SG187193A1 - Combinations of hepatitis c virus inhibitors - Google Patents
Combinations of hepatitis c virus inhibitors Download PDFInfo
- Publication number
- SG187193A1 SG187193A1 SG2013005905A SG2013005905A SG187193A1 SG 187193 A1 SG187193 A1 SG 187193A1 SG 2013005905 A SG2013005905 A SG 2013005905A SG 2013005905 A SG2013005905 A SG 2013005905A SG 187193 A1 SG187193 A1 SG 187193A1
- Authority
- SG
- Singapore
- Prior art keywords
- compound
- pharmaceutically acceptable
- formula
- acceptable salt
- hcv
- Prior art date
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
Landscapes
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- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
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| US37139910P | 2010-08-06 | 2010-08-06 | |
| PCT/US2011/046285 WO2012018829A1 (en) | 2010-08-06 | 2011-08-02 | Combinations of hepatitis c virus inhibitors |
Publications (1)
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| SG187193A1 true SG187193A1 (en) | 2013-03-28 |
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| SG2014008346A SG2014008346A (en) | 2010-08-06 | 2011-08-02 | Combinations of hepatitis c virus inhibitors |
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| Application Number | Title | Priority Date | Filing Date |
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Country Status (14)
| Country | Link |
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| US (3) | US20120196794A1 (enExample) |
| EP (1) | EP2600835B1 (enExample) |
| JP (2) | JP6196154B2 (enExample) |
| KR (1) | KR101846596B1 (enExample) |
| CN (2) | CN103153280B (enExample) |
| AU (1) | AU2011285890B2 (enExample) |
| BR (1) | BR112013002922A2 (enExample) |
| CA (1) | CA2807589C (enExample) |
| EA (1) | EA022303B1 (enExample) |
| ES (1) | ES2685174T3 (enExample) |
| IL (1) | IL224369B (enExample) |
| MX (1) | MX2013001170A (enExample) |
| SG (2) | SG187193A1 (enExample) |
| WO (1) | WO2012018829A1 (enExample) |
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| US8329159B2 (en) | 2006-08-11 | 2012-12-11 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
| US20110269956A1 (en) | 2009-11-11 | 2011-11-03 | Bristol-Myers Squibb Company | Hepatitis C Virus Inhibitors |
| US20110274648A1 (en) | 2009-11-11 | 2011-11-10 | Bristol-Myers Squibb Company | Hepatitis C Virus Inhibitors |
| US20110281910A1 (en) | 2009-11-12 | 2011-11-17 | Bristol-Myers Squibb Company | Hepatitis C Virus Inhibitors |
| US8362020B2 (en) | 2009-12-30 | 2013-01-29 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
| US20120196794A1 (en) * | 2010-08-06 | 2012-08-02 | Bristol-Myers Squibb Company | Combinations of Hepatitis C Virus Inhibitors |
| BR112013004520A2 (pt) | 2010-08-26 | 2016-06-07 | Univ Emory | inibidores potentes e seletivos do virus da hepatite c |
| US8552047B2 (en) | 2011-02-07 | 2013-10-08 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
| US9243025B2 (en) * | 2011-03-31 | 2016-01-26 | Idenix Pharmaceuticals, Llc | Compounds and pharmaceutical compositions for the treatment of viral infections |
| US8957203B2 (en) | 2011-05-05 | 2015-02-17 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
| US9546160B2 (en) | 2011-05-12 | 2017-01-17 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
| US8691757B2 (en) | 2011-06-15 | 2014-04-08 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
| US8466159B2 (en) | 2011-10-21 | 2013-06-18 | Abbvie Inc. | Methods for treating HCV |
| US8492386B2 (en) | 2011-10-21 | 2013-07-23 | Abbvie Inc. | Methods for treating HCV |
| CN104023726A (zh) | 2011-10-21 | 2014-09-03 | 艾伯维公司 | 用于治疗hcv的一种或多种daa的联合治疗(例如，与abt-072或abt-333) |
| DE112012003510T5 (de) * | 2011-10-21 | 2015-03-19 | Abbvie Inc. | Verfahren zur Behandlung von HCV umfassend mindestens zwei direkt wirkende antivirale Wirkstoffe, Ribavirin aber nicht Interferon |
| US9326973B2 (en) | 2012-01-13 | 2016-05-03 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
| JP6154474B2 (ja) | 2012-10-19 | 2017-06-28 | ブリストル−マイヤーズ スクイブ カンパニーＢｒｉｓｔｏｌ−Ｍｙｅｒｓ Ｓｑｕｉｂｂ Ｃｏｍｐａｎｙ | Ｃ型肝炎ウイルス阻害剤 |
| EP2914613B1 (en) | 2012-11-02 | 2017-11-22 | Bristol-Myers Squibb Company | Hepatitis c virus inhibitors |
| WO2014071007A1 (en) | 2012-11-02 | 2014-05-08 | Bristol-Myers Squibb Company | Hepatitis c virus inhibitors |
| US9643999B2 (en) | 2012-11-02 | 2017-05-09 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
| EP2914614B1 (en) | 2012-11-05 | 2017-08-16 | Bristol-Myers Squibb Company | Hepatitis c virus inhibitors |
| EP2964664B1 (en) | 2013-03-07 | 2017-01-11 | Bristol-Myers Squibb Company | Hepatitis c virus inhibitors |
| US9717712B2 (en) | 2013-07-02 | 2017-08-01 | Bristol-Myers Squibb Company | Combinations comprising tricyclohexadecahexaene derivatives for use in the treatment of hepatitis C virus |
| US20150023913A1 (en) | 2013-07-02 | 2015-01-22 | Bristol-Myers Squibb Company | Hepatitis C Virus Inhibitors |
| JP2016527232A (ja) | 2013-07-17 | 2016-09-08 | ブリストル−マイヤーズ スクイブ カンパニーＢｒｉｓｔｏｌ−Ｍｙｅｒｓ Ｓｑｕｉｂｂ Ｃｏｍｐａｎｙ | Ｈｃｖの治療に使用するためのビフェニル誘導体を含む組み合わせ |
| US10617675B2 (en) | 2015-08-06 | 2020-04-14 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
| JP7129703B2 (ja) | 2016-04-28 | 2022-09-02 | エモリー ユニバーシティー | アルキン含有ヌクレオチド及びヌクレオシド治療組成物並びにそれらに関連した使用 |
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| US7456166B2 (en) * | 2006-05-17 | 2008-11-25 | Bristol-Myers Squibb Company | Cyclopropyl fused indolobenzazepine HCV NS5B inhibitors |
| US8329159B2 (en) * | 2006-08-11 | 2012-12-11 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
| WO2010042834A1 (en) * | 2008-10-09 | 2010-04-15 | Anadys Pharmaceuticals, Inc. | A method of inhibiting hepatitis c virus by combination of a 5,6-dihydro-1h-pyridin-2-one and one or more additional antiviral compounds |
| US8415374B2 (en) * | 2009-10-12 | 2013-04-09 | Bristol-Myers Squibb Company | Combinations of hepatitis C virus inhibitors |
| US20120196794A1 (en) * | 2010-08-06 | 2012-08-02 | Bristol-Myers Squibb Company | Combinations of Hepatitis C Virus Inhibitors |
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- 2011-08-02 CA CA2807589A patent/CA2807589C/en not_active Expired - Fee Related
- 2011-08-02 SG SG2014008346A patent/SG2014008346A/en unknown
- 2011-08-02 ES ES11815206.5T patent/ES2685174T3/es active Active
- 2011-08-02 KR KR1020137005628A patent/KR101846596B1/ko not_active Expired - Fee Related
- 2011-08-02 CN CN201510608270.5A patent/CN105148275A/zh active Pending
-
2013
- 2013-01-23 IL IL224369A patent/IL224369B/en not_active IP Right Cessation
-
2014
- 2014-04-28 US US14/263,101 patent/US20140235617A1/en not_active Abandoned
-
2015
- 2015-07-31 US US14/814,891 patent/US20150335655A1/en not_active Abandoned
-
2016
- 2016-03-31 JP JP2016072377A patent/JP2016155844A/ja not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| CN103153280B (zh) | 2015-09-09 |
| EA201390155A1 (ru) | 2013-05-30 |
| CA2807589A1 (en) | 2012-02-09 |
| AU2011285890B2 (en) | 2014-12-18 |
| ES2685174T3 (es) | 2018-10-05 |
| JP2016155844A (ja) | 2016-09-01 |
| JP6196154B2 (ja) | 2017-09-13 |
| MX2013001170A (es) | 2013-02-15 |
| IL224369B (en) | 2019-08-29 |
| US20120196794A1 (en) | 2012-08-02 |
| BR112013002922A2 (pt) | 2016-06-07 |
| CN103153280A (zh) | 2013-06-12 |
| KR20140002611A (ko) | 2014-01-08 |
| WO2012018829A1 (en) | 2012-02-09 |
| EP2600835A1 (en) | 2013-06-12 |
| SG2014008346A (en) | 2014-05-29 |
| CN105148275A (zh) | 2015-12-16 |
| JP2013535487A (ja) | 2013-09-12 |
| US20150335655A1 (en) | 2015-11-26 |
| EA022303B1 (ru) | 2015-12-30 |
| EP2600835A4 (en) | 2013-11-20 |
| KR101846596B1 (ko) | 2018-04-06 |
| AU2011285890A1 (en) | 2013-03-21 |
| CA2807589C (en) | 2016-08-30 |
| US20140235617A1 (en) | 2014-08-21 |
| EP2600835B1 (en) | 2018-05-30 |
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