SG11202008543RA - Pyrrolidineamide derivatives and uses thereof - Google Patents

Pyrrolidineamide derivatives and uses thereof

Info

Publication number
SG11202008543RA
SG11202008543RA SG11202008543RA SG11202008543RA SG11202008543RA SG 11202008543R A SG11202008543R A SG 11202008543RA SG 11202008543R A SG11202008543R A SG 11202008543RA SG 11202008543R A SG11202008543R A SG 11202008543RA SG 11202008543R A SG11202008543R A SG 11202008543RA
Authority
SG
Singapore
Prior art keywords
pyrrolidineamide
derivatives
pyrrolidineamide derivatives
Prior art date
Application number
SG11202008543RA
Other languages
English (en)
Inventor
Chuanfei Jin
Kangzhi Chen
Yingjun Zhang
Original Assignee
Sunshine Lake Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sunshine Lake Pharma Co Ltd filed Critical Sunshine Lake Pharma Co Ltd
Publication of SG11202008543RA publication Critical patent/SG11202008543RA/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • C07D207/09Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/427Thiazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychology (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Vascular Medicine (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Urology & Nephrology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
SG11202008543RA 2018-03-08 2019-03-07 Pyrrolidineamide derivatives and uses thereof SG11202008543RA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CN201810192198 2018-03-08
PCT/CN2019/077249 WO2019170115A1 (en) 2018-03-08 2019-03-07 Pyrrolidineamide derivatives and uses thereof

Publications (1)

Publication Number Publication Date
SG11202008543RA true SG11202008543RA (en) 2020-10-29

Family

ID=67845842

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11202008543RA SG11202008543RA (en) 2018-03-08 2019-03-07 Pyrrolidineamide derivatives and uses thereof

Country Status (8)

Country Link
US (1) US11225460B2 (https=)
EP (1) EP3762364B1 (https=)
JP (1) JP7405756B2 (https=)
CN (1) CN110240557B (https=)
AU (1) AU2019230883B2 (https=)
CA (1) CA3092747A1 (https=)
SG (1) SG11202008543RA (https=)
WO (1) WO2019170115A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20240317681A1 (en) * 2020-07-07 2024-09-26 Sunshine Lake Pharma Co., Ltd. Pyrrolidine amide derivative salt and use thereof
CN113896671B (zh) * 2020-07-07 2023-06-09 广东东阳光药业有限公司 吡咯烷酰胺衍生物的盐及其用途
CN113896670B (zh) * 2020-07-07 2023-06-09 广东东阳光药业有限公司 吡咯烷酰胺衍生物的盐及其用途
CN114573491B (zh) * 2020-12-01 2023-12-08 广东东阳光药业股份有限公司 吡咯烷酰胺衍生物的制备方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL94466A (en) 1989-05-25 1995-01-24 Erba Carlo Spa Pharmaceutical preparations containing the history of A-amino carboxamide N-phenylalkyl are converted into such new compounds and their preparation
WO2000033788A2 (en) 1998-12-11 2000-06-15 American Biogenetic Sciences Inc. Substituted nitrogen heterocyclic compounds and therapeutic uses thereof
FR2799461B1 (fr) 1999-10-11 2002-01-04 Sod Conseils Rech Applic Derives d'heterocycles a 5 chainons, leur preparation et leur application a titre de medicaments
MY134480A (en) * 2002-09-20 2007-12-31 Hoffmann La Roche 4-pyrrolidino-phenyl-benzyl ether derivatives
EP1524265A1 (en) * 2003-10-15 2005-04-20 Newron Pharmaceuticals S.p.A. Prolinamide derivatives as sodium and/or calcium channel blockers or selective MAO-B inhibitors
WO2006013049A2 (en) * 2004-08-02 2006-02-09 F.Hoffmann-La Roche Ag Benzyloxy derivatives as maob inhibitors
US7501528B2 (en) 2005-03-15 2009-03-10 Hoffmann-La Roche Inc. Method for preparing enantiomerically pure 4-pyrrolidino phenylbenzyl ether derivatives
US20070078172A1 (en) 2005-06-16 2007-04-05 Jenrin Discovery Mao-b inhibitors useful for treating obesity
BRPI0821026A2 (pt) 2007-12-19 2015-06-16 Newron Pharmaceutical S P A Derivados de alfa-minoamidas úteis no tratamento de transtornos psiquiátricos
CA2886904A1 (en) * 2012-10-02 2014-04-10 Cyril Montagne Pyrrolidines
EP3601255A1 (en) 2017-03-21 2020-02-05 AbbVie Deutschland GmbH & Co. KG Proline amide compounds and their azetidine analogues carrying a specifically substituted benzyl radical

Also Published As

Publication number Publication date
CN110240557A (zh) 2019-09-17
WO2019170115A1 (en) 2019-09-12
CN110240557B (zh) 2023-05-09
AU2019230883A1 (en) 2020-09-24
EP3762364A1 (en) 2021-01-13
JP7405756B2 (ja) 2023-12-26
US20210053918A1 (en) 2021-02-25
AU2019230883B2 (en) 2024-02-01
JP2021515019A (ja) 2021-06-17
EP3762364B1 (en) 2023-08-23
US11225460B2 (en) 2022-01-18
CA3092747A1 (en) 2019-09-12
EP3762364A4 (en) 2021-08-04

Similar Documents

Publication Publication Date Title
IL278171A (en) Glucose-dependent insulin polypeptide and its uses
ZA202001340B (en) Heterocyclic compound and use thereof
IL273236A (en) Pyrazolopyrimidine compounds and their uses
IL294052B2 (en) Fluoroalkyl oxadiazoles and their uses
IL283533A (en) Pentatein derivatives and their uses
IL277502A (en) Compounds and uses for them
IL278973A (en) New benzodiazepine histories and uses
IL272808B (en) Pyridineamine-pyridone and pyrimidineamine-pyridone compounds
GB2577419B (en) Lipo-glycopeptide cleavable derivatives and uses thereof
IL279441A (en) History of N-converted tetrahydrothinopyridines and their uses
IL269836B (en) Converted N-arylethyl-2-aminoquinoline-4-carboxamides and their use
GB201801102D0 (en) New compounds and uses
IL287503A (en) Thio-semicarbazide compounds and their use
IL279483A (en) Cyanotriazole compounds and their uses
SG11202008543RA (en) Pyrrolidineamide derivatives and uses thereof
IL292482B1 (en) Azaindolylpyridone and diazaindolylpyridone compounds
IL282527A (en) 5-Azaindazole history and their use
IL282526A (en) 5-Azaindazole history and their use
SG11202010985TA (en) Heterocyclic derivatives and use thereof
SG11202103533UA (en) Alkoxybenzaldehyde derivatives and precursors thereof
IL275211A (en) Fast and flexible segment chains - division
GB201700404D0 (en) Compounds and composistions
IL280369A (en) Myokines and their uses
IL269843B (en) Converted N-arylethyl-2-arylquinoline-4-carboxamides and their use
GB201806349D0 (en) New compounds and uses