SG187877A1 - Novel peptides which have analgesic effects and which inhibit asic channels - Google Patents
Novel peptides which have analgesic effects and which inhibit asic channels Download PDFInfo
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- SG187877A1 SG187877A1 SG2013011705A SG2013011705A SG187877A1 SG 187877 A1 SG187877 A1 SG 187877A1 SG 2013011705 A SG2013011705 A SG 2013011705A SG 2013011705 A SG2013011705 A SG 2013011705A SG 187877 A1 SG187877 A1 SG 187877A1
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- peptide
- asicalgin
- pain
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- asicla
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/46—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
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- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
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- A—HUMAN NECESSITIES
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- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- A—HUMAN NECESSITIES
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- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/1703—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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- Animal Behavior & Ethology (AREA)
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- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Gastroenterology & Hepatology (AREA)
- Biochemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Toxicology (AREA)
- Zoology (AREA)
- Psychiatry (AREA)
- Rheumatology (AREA)
- Physical Education & Sports Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Urology & Nephrology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR1003136A FR2963010B1 (fr) | 2010-07-26 | 2010-07-26 | Nouveaux peptides avec des effets analgesiques et inhibant les canaux asic |
| PCT/FR2011/051800 WO2012022894A1 (fr) | 2010-07-26 | 2011-07-26 | Nouveaux peptides avec des effets analgesiques et inhibant les canaux asic |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SG187877A1 true SG187877A1 (en) | 2013-03-28 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SG2013011705A SG187877A1 (en) | 2010-07-26 | 2011-07-26 | Novel peptides which have analgesic effects and which inhibit asic channels |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US8987207B2 (enExample) |
| EP (1) | EP2598523B1 (enExample) |
| JP (1) | JP6000245B2 (enExample) |
| CN (1) | CN103097404B (enExample) |
| AU (1) | AU2011290589A1 (enExample) |
| BR (1) | BR112013001863A2 (enExample) |
| CA (1) | CA2806471C (enExample) |
| FR (1) | FR2963010B1 (enExample) |
| MX (1) | MX336586B (enExample) |
| RU (1) | RU2583299C2 (enExample) |
| SG (1) | SG187877A1 (enExample) |
| WO (1) | WO2012022894A1 (enExample) |
| ZA (1) | ZA201300662B (enExample) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN105233286B (zh) * | 2015-09-10 | 2018-10-30 | 上海交通大学医学院 | 含酸敏感离子通道调控剂的制剂及其在治疗瘙痒中的用途 |
| CN105412932B (zh) * | 2015-10-26 | 2019-08-16 | 上海交通大学医学院 | 含ASIC1a与RIP1结合抑制剂的制剂及其抑制神经元死亡的用途 |
| CN112717135A (zh) * | 2016-11-22 | 2021-04-30 | 上海交通大学医学院 | 酸敏感离子通道调控剂的用途 |
| CN107384952A (zh) * | 2017-08-23 | 2017-11-24 | 湖南甲骨文生物医药有限公司 | 用于筛选ASICs作用蛋白的酵母双杂交诱饵载体的构建方法 |
| CN114729034B (zh) * | 2019-06-04 | 2024-01-12 | 上海科技大学 | 亲和力成熟的抗ASIC1a抗体 |
| RU2768484C1 (ru) * | 2021-05-24 | 2022-03-24 | Закрытое акционерное общество "СКАЙ ЛТД" | Фармацевтическая композиция иммуностимулирующих веществ мурамилпептидной природы |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5776896A (en) | 1996-01-03 | 1998-07-07 | Zeneca Limited | Analgesic peptides from venom of grammostola spatulata and use thereof |
| JP4959226B2 (ja) * | 2006-05-19 | 2012-06-20 | 独立行政法人産業技術総合研究所 | スリーフィンガー様蛋白質ライブラリ |
| JP2008193923A (ja) * | 2007-02-09 | 2008-08-28 | Janusys Kk | 蛋白質ライブラリ |
-
2010
- 2010-07-26 FR FR1003136A patent/FR2963010B1/fr not_active Expired - Fee Related
-
2011
- 2011-07-26 CN CN201180043328.6A patent/CN103097404B/zh active Active
- 2011-07-26 WO PCT/FR2011/051800 patent/WO2012022894A1/fr not_active Ceased
- 2011-07-26 SG SG2013011705A patent/SG187877A1/en unknown
- 2011-07-26 CA CA2806471A patent/CA2806471C/fr active Active
- 2011-07-26 MX MX2013001020A patent/MX336586B/es unknown
- 2011-07-26 JP JP2013521194A patent/JP6000245B2/ja active Active
- 2011-07-26 RU RU2013108262/10A patent/RU2583299C2/ru active
- 2011-07-26 US US13/812,457 patent/US8987207B2/en active Active
- 2011-07-26 AU AU2011290589A patent/AU2011290589A1/en not_active Abandoned
- 2011-07-26 BR BR112013001863A patent/BR112013001863A2/pt not_active Application Discontinuation
- 2011-07-26 EP EP11752299.5A patent/EP2598523B1/fr active Active
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2013
- 2013-01-24 ZA ZA2013/00662A patent/ZA201300662B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP2598523B1 (fr) | 2015-09-09 |
| BR112013001863A2 (pt) | 2016-05-31 |
| CN103097404A (zh) | 2013-05-08 |
| FR2963010A1 (fr) | 2012-01-27 |
| WO2012022894A1 (fr) | 2012-02-23 |
| EP2598523A1 (fr) | 2013-06-05 |
| AU2011290589A1 (en) | 2013-03-07 |
| JP6000245B2 (ja) | 2016-09-28 |
| RU2013108262A (ru) | 2014-09-10 |
| MX336586B (es) | 2016-01-21 |
| ZA201300662B (en) | 2013-09-25 |
| FR2963010B1 (fr) | 2014-08-15 |
| CA2806471C (fr) | 2020-07-07 |
| MX2013001020A (es) | 2014-04-14 |
| WO2012022894A4 (fr) | 2012-04-12 |
| RU2583299C2 (ru) | 2016-05-10 |
| JP2013535965A (ja) | 2013-09-19 |
| CN103097404B (zh) | 2015-09-16 |
| US8987207B2 (en) | 2015-03-24 |
| CA2806471A1 (fr) | 2012-02-23 |
| US20130196923A1 (en) | 2013-08-01 |
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