SG11202107372QA - Modified release tablet formulations containing phosphodiesterase inhibitors - Google Patents

Modified release tablet formulations containing phosphodiesterase inhibitors

Info

Publication number
SG11202107372QA
SG11202107372QA SG11202107372QA SG11202107372QA SG11202107372QA SG 11202107372Q A SG11202107372Q A SG 11202107372QA SG 11202107372Q A SG11202107372Q A SG 11202107372QA SG 11202107372Q A SG11202107372Q A SG 11202107372QA SG 11202107372Q A SG11202107372Q A SG 11202107372QA
Authority
SG
Singapore
Prior art keywords
formulations containing
modified release
release tablet
phosphodiesterase inhibitors
tablet formulations
Prior art date
Application number
SG11202107372QA
Other languages
English (en)
Inventor
Marianne Rasmussen
Karin Green Høy
Carsten Ravn
Jari Pajander
Poul E Bertelsen
Gitte Pommergaard Pedersen
Original Assignee
Union Therapeutics As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Union Therapeutics As filed Critical Union Therapeutics As
Publication of SG11202107372QA publication Critical patent/SG11202107372QA/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4436Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a heterocyclic ring having sulfur as a ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Inorganic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Dermatology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
SG11202107372QA 2019-01-15 2020-01-14 Modified release tablet formulations containing phosphodiesterase inhibitors SG11202107372QA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP19151782 2019-01-15
PCT/EP2020/050798 WO2020148271A1 (fr) 2019-01-15 2020-01-14 Formulations de comprimés à libération modifiée contenant des inhibiteurs de phosphodiestérase

Publications (1)

Publication Number Publication Date
SG11202107372QA true SG11202107372QA (en) 2021-08-30

Family

ID=65030955

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11202107372QA SG11202107372QA (en) 2019-01-15 2020-01-14 Modified release tablet formulations containing phosphodiesterase inhibitors

Country Status (23)

Country Link
US (1) US20210386674A1 (fr)
EP (2) EP4282414A3 (fr)
JP (1) JP2022518703A (fr)
KR (1) KR20210117300A (fr)
CN (1) CN113423389A (fr)
AU (1) AU2020208761A1 (fr)
BR (1) BR112021013675A2 (fr)
CA (1) CA3125811A1 (fr)
DK (1) DK3911304T3 (fr)
EA (1) EA202191955A1 (fr)
ES (1) ES2957495T3 (fr)
FI (1) FI3911304T3 (fr)
HR (1) HRP20231127T1 (fr)
HU (1) HUE064539T2 (fr)
IL (1) IL284815A (fr)
LT (1) LT3911304T (fr)
MX (1) MX2021008536A (fr)
PL (1) PL3911304T3 (fr)
PT (1) PT3911304T (fr)
RS (1) RS64672B1 (fr)
SG (1) SG11202107372QA (fr)
SI (1) SI3911304T1 (fr)
WO (1) WO2020148271A1 (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL271399B (en) 2017-06-20 2022-07-01 Leo Pharma As Methods for the preparation of heterocyclic 3,1-benzodioxole compounds
EP3724196B9 (fr) 2017-12-15 2023-03-22 UNION therapeutics A/S Azétidine dihydrothiénopyridines substituées et leur utilisation en tant qu'inhibiteurs de phosphodiestérase
AU2022245186A1 (en) 2021-03-22 2023-10-05 UNION therapeutics A/S Treatment of hidradenitis suppurativa with orismilast
US11504332B2 (en) * 2021-03-23 2022-11-22 Vk Research Associates Inc. Phosphodiesterase-4 inhibitor combinations, methods of making, and methods of use thereof
GB202205715D0 (en) 2022-04-19 2022-06-01 Union Therapeutics As Treatment of neutrophilic dermatoses

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY121142A (en) * 1999-02-23 2005-12-30 Smithkline Beecham Corp Controlled release formulation for treating copd
US20050186276A1 (en) * 2003-07-17 2005-08-25 Pfizer Inc Pharmaceutical formulations
EP1937217A2 (fr) * 2005-09-13 2008-07-02 Elan Pharma International Limited Formulations nanoparticulaires de tadalafil
EP2266541A1 (fr) * 2009-06-18 2010-12-29 Krka Tovarna Zdravil, D.D., Novo Mesto Composition pharmaceutique solide comprenant du rivaroxaban
HUE044301T2 (hu) * 2010-06-24 2019-10-28 Leo Pharma As Benzodioxol-származékok, mint foszfodiészteráz inhibitorok
US20130218196A1 (en) * 2010-08-02 2013-08-22 Murdoch Childrens Research Institute An ischemia and reperfusion device
TW201613934A (en) 2014-06-23 2016-04-16 Leo Pharma As Methods for the preparation of 1,3-benzodioxole heterocyclic compounds
KR20180095888A (ko) 2015-12-18 2018-08-28 레오 파마 에이/에스 1,3-벤조디옥솔 복소환형 화합물의 제조 방법
IL271399B (en) 2017-06-20 2022-07-01 Leo Pharma As Methods for the preparation of heterocyclic 3,1-benzodioxole compounds

Also Published As

Publication number Publication date
EP3911304B1 (fr) 2023-09-06
EP4282414A3 (fr) 2024-02-21
PL3911304T3 (pl) 2023-12-04
CA3125811A1 (fr) 2020-07-23
WO2020148271A1 (fr) 2020-07-23
EP3911304A1 (fr) 2021-11-24
AU2020208761A1 (en) 2021-08-19
LT3911304T (lt) 2023-11-10
BR112021013675A2 (pt) 2021-09-14
HUE064539T2 (hu) 2024-03-28
KR20210117300A (ko) 2021-09-28
HRP20231127T1 (hr) 2024-01-05
RS64672B1 (sr) 2023-11-30
EP4282414A2 (fr) 2023-11-29
CN113423389A (zh) 2021-09-21
US20210386674A1 (en) 2021-12-16
JP2022518703A (ja) 2022-03-16
FI3911304T3 (fi) 2023-09-25
IL284815A (en) 2021-08-31
EA202191955A1 (ru) 2021-10-07
MX2021008536A (es) 2021-11-12
ES2957495T3 (es) 2024-01-19
SI3911304T1 (sl) 2023-12-29
DK3911304T3 (da) 2023-10-02
PT3911304T (pt) 2023-09-28

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