SE435291B - PROCEDURE FOR PREPARING 7-ACYLAMINO-3 (1- (2-SULFAMINOETHYL) -TETRAZOL-5-YLTIOMETHYL) -3-CEFEM-4-CARBONIC ACID - Google Patents

PROCEDURE FOR PREPARING 7-ACYLAMINO-3 (1- (2-SULFAMINOETHYL) -TETRAZOL-5-YLTIOMETHYL) -3-CEFEM-4-CARBONIC ACID

Info

Publication number
SE435291B
SE435291B SE7610722A SE7610722A SE435291B SE 435291 B SE435291 B SE 435291B SE 7610722 A SE7610722 A SE 7610722A SE 7610722 A SE7610722 A SE 7610722A SE 435291 B SE435291 B SE 435291B
Authority
SE
Sweden
Prior art keywords
yltiomethyl
sulfaminoethyl
cefem
tetrazol
acylamino
Prior art date
Application number
SE7610722A
Other languages
Swedish (sv)
Other versions
SE7610722L (en
Inventor
D A Berges
Original Assignee
Smithkline Beckman Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/704,142 external-priority patent/US4118491A/en
Application filed by Smithkline Beckman Corp filed Critical Smithkline Beckman Corp
Publication of SE7610722L publication Critical patent/SE7610722L/en
Publication of SE435291B publication Critical patent/SE435291B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04—Five-membered rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36—Methylene radicals, substituted by sulfur atoms
SE7610722A 1975-10-30 1976-09-28 PROCEDURE FOR PREPARING 7-ACYLAMINO-3 (1- (2-SULFAMINOETHYL) -TETRAZOL-5-YLTIOMETHYL) -3-CEFEM-4-CARBONIC ACID SE435291B (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US62716475A 1975-10-30 1975-10-30
US66583776A 1976-03-11 1976-03-11
US05/704,142 US4118491A (en) 1976-03-11 1976-07-12 7-Acyl-3-(sulfaminoalkyl substituted tetrazolylthiomethyl)cephalosporins, antibacterial compositions containing them and methods of treating bacterial infections with them

Publications (2)

Publication Number Publication Date
SE7610722L SE7610722L (en) 1977-05-01
SE435291B true SE435291B (en) 1984-09-17

Family

ID=27417417

Family Applications (3)

Application Number Title Priority Date Filing Date
SE8006413A SE452621B (en) 1975-10-30 1976-09-28 7-AMINO CEPHALOSPORINE DERIVATIVES FOR USE AS INTERMEDIATE PRODUCTS FOR THE PREPARATION OF SIMILAR 7-SUBSTITUTED CEPHALOSPORINE DERIVATIVES
SE7610722A SE435291B (en) 1975-10-30 1976-09-28 PROCEDURE FOR PREPARING 7-ACYLAMINO-3 (1- (2-SULFAMINOETHYL) -TETRAZOL-5-YLTIOMETHYL) -3-CEFEM-4-CARBONIC ACID
SE8006414A SE437025B (en) 1975-10-30 1980-09-12 1- (2-SULFAMINOETHYL) -TETRAZOL-5-THIOL USED FOR THE PREPARATION OF CEPHALOSPORINE COMPOUNDS WITH ANTIBACTERIAL ACTIVITY

Family Applications Before (1)

Application Number Title Priority Date Filing Date
SE8006413A SE452621B (en) 1975-10-30 1976-09-28 7-AMINO CEPHALOSPORINE DERIVATIVES FOR USE AS INTERMEDIATE PRODUCTS FOR THE PREPARATION OF SIMILAR 7-SUBSTITUTED CEPHALOSPORINE DERIVATIVES

Family Applications After (1)

Application Number Title Priority Date Filing Date
SE8006414A SE437025B (en) 1975-10-30 1980-09-12 1- (2-SULFAMINOETHYL) -TETRAZOL-5-THIOL USED FOR THE PREPARATION OF CEPHALOSPORINE COMPOUNDS WITH ANTIBACTERIAL ACTIVITY

Country Status (17)

Country Link
JP (1) JPS6053026B2 (en)
AT (1) AT353957B (en)
AU (1) AU505141B2 (en)
CA (1) CA1071188A (en)
CH (1) CH627757A5 (en)
DE (1) DE2649545A1 (en)
DK (1) DK463176A (en)
ES (1) ES452769A1 (en)
FI (1) FI60868C (en)
FR (3) FR2361896A1 (en)
GB (3) GB1570095A (en)
GR (1) GR61667B (en)
IE (1) IE44393B1 (en)
IL (3) IL50546A (en)
LU (1) LU76092A1 (en)
NL (1) NL7612010A (en)
SE (3) SE452621B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4117123A (en) * 1977-06-09 1978-09-26 Smithkline Corporation 7-Acylamino-3-[1-(2-sulfamidoethyl)tetrazol-5-ylthiomethyl]-3-cephem-4-carboxylic acids
AT383811B (en) * 1983-09-22 1987-08-25 Biochemie Gmbh Process for the preparation of monoalkali metal salts of 7-amino-3-cephem-4-carboxylic acid derivatives
US4717531A (en) * 1983-09-23 1988-01-05 Westinghouse Electric Corp. Fuel transfer system upender using translation drive

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR207752A1 (en) * 1973-03-30 1976-10-29 Fujisawa Pharmaceutical Co PROCEDURE FOR OBTAINING 7-AMINO-SUBSTITUTED-3-THIOMETHYL SUBSTITUTED-3-CEFEM-4-CARBOXYL ACIDS
NL7414119A (en) * 1973-10-31 1975-05-02 Fujisawa Pharmaceutical Co PROCESS FOR PREPARING 1H-TETRAZOL-5-THIOL DERIVATIVES AND 1-SUBSTITUATED 1H-TETRAZOL-5-THIOLS.
GB1449420A (en) * 1973-11-26 1976-09-15 Sankyo Co 7alpha-methoxycephalosporing derivatives
NZ176206A (en) * 1973-12-25 1978-03-06 Takeda Chemical Industries Ltd Cephalosporins
US4066762A (en) * 1976-07-12 1978-01-03 Smithkline Corporation Derivatives of 7-(2-substituted-2-hydroxyiminoacetamido)-3-(1-substituted tetrazol-5-ylthiomethyl-3-cephem-4-carboxylic acid

Also Published As

Publication number Publication date
IE44393L (en) 1977-09-11
FR2337720A1 (en) 1977-08-05
GB1570094A (en) 1980-06-25
FI60868C (en) 1982-04-13
AU505141B2 (en) 1979-11-08
SE8006413L (en) 1980-09-12
FI60868B (en) 1981-12-31
FR2351982B1 (en) 1981-07-03
LU76092A1 (en) 1977-05-17
GB1570093A (en) 1980-06-25
GR61667B (en) 1978-12-05
IE44393B1 (en) 1981-11-18
SE437025B (en) 1985-02-04
AU1870276A (en) 1978-04-20
SE7610722L (en) 1977-05-01
GB1570095A (en) 1980-06-25
SE452621B (en) 1987-12-07
CA1071188A (en) 1980-02-05
ES452769A1 (en) 1978-01-16
FR2337720B1 (en) 1981-07-10
NL7612010A (en) 1977-05-03
SE8006414L (en) 1980-09-12
JPS5257191A (en) 1977-05-11
FR2361896A1 (en) 1978-03-17
DE2649545A1 (en) 1977-05-12
FI763044A (en) 1977-05-01
JPS6053026B2 (en) 1985-11-22
FR2361896B1 (en) 1979-02-23
IL50546A0 (en) 1976-11-30
IL50546A (en) 1980-07-31
FR2351982A1 (en) 1977-12-16
IL56757A0 (en) 1979-05-31
IL56758A0 (en) 1979-05-31
ATA807276A (en) 1979-05-15
CH627757A5 (en) 1982-01-29
AT353957B (en) 1979-12-10
DK463176A (en) 1977-05-01

Similar Documents

Publication Publication Date Title
SE442295B (en) PROCEDURE FOR PREPARING 4-AMINO-5-EN-HEXANIC ACID
SE434394B (en) ANALOGY PROCEDURE FOR PREPARING QUINOLONALKANIC ACID DERIVATIVES
SE420199B (en) PROCEDURE FOR PREPARING 16-OXIDATED PROSTANIC ACID DERIVATIVES
SE429970B (en) PROCEDURE FOR PREPARING GLUCOPYRANOSIDO-1,6-MANNIT
SE436572B (en) PROCEDURE FOR PREPARING ANDROSTADIEN-17-CARBONIC ACID ESTERS
SE431089B (en) PROCEDURE FOR PREPARING BETA-METYLTIO-PROPIONAL HEAD
SE441360B (en) PROCEDURE FOR PREPARING PHOSPHONIC ACID DERIVATIVES
SE434057B (en) PROCEDURE FOR PREPARING NEW RIFAMYCINE COMPOUNDS
SE431652B (en) PROCEDURE FOR PREPARING 7BETA-AMINO-3CEFEM-3OL-4-CARBOXYLIC ACID DERIVATIVES
SE433745B (en) PROCEDURE FOR PREPARING TETRAHYDROISOKINOLIN DERIVATIVES
SE7802609L (en) PROCEDURE FOR PREPARING 1-AZAXANTONE-3-CARBOXYLIC ACID DERIVATIVE
SE416479B (en) PROCEDURE FOR PREPARING HOGRENA ALKOLYMETHALOGENIC CRYSTALS
SE7613768L (en) PROCEDURE FOR PREPARING PENICILLINES
SE428296B (en) ANALOGY PROCEDURE FOR PREPARING SUBSTITUTED DIPHONYL SULPHIDS
NO141050C (en) PROCEDURE FOR PREPARING 5-FLUORO-2-METHYL-1- (P-METHYLSULPHINYLBENZYLIDE) -IND-2-EN-3-YL-ACETIC ACID
NO821484L (en) PROCEDURE FOR PREPARING PHOSPHONIC ACID DERIVATIVES
SE420093B (en) PROCEDURE FOR PREPARING 5-PHENYL-2-FURAMIDOXIMER
SE434157B (en) PROCEDURE FOR PREPARING 6-AMINOPENICILLANIC ACID
IT1068946B (en) PROCEDURE FOR PREPARING TRIEMTYL HYDROKINONE
SE435291B (en) PROCEDURE FOR PREPARING 7-ACYLAMINO-3 (1- (2-SULFAMINOETHYL) -TETRAZOL-5-YLTIOMETHYL) -3-CEFEM-4-CARBONIC ACID
NO142121C (en) PROCEDURE FOR PREPARING ACID PROPERTY SOLUTIONS
SE427184B (en) PROCEDURE FOR PREPARING 7-AMINOCEPHALOSPORANIC ACID DERIVATIVES
SE414927B (en) PROCEDURE FOR PREPARING 1-METHYL-2- (PHENYLOXIMETHYL) -5-NITROIMIDAZOLES
SE428689B (en) PROCEDURE FOR PREPARING AROYL-PHENYL AGREEMENT COMPOUNDS
SE7607026L (en) PROCEDURE FOR THE PREPARATION OF 5-ALKYLPICOLIC ACID

Legal Events

Date Code Title Description
NUG Patent has lapsed

Ref document number: 7610722-6

Effective date: 19880622

Format of ref document f/p: F