NL7612010A - PROCESS FOR THE PREPARATION OF CEPHALOSPORIN COMPOUNDS AND PHARMACEUTICAL MIXTURES CONTAINING THESE COMPOUNDS. - Google Patents

PROCESS FOR THE PREPARATION OF CEPHALOSPORIN COMPOUNDS AND PHARMACEUTICAL MIXTURES CONTAINING THESE COMPOUNDS.

Info

Publication number
NL7612010A
NL7612010A NL7612010A NL7612010A NL7612010A NL 7612010 A NL7612010 A NL 7612010A NL 7612010 A NL7612010 A NL 7612010A NL 7612010 A NL7612010 A NL 7612010A NL 7612010 A NL7612010 A NL 7612010A
Authority
NL
Netherlands
Prior art keywords
compounds
preparation
mixtures containing
cephalosporin
pharmaceutical mixtures
Prior art date
Application number
NL7612010A
Other languages
Dutch (nl)
Original Assignee
Smithkline Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/704,142 external-priority patent/US4118491A/en
Application filed by Smithkline Corp filed Critical Smithkline Corp
Publication of NL7612010A publication Critical patent/NL7612010A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D257/00Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04Five-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/247-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36Methylene radicals, substituted by sulfur atoms
NL7612010A 1975-10-30 1976-10-29 PROCESS FOR THE PREPARATION OF CEPHALOSPORIN COMPOUNDS AND PHARMACEUTICAL MIXTURES CONTAINING THESE COMPOUNDS. NL7612010A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US62716475A 1975-10-30 1975-10-30
US66583776A 1976-03-11 1976-03-11
US05/704,142 US4118491A (en) 1976-03-11 1976-07-12 7-Acyl-3-(sulfaminoalkyl substituted tetrazolylthiomethyl)cephalosporins, antibacterial compositions containing them and methods of treating bacterial infections with them

Publications (1)

Publication Number Publication Date
NL7612010A true NL7612010A (en) 1977-05-03

Family

ID=27417417

Family Applications (1)

Application Number Title Priority Date Filing Date
NL7612010A NL7612010A (en) 1975-10-30 1976-10-29 PROCESS FOR THE PREPARATION OF CEPHALOSPORIN COMPOUNDS AND PHARMACEUTICAL MIXTURES CONTAINING THESE COMPOUNDS.

Country Status (17)

Country Link
JP (1) JPS6053026B2 (en)
AT (1) AT353957B (en)
AU (1) AU505141B2 (en)
CA (1) CA1071188A (en)
CH (1) CH627757A5 (en)
DE (1) DE2649545A1 (en)
DK (1) DK463176A (en)
ES (1) ES452769A1 (en)
FI (1) FI60868C (en)
FR (3) FR2361896A1 (en)
GB (3) GB1570095A (en)
GR (1) GR61667B (en)
IE (1) IE44393B1 (en)
IL (3) IL50546A (en)
LU (1) LU76092A1 (en)
NL (1) NL7612010A (en)
SE (3) SE452621B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4117123A (en) * 1977-06-09 1978-09-26 Smithkline Corporation 7-Acylamino-3-[1-(2-sulfamidoethyl)tetrazol-5-ylthiomethyl]-3-cephem-4-carboxylic acids
AT383811B (en) * 1983-09-22 1987-08-25 Biochemie Gmbh Process for the preparation of monoalkali metal salts of 7-amino-3-cephem-4-carboxylic acid derivatives
US4717531A (en) * 1983-09-23 1988-01-05 Westinghouse Electric Corp. Fuel transfer system upender using translation drive

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR207752A1 (en) * 1973-03-30 1976-10-29 Fujisawa Pharmaceutical Co PROCEDURE FOR OBTAINING 7-AMINO-SUBSTITUTED-3-THIOMETHYL SUBSTITUTED-3-CEFEM-4-CARBOXYL ACIDS
NL7414119A (en) * 1973-10-31 1975-05-02 Fujisawa Pharmaceutical Co PROCESS FOR PREPARING 1H-TETRAZOL-5-THIOL DERIVATIVES AND 1-SUBSTITUATED 1H-TETRAZOL-5-THIOLS.
GB1449420A (en) * 1973-11-26 1976-09-15 Sankyo Co 7alpha-methoxycephalosporing derivatives
NZ176206A (en) * 1973-12-25 1978-03-06 Takeda Chemical Industries Ltd Cephalosporins
US4066762A (en) * 1976-07-12 1978-01-03 Smithkline Corporation Derivatives of 7-(2-substituted-2-hydroxyiminoacetamido)-3-(1-substituted tetrazol-5-ylthiomethyl-3-cephem-4-carboxylic acid

Also Published As

Publication number Publication date
IE44393L (en) 1977-09-11
FR2337720A1 (en) 1977-08-05
GB1570094A (en) 1980-06-25
FI60868C (en) 1982-04-13
AU505141B2 (en) 1979-11-08
SE8006413L (en) 1980-09-12
FI60868B (en) 1981-12-31
FR2351982B1 (en) 1981-07-03
LU76092A1 (en) 1977-05-17
GB1570093A (en) 1980-06-25
GR61667B (en) 1978-12-05
IE44393B1 (en) 1981-11-18
SE437025B (en) 1985-02-04
AU1870276A (en) 1978-04-20
SE7610722L (en) 1977-05-01
GB1570095A (en) 1980-06-25
SE452621B (en) 1987-12-07
CA1071188A (en) 1980-02-05
ES452769A1 (en) 1978-01-16
FR2337720B1 (en) 1981-07-10
SE8006414L (en) 1980-09-12
JPS5257191A (en) 1977-05-11
FR2361896A1 (en) 1978-03-17
DE2649545A1 (en) 1977-05-12
SE435291B (en) 1984-09-17
FI763044A (en) 1977-05-01
JPS6053026B2 (en) 1985-11-22
FR2361896B1 (en) 1979-02-23
IL50546A0 (en) 1976-11-30
IL50546A (en) 1980-07-31
FR2351982A1 (en) 1977-12-16
IL56757A0 (en) 1979-05-31
IL56758A0 (en) 1979-05-31
ATA807276A (en) 1979-05-15
CH627757A5 (en) 1982-01-29
AT353957B (en) 1979-12-10
DK463176A (en) 1977-05-01

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Legal Events

Date Code Title Description
BA A request for search or an international-type search has been filed
A85 Still pending on 85-01-01
BB A search report has been drawn up
BC A request for examination has been filed
BV The patent application has lapsed