SE447482B - Forfarande for framstellning av somatostatinanaloger - Google Patents

Forfarande for framstellning av somatostatinanaloger

Info

Publication number
SE447482B
SE447482B SE7802015A SE7802015A SE447482B SE 447482 B SE447482 B SE 447482B SE 7802015 A SE7802015 A SE 7802015A SE 7802015 A SE7802015 A SE 7802015A SE 447482 B SE447482 B SE 447482B
Authority
SE
Sweden
Prior art keywords
phe
thr
boc
cys
group
Prior art date
Application number
SE7802015A
Other languages
English (en)
Swedish (sv)
Other versions
SE7802015L (sv
Inventor
D Sarantakis
Original Assignee
American Home Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/778,517 external-priority patent/US4077952A/en
Priority claimed from US05/830,930 external-priority patent/US4104267A/en
Priority claimed from US05/864,173 external-priority patent/US4190575A/en
Application filed by American Home Prod filed Critical American Home Prod
Publication of SE7802015L publication Critical patent/SE7802015L/xx
Publication of SE447482B publication Critical patent/SE447482B/sv

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1002—Tetrapeptides with the first amino acid being neutral
    • C07K5/1005—Tetrapeptides with the first amino acid being neutral and aliphatic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/655—Somatostatins
    • C07K14/6555—Somatostatins at least 1 amino acid in D-form
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Endocrinology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Emergency Medicine (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Toxicology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
SE7802015A 1977-02-22 1978-02-21 Forfarande for framstellning av somatostatinanaloger SE447482B (sv)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US77095377A 1977-02-22 1977-02-22
US05/778,517 US4077952A (en) 1977-03-17 1977-03-17 Somatostatin analogs
US05/830,930 US4104267A (en) 1977-02-22 1977-09-06 Somatostatin analogs
GB4047177 1977-09-29
US05/864,173 US4190575A (en) 1977-12-27 1977-12-27 Polypeptides related to somatostatin

Publications (2)

Publication Number Publication Date
SE7802015L SE7802015L (sv) 1978-10-16
SE447482B true SE447482B (sv) 1986-11-17

Family

ID=27516344

Family Applications (1)

Application Number Title Priority Date Filing Date
SE7802015A SE447482B (sv) 1977-02-22 1978-02-21 Forfarande for framstellning av somatostatinanaloger

Country Status (5)

Country Link
DE (1) DE2807403A1 (da)
DK (1) DK150618C (da)
FR (1) FR2382433A1 (da)
IE (1) IE46462B1 (da)
SE (1) SE447482B (da)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE7810156L (sv) * 1977-12-13 1979-06-14 American Home Prod Somatostatinanaloger
LU80207A1 (de) * 1978-09-07 1980-04-21 H Kalbacher Neue substituierte kohlensaeureester und urethane,verfahren zu ihrer herstellung und deren verwendung
US4225472A (en) * 1979-05-29 1980-09-30 American Home Products Corporation Truncated somatostatin analogs

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4061608A (en) * 1976-07-13 1977-12-06 American Home Products Corporation Arg 4 -somatostatin and analogues thereof

Also Published As

Publication number Publication date
IE46462B1 (en) 1983-06-15
DE2807403C2 (da) 1990-11-29
DE2807403A1 (de) 1978-08-31
DK150618B (da) 1987-04-21
FR2382433A1 (fr) 1978-09-29
IE780348L (en) 1978-08-22
SE7802015L (sv) 1978-10-16
DK76378A (da) 1978-08-23
FR2382433B1 (da) 1983-12-09
DK150618C (da) 1987-10-19

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