2011-02-25 Transcept Pharmaceuticals Inc Solid compositions and methods for treating middle-of-the night insomnia
US20070287740A1 (en) * 2005-05-25 2007-12-13 Transcept Pharmaceuticals, Inc. Compositions and methods of treating middle-of-the night insomnia
US20070225322A1 (en) * 2005-05-25 2007-09-27 Transoral Pharmaceuticals, Inc. Compositions and methods for treating middle-of-the night insomnia
CA2626242A1 (en) * 2005-10-17 2007-04-26 Mallinckrodt Inc. Polymorph transformation of zolpidem in tablet matrix
US20070098788A1 (en) * 2005-10-28 2007-05-03 Gore Subhash P Non-benzodiazepine hypnotic compositions
US8148393B2 (en) * 2005-11-18 2012-04-03 Synthon Bv Zolpidem tablets
US7989207B2 (en) * 2006-02-17 2011-08-02 Tyco Healthcare Group Lp Testing lumenectomy samples for markers of non-vascular diseases
DK2007752T3 (da) 2006-03-31 2010-11-15 Janssen Pharmaceutica Nv Benzimidazol-2-yl-pyrimidiner og -pyraziner som modulatorer af histamin H4-receptoren
US20080145425A1 (en) * 2006-12-15 2008-06-19 Pliva Research & Development Limited Pharmaceutical composition of zolpidem
US9371311B2 (en) 2008-06-30 2016-06-21 Janssen Pharmaceutica Nv Benzoimidazol-2-yl pyrimidine derivatives
WO2010074753A1 (en) 2008-12-23 2010-07-01 Map Pharmaceuticals, Inc. Inhalation devices and related methods for administration of sedative hypnotic compounds
AU2014225675B2 (en) 2013-03-06 2018-10-04 Janssen Pharmaceutica Nv Benzoimidazol-2-yl pyrimidine modulators of the histamine H4 receptor
CN104610253B (zh) * 2015-01-26 2016-11-16 郑州大学 2‑三氟甲基‑2‑羟基‑2‑(2‑芳基吡啶并[1,2‑α]咪唑)乙酸酯类化合物
CN106432233B (zh) * 2016-09-20 2018-08-14 华东理工大学 N,N,6-三甲基-2-(4-甲基苯基)咪唑并[1,2-a]吡啶-3-乙酰胺的制备方法
EP3611256A1 (en) * 2018-08-14 2020-02-19 Universität Heidelberg Application of imidazopyridine derivatives in regenerative medicine

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2492382A1 (fr) * 1980-10-22 1982-04-23 Synthelabo Derives d'imidazo (1,2-a) pyridine, leur preparation et leur application en therapeutique
FR2600650B1 (fr) 1986-06-27 1988-09-09 Synthelabo Procede de preparation d'imidazopyridines et composes intermediaires

Also Published As

Publication number Publication date
DK1038875T3 (da) 2003-09-29
PT1038875E (pt) 2003-10-31
EP1038875B1 (en) 2003-06-04
EP1038875A3 (en) 2001-09-12
DE69908546D1 (de) 2003-07-10
US6281360B1 (en) 2001-08-28
ES2195510T3 (es) 2003-12-01
US6242460B1 (en) 2001-06-05
EP1038875A2 (en) 2000-09-27
DE69908546T2 (de) 2004-04-29
ATE242241T1 (de) 2003-06-15

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