SE405731B - Analogiforfaranden for framstellning av nya imidazolderivat med antiinflammatorisk och analgetisk verkan - Google Patents
Analogiforfaranden for framstellning av nya imidazolderivat med antiinflammatorisk och analgetisk verkanInfo
- Publication number
- SE405731B SE405731B SE7205565A SE556572A SE405731B SE 405731 B SE405731 B SE 405731B SE 7205565 A SE7205565 A SE 7205565A SE 556572 A SE556572 A SE 556572A SE 405731 B SE405731 B SE 405731B
- Authority
- SE
- Sweden
- Prior art keywords
- analogical
- inflammatory
- procedures
- preparation
- analgetic effect
- Prior art date
Links
- RAXXELZNTBOGNW-UHFFFAOYSA-N 1H-imidazole Chemical class C1=CNC=N1 RAXXELZNTBOGNW-UHFFFAOYSA-N 0.000 title 1
- 230000000202 analgesic effect Effects 0.000 title 1
- 230000003110 anti-inflammatory effect Effects 0.000 title 1
- 238000000034 method Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
- C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D241/12—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/44—Radicals substituted by doubly-bound oxygen, sulfur, or nitrogen atoms, or by two such atoms singly-bound to the same carbon atom
- C07D213/46—Oxygen atoms
- C07D213/50—Ketonic radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH687571A CH554415A (de) | 1970-06-01 | 1971-05-10 | Verfahren zur herstellung von zitronensaeure durch submerse gaerung. |
| CH696771A CH561202A5 (is") | 1971-05-10 | 1971-05-11 | |
| CH697571 | 1971-05-12 | ||
| CH425072A CH579072A5 (is") | 1971-05-10 | 1972-03-22 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SE405731B true SE405731B (sv) | 1978-12-27 |
Family
ID=27428754
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SE7205565A SE405731B (sv) | 1971-05-10 | 1972-04-27 | Analogiforfaranden for framstellning av nya imidazolderivat med antiinflammatorisk och analgetisk verkan |
Country Status (10)
| Country | Link |
|---|---|
| AT (4) | AT319940B (is") |
| AU (1) | AU472065B2 (is") |
| BE (1) | BE783244A (is") |
| CA (1) | CA1012148A (is") |
| CH (5) | CH561202A5 (is") |
| DE (1) | DE2221546A1 (is") |
| FR (1) | FR2137740B1 (is") |
| GB (1) | GB1381031A (is") |
| NL (1) | NL7206346A (is") |
| SE (1) | SE405731B (is") |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK513580A (da) * | 1980-01-07 | 1981-07-08 | Du Pont | Fremgangsmaade til fremstilling af 4,5-diaryl-alfa (polyhalogenalkyl)-1h-imidazol-2-methanoler |
| DD201677A5 (de) * | 1980-07-25 | 1983-08-03 | Ciba Geigy | Verfahren zur herstellung von trisubstituierten imidazolderivaten |
| US4372964A (en) * | 1980-10-30 | 1983-02-08 | E. I. Du Pont De Nemours And Company | Antiinflammatory 4,5-diaryl-1H-imidazole-2-methanols |
| GB2123831B (en) * | 1981-07-20 | 1986-01-15 | Ciba Geigy Ag | Trisubstituted oxazo compounds |
| AU554104B2 (en) * | 1981-09-01 | 1986-08-07 | F. Hoffmann-La Roche Ag | Heterocyclic compounds and fungicides containing same |
| EP0084756A1 (de) * | 1982-01-22 | 1983-08-03 | Ciba-Geigy Ag | Trisubstituierte Oxazaverbindungen |
| EP0084757A1 (de) * | 1982-01-25 | 1983-08-03 | Ciba-Geigy Ag | Trisubstituierte Diaza-Derivate |
| IL83467A0 (en) * | 1986-08-15 | 1988-01-31 | Fujisawa Pharmaceutical Co | Imidazole derivatives,processes for their preparation and pharmaceutical compositions containing the same |
| US5656644A (en) * | 1994-07-20 | 1997-08-12 | Smithkline Beecham Corporation | Pyridyl imidazoles |
| US5916891A (en) | 1992-01-13 | 1999-06-29 | Smithkline Beecham Corporation | Pyrimidinyl imidazoles |
| MX9300141A (es) * | 1992-01-13 | 1994-07-29 | Smithkline Beecham Corp | Compuestos de imidazol novedosos, procedimiento para su preparacion y composiciones farmaceuticas que lo contienen. |
| ES2053401B1 (es) * | 1992-01-13 | 1995-03-01 | Smithkline Beecham Corp | Compuestos de imidazol y procedimientos para su prepacion. |
| EP1306377A3 (en) * | 1993-11-08 | 2003-05-07 | Smithkline Beecham Corporation | Pyridyl-oxazoles and their use as cytokines inhibitors |
| US5620999A (en) * | 1994-07-28 | 1997-04-15 | Weier; Richard M. | Benzenesulfonamide subtituted imidazolyl compounds for the treatment of inflammation |
| US6426360B1 (en) * | 1994-07-28 | 2002-07-30 | G D Searle & Co. | 4,5-substituted imidazolyl compounds for the treatment of inflammation |
| AU4301096A (en) * | 1994-12-13 | 1996-07-03 | F. Hoffmann-La Roche Ag | Imidazole derivatives as protein kinase inhibitors in particular egf-r tyrosine kinase |
| US6127545A (en) * | 1997-04-18 | 2000-10-03 | Merck & Co., Inc. | Process for making 2-aryl-3-aryl-5-halo pyridines useful as COX-2 inhibitors |
| TW492959B (en) * | 1997-04-18 | 2002-07-01 | Merck & Co Inc | Process for making 2-aryl-3-aryl-5-halo pyridines useful as cox-2 inhibitors |
| US6130334A (en) * | 1998-04-15 | 2000-10-10 | Merck & Co., Inc. | Process for making 2-aryl-3-aryl-5-halo pyridines useful as COX-2 inhibitors |
| AU4798000A (en) * | 1999-04-09 | 2000-11-14 | Smithkline Beecham Corporation | Triarylimidazoles |
| AR029803A1 (es) * | 2000-02-21 | 2003-07-16 | Smithkline Beecham Plc | Imidazoles sustituidos con piridilo y composiciones farmaceuticas que las comprenden |
| GB0007405D0 (en) | 2000-03-27 | 2000-05-17 | Smithkline Beecham Corp | Compounds |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3192211A (en) * | 1962-05-03 | 1965-06-29 | Nl Combinatie Chem Ind | 5-phenyl-5-(2-pyrazyl)-hydantoin |
| US3538104A (en) * | 1969-02-28 | 1970-11-03 | Geigy Chem Corp | Pyridyl-2-imidazolones |
-
1971
- 1971-05-11 CH CH696771A patent/CH561202A5/xx not_active IP Right Cessation
- 1971-05-11 CH CH76875A patent/CH561717A5/xx not_active IP Right Cessation
- 1971-05-11 CH CH76775A patent/CH561716A5/xx not_active IP Right Cessation
- 1971-05-11 CH CH76975A patent/CH561718A5/xx not_active IP Right Cessation
-
1972
- 1972-03-22 CH CH425072A patent/CH579072A5/xx not_active IP Right Cessation
- 1972-04-27 SE SE7205565A patent/SE405731B/xx unknown
- 1972-04-28 GB GB1978172A patent/GB1381031A/en not_active Expired
- 1972-05-03 DE DE19722221546 patent/DE2221546A1/de not_active Withdrawn
- 1972-05-08 CA CA141,520A patent/CA1012148A/en not_active Expired
- 1972-05-09 AU AU42055/72A patent/AU472065B2/en not_active Expired
- 1972-05-10 AT AT386673A patent/AT319940B/de not_active IP Right Cessation
- 1972-05-10 AT AT386573A patent/AT319939B/de not_active IP Right Cessation
- 1972-05-10 AT AT408972A patent/AT316544B/de not_active IP Right Cessation
- 1972-05-10 BE BE783244A patent/BE783244A/xx not_active IP Right Cessation
- 1972-05-10 AT AT386773A patent/AT319941B/de not_active IP Right Cessation
- 1972-05-10 NL NL7206346A patent/NL7206346A/xx not_active Application Discontinuation
- 1972-05-10 FR FR7216738A patent/FR2137740B1/fr not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| DE2221546A1 (de) | 1972-11-16 |
| AT319940B (de) | 1975-01-10 |
| CH561717A5 (is") | 1975-05-15 |
| NL7206346A (is") | 1972-11-14 |
| FR2137740B1 (is") | 1975-08-01 |
| CH579072A5 (is") | 1976-08-31 |
| CH561716A5 (is") | 1975-05-15 |
| AU4205572A (en) | 1973-11-15 |
| AT319941B (de) | 1975-01-10 |
| CH561202A5 (is") | 1975-04-30 |
| FR2137740A1 (is") | 1972-12-29 |
| AU472065B2 (en) | 1976-05-13 |
| BE783244A (fr) | 1972-11-10 |
| CA1012148A (en) | 1977-06-14 |
| GB1381031A (en) | 1975-01-22 |
| AT319939B (de) | 1975-01-10 |
| AT316544B (de) | 1974-07-10 |
| CH561718A5 (is") | 1975-05-15 |
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