SG11201605790VA - Antimicrobial peptidomimetics - Google Patents

Antimicrobial peptidomimetics

Info

Publication number
SG11201605790VA
SG11201605790VA SG11201605790VA SG11201605790VA SG11201605790VA SG 11201605790V A SG11201605790V A SG 11201605790VA SG 11201605790V A SG11201605790V A SG 11201605790VA SG 11201605790V A SG11201605790V A SG 11201605790VA SG 11201605790V A SG11201605790V A SG 11201605790VA
Authority
SG
Singapore
Prior art keywords
peptidomimetics
antimicrobial
antimicrobial peptidomimetics
Prior art date
Application number
SG11201605790VA
Other languages
English (en)
Inventor
Brian Cheng San Chia
Original Assignee
Agency Science Tech & Res
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB1401036.7A external-priority patent/GB2522412A/en
Application filed by Agency Science Tech & Res filed Critical Agency Science Tech & Res
Priority to SG11201605790VA priority Critical patent/SG11201605790VA/en
Publication of SG11201605790VA publication Critical patent/SG11201605790VA/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0802—Tripeptides with the first amino acid being neutral
    • C07K5/0812—Tripeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
    • C07K1/061—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/10—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using coupling agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/0212—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -N-C-N-C(=0)-, e.g. retro-inverso peptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06086—Dipeptides with the first amino acid being basic
    • C07K5/06095—Arg-amino acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1024—Tetrapeptides with the first amino acid being heterocyclic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Analytical Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
SG11201605790VA 2014-01-22 2015-01-22 Antimicrobial peptidomimetics SG11201605790VA (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
SG11201605790VA SG11201605790VA (en) 2014-01-22 2015-01-22 Antimicrobial peptidomimetics

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB1401036.7A GB2522412A (en) 2014-01-22 2014-01-22 Antimicrobial peptidomimetics
SG10201406683W 2014-10-16
SG11201605790VA SG11201605790VA (en) 2014-01-22 2015-01-22 Antimicrobial peptidomimetics
PCT/SG2015/050006 WO2015112093A2 (en) 2014-01-22 2015-01-22 Antimicrobial peptidomimetics

Publications (1)

Publication Number Publication Date
SG11201605790VA true SG11201605790VA (en) 2016-08-30

Family

ID=53682081

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201605790VA SG11201605790VA (en) 2014-01-22 2015-01-22 Antimicrobial peptidomimetics

Country Status (6)

Country Link
US (2) US10053490B2 (ja)
EP (1) EP3071591B1 (ja)
JP (1) JP6516758B2 (ja)
CN (1) CN105934440A (ja)
SG (1) SG11201605790VA (ja)
WO (1) WO2015112093A2 (ja)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP6516758B2 (ja) 2014-01-22 2019-05-22 エイジェンシー・フォー・サイエンス，テクノロジー・アンド・リサーチ 抗菌ペプチド模倣物
US20200157144A1 (en) * 2017-08-01 2020-05-21 Agency For Science, Technology And Research Antimicrobial peptidomimetics
CN107540574B (zh) * 2017-09-19 2021-06-11 成都西岭源药业有限公司 R-联苯丙氨醇的制备方法

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5776939A (en) * 1997-06-12 1998-07-07 Eli Lilly And Company Drug resistance and multidrug resistance modulators
GB0005703D0 (en) * 2000-03-09 2000-05-03 Alpharma As Compounds
US6600015B2 (en) 2000-04-04 2003-07-29 Hoffmann-La Roche Inc. Selective linear peptides with melanocortin-4 receptor (MC4-R) agonist activity
US6699997B2 (en) * 2000-06-28 2004-03-02 Teva Pharmaceutical Industries Ltd. Carvedilol
US20060128614A1 (en) 2002-09-20 2006-06-15 Jya-Wei Cheng Antimicrobial peptides with reduced hemolysis and methods of their use
JP4931604B2 (ja) * 2004-01-23 2012-05-16 コーネル リサーチ ファウンデイション インコーポレイテッド 酸化的損傷を低減する方法
EP2019819A4 (en) * 2006-05-09 2011-01-19 Neobiotics Ab INNOVATIVE PEPTIDE DERIVATIVES AS ANTIMICROBIAL AGENTS FOR THE TREATMENT OF INJURIES
JP2008063285A (ja) * 2006-09-08 2008-03-21 Univ Nagoya 高親和性ペプチドの設計法及び調製法、並びに高親和性ペプチド
WO2009145839A1 (en) * 2008-04-04 2009-12-03 Government Of The United States Of America, As Represented By The Secretary, Department Of Health And Human Services Polyamine compounds that bind tar rna of hiv and methods of treating viral disorders
GB0818074D0 (en) * 2008-10-02 2008-11-05 Lytix Biopharma As Treatment of biofilms
DE102009035593A1 (de) 2008-10-29 2010-05-06 Philipps-Universität Marburg N-terminal modifizierte Tetrapeptidderivate mit C-terminalem Argininmetikum
US20120083452A1 (en) * 2010-09-30 2012-04-05 Perricone Nicholas V Topical Anesthetic Uses of Szeto-Schiller Peptides
EP2625192A1 (en) * 2010-10-08 2013-08-14 Solvay Sa A bioactive amino acid sequence and use therefrom
US20150118315A1 (en) * 2011-06-14 2015-04-30 Stealth Peptides International, Inc. Aromatic-cationic peptides and uses of same
EP2788013A4 (en) * 2011-12-09 2015-08-19 Stealth Peptides Int Inc AROMATIC-CATIONIC PEPTIDES AND USES THEREOF
WO2013138666A1 (en) * 2012-03-16 2013-09-19 Sanford-Burnham Medical Research Institute Inhibitors of furin and other pro-protein convertases
JP6516758B2 (ja) 2014-01-22 2019-05-22 エイジェンシー・フォー・サイエンス，テクノロジー・アンド・リサーチ 抗菌ペプチド模倣物

Also Published As

Publication number Publication date
US10053490B2 (en) 2018-08-21
WO2015112093A2 (en) 2015-07-30
EP3071591A4 (en) 2017-08-16
US20160333048A1 (en) 2016-11-17
JP6516758B2 (ja) 2019-05-22
CN105934440A (zh) 2016-09-07
WO2015112093A3 (en) 2015-11-26
EP3071591A2 (en) 2016-09-28
US10787483B2 (en) 2020-09-29
JP2017507916A (ja) 2017-03-23
EP3071591B1 (en) 2021-05-05
US20180354989A1 (en) 2018-12-13

Similar Documents

Publication Publication Date Title
GB2540054B (en) Antimicrobial compositions
IL253087A0 (en) Antimicrobial preparation
LT3226858T (lt) Imidazolo pagrindo antimikrobiniai agentai
ZA201606715B (en) Antibacterial compounds
GB201412238D0 (en) Compound
GB201402267D0 (en) Antibacterial agents
IL248987B (en) Antimicrobial liquid
ZA201703686B (en) Antimicrobial cover
IL250405A0 (en) Antibacterial sideromycins
SG11201605790VA (en) Antimicrobial peptidomimetics
GB2528521B (en) Novel antimicrobial peptides
GB201405891D0 (en) Modified antimicrobial peptides
GB201403268D0 (en) Antimicrobial surface
GB201504305D0 (en) An antimicrobial maeterial
GB2524077B (en) Aperture protector
GB201401036D0 (en) Antimicrobial peptidomimetics
PL3393242T3 (pl) Preparat antybakteryjny
GB2552572B (en) Antimicrobial compositions
GB201401445D0 (en) Antimicrobial compound
GB201417939D0 (en) Antibacterial compounds
GB201417941D0 (en) Antibacterial compounds
PL2939524T3 (pl) Maszyna żniwna
AU2014324V (en) MALOF002 Acmena smithii
GB201414205D0 (en) Antibacterial compounds
GB201419176D0 (en) Attachment arrangement