SG27001G - Ether prodrugs of anti-inflammatory oxicams - Google Patents

Ether prodrugs of anti-inflammatory oxicams

Info

Publication number
SG27001G
SG27001G SG305/89A SG1989903058A SG27001G SG 27001 G SG27001 G SG 27001G SG 305/89 A SG305/89 A SG 305/89A SG 1989903058 A SG1989903058 A SG 1989903058A SG 27001 G SG27001 G SG 27001G
Authority
SG
Singapore
Prior art keywords
oxicams
inflammatory
ether prodrugs
prodrugs
ether
Prior art date
Application number
SG305/89A
Other languages
English (en)
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of SG27001G publication Critical patent/SG27001G/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C68/00Preparation of esters of carbonic or haloformic acids
    • C07C68/02Preparation of esters of carbonic or haloformic acids from phosgene or haloformates
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
SG305/89A 1983-12-21 1984-12-19 Ether prodrugs of anti-inflammatory oxicams SG27001G (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US56390283A 1983-12-21 1983-12-21
US06/606,113 US4551452A (en) 1983-12-21 1984-05-02 Anti-inflammatory 2-methyl-2H-1,2-benzo-(or -thieno-)thiazine-3-carboxamide 1,1-dioxide derivatives, compositions, and method of use therefor

Publications (1)

Publication Number Publication Date
SG27001G true SG27001G (en) 1989-08-11

Family

ID=27073413

Family Applications (1)

Application Number Title Priority Date Filing Date
SG305/89A SG27001G (en) 1983-12-21 1984-12-19 Ether prodrugs of anti-inflammatory oxicams

Country Status (26)

Country Link
US (1) US4551452A (fr)
EP (1) EP0147177B1 (fr)
KR (1) KR860002035B1 (fr)
AU (1) AU552940B2 (fr)
BG (1) BG47946A3 (fr)
CA (1) CA1255302A (fr)
DD (1) DD229125A5 (fr)
DE (1) DE3466776D1 (fr)
DK (1) DK166678B1 (fr)
EG (1) EG17049A (fr)
ES (1) ES8604215A1 (fr)
FI (1) FI79850C (fr)
GR (1) GR82512B (fr)
HK (1) HK58589A (fr)
HU (1) HU201063B (fr)
IE (1) IE57680B1 (fr)
IL (1) IL73873A (fr)
MX (2) MX174596B (fr)
NO (1) NO161317C (fr)
NZ (1) NZ210632A (fr)
PH (1) PH21447A (fr)
PL (1) PL145989B1 (fr)
PT (1) PT79700B (fr)
RO (1) RO90048A (fr)
SG (1) SG27001G (fr)
YU (1) YU43677B (fr)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5017567A (en) * 1983-11-25 1991-05-21 Schering Corporation Carboxyalkyl dipeptides as antiglaucoma agents
US4616012A (en) * 1983-11-25 1986-10-07 Schering Corporation Carboxyalkyl dipeptides as antiglaucoma agents
US4778795A (en) * 1983-11-25 1988-10-18 Schering Corporation Carboxyalkyl dipeptides as antiglaucoma agents
US4906635A (en) * 1983-11-25 1990-03-06 Schering Corporation Carboxyalkyl dipeptides as antiglaucoma agents
US4623486A (en) * 1985-05-29 1986-11-18 Pfizer Inc. [4-substituted benzoyloxy]-N-substituted-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxides having anti-arthritic activity
KR890001236B1 (ko) * 1985-10-02 1989-04-28 화이자 인코포레이티드 소염제 조성물의 제조방법
US4771071A (en) * 1986-05-05 1988-09-13 Merck & Co., Inc. Antihypercholesterolemic compounds
MX6506A (es) * 1986-05-16 1993-10-01 Pfizer Derivados de dioxido de benzotiazina y procedimiento para su preparacion
US5081118A (en) * 1987-10-26 1992-01-14 Pfizer Inc. Benzothiazine dioxide derivatives
NZ226477A (en) * 1987-10-29 1990-07-26 Cl Pharma Substituted thieno (2,3-e)-1,2 thiazine derivatives and pharmaceutical compositions
ZA945190B (en) * 1993-07-30 1995-02-24 Kotobuki Seiyaku Co Ltd Carboxymethylidenecycloheptimidazole derivatives method or manufacturing the same and therapeutic agents containing these compounds
IT1308633B1 (it) 1999-03-02 2002-01-09 Nicox Sa Nitrossiderivati.
CN100389114C (zh) * 2006-01-17 2008-05-21 南京新港医药有限公司 一种安吡昔康的精制方法
US20090221703A1 (en) 2006-07-09 2009-09-03 Chongxi Yu High penetration composition and uses thereof
US20090238763A1 (en) 2006-07-09 2009-09-24 Chongxi Yu High penetration compositions and uses thereof
CN101522692A (zh) * 2006-10-11 2009-09-02 于崇曦 具有快速皮肤穿透速度的带正电荷的水溶性的昔康及其相关化合物的前药
JP2010529101A (ja) * 2007-06-04 2010-08-26 テックフィールズ インコーポレイテッド 非常に速い皮膚及び膜浸透速度を有するnsaiaプロドラッグ及びその新規医薬使用
MX362949B (es) 2008-12-04 2019-02-27 Yu Chongxi Composiciones de alta penetracion y sus aplicaciones.
WO2013093931A2 (fr) 2011-09-19 2013-06-27 Sun Pharma Advanced Research Company Ltd. Nouveaux promédicaments de médicaments phénoliques

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3591584A (en) * 1968-08-27 1971-07-06 Pfizer Benzothiazine dioxides
US3787324A (en) * 1971-03-01 1974-01-22 Warner Lambert Co 4-hydroxy-3-(3-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,dioxides and process for their production
US3892740A (en) * 1974-10-15 1975-07-01 Pfizer Process for the production of carboxamides of oxo-1,2-benzothiazine-1,1-dioxides
AU518216B2 (en) * 1977-09-06 1981-09-17 Hafslund Nycomed Pharma Aktiengesellschaft Thienothiazine derivatives
US4309427A (en) * 1981-01-15 1982-01-05 Pfizer Inc. Benzothiazine dioxide derivatives
IT1168064B (it) * 1981-11-12 1987-05-20 Prodotti Antibiotici Spa Composto ad azione antinfiammatoria
IT8219486A0 (it) * 1982-02-05 1982-02-05 Chiesi Farma Spa Nuovi composti ad attivita'antiinfiammatoria, procedimento per la loro preparazione e relative composizioni farmaceutiche.

Also Published As

Publication number Publication date
HUT37426A (en) 1985-12-28
DK614984A (da) 1985-07-17
DK614984D0 (da) 1984-12-20
KR860002035B1 (ko) 1986-11-17
NO845145L (no) 1985-06-24
AU3699784A (en) 1985-07-04
HU201063B (en) 1990-09-28
DE3466776D1 (en) 1987-11-19
EP0147177A3 (en) 1985-08-14
FI79850B (fi) 1989-11-30
EG17049A (en) 1991-03-30
IL73873A0 (en) 1985-03-31
PL145989B1 (en) 1988-12-31
GR82512B (en) 1985-04-22
HK58589A (en) 1989-07-28
RO90048A (fr) 1986-09-30
DD229125A5 (de) 1985-10-30
YU43677B (en) 1989-10-31
PH21447A (en) 1987-10-28
YU216084A (en) 1986-10-31
PT79700A (en) 1985-01-01
NO161317B (no) 1989-04-24
BG47946A3 (en) 1990-10-15
AU552940B2 (en) 1986-06-26
ES8604215A1 (es) 1986-01-16
CA1255302A (fr) 1989-06-06
IE843260L (en) 1985-06-21
EP0147177A2 (fr) 1985-07-03
DK166678B1 (da) 1993-06-28
MX174596B (es) 1994-05-30
IE57680B1 (en) 1993-02-24
KR850004492A (ko) 1985-07-15
ES538907A0 (es) 1986-01-16
FI79850C (fi) 1990-03-12
EP0147177B1 (fr) 1987-10-14
NO161317C (no) 1989-08-02
PT79700B (en) 1986-12-30
FI845074L (fi) 1985-06-22
FI845074A0 (fi) 1984-12-20
US4551452A (en) 1985-11-05
NZ210632A (en) 1987-02-20
MX9203740A (es) 1992-09-01
PL251040A1 (en) 1985-10-22
IL73873A (en) 1988-02-29

Similar Documents

Publication Publication Date Title
DE3466776D1 (en) Ether prodrugs of anti-inflammatory oxicams
JPS57150628A (en) Manufacture of alpha-alkylacrolein
JPS57193374A (en) Manufacture of jet-nozzle-duct
JPS57154140A (en) Manufacture of hydroxyarylophenone
JPS57209926A (en) Manufacture of polyoxyalkylene monoallyl- or -methallyl ether
GB8321678D0 (en) Production of methanol
JPS57203037A (en) Manufacture of p-nitrophenetol
JPS57212145A (en) Manufacture of cyclohexyamine
JPS57185286A (en) Manufacture of isosorbit-5-nitrate
JPS57139030A (en) Manufacture of unsaturated ether
GB8327533D0 (en) Manufacture of slates
GB8504355D0 (en) Prodrugs of anti-inflammatory oxicams
JPS57159759A (en) Manufacture of 4-haloazetidine-2-ones
JPS57149245A (en) Manufacture of polychlorobenzoylchloride
ZA849926B (en) Ether prodrugs of antiinflammatory oxicams
JPS57203075A (en) Manufacture of halogen-2-mercaptobenzoxazole
DE3377985D1 (en) Production of hydroquinone
JPS57209294A (en) Manufacture of silylisocyanate
KE3883A (en) Ether prodrugs of anti-inflammatory oxicams
GB8304857D0 (en) Manufacture of nitrophenetoles
DE3377777D1 (en) Improvements relating to the manufacture of toilets
GB8328172D0 (en) Manufacture of fiberglass etc
IL72271A (en) Manufacture of 2-isopropyl-4-methyl-6-hydroxypyrimidine
JPS57209263A (en) Manufacture of n-monosubstituted-o-alkylurethane
JPS57169436A (en) Manufacture of methanol