SE393374B - PROCEDURE FOR THE PREPARATION OF 2-ALKYL-2-DIALKYLAMINO-2, '6'-ACETOXYLIDIDES WITH LOCAL AESTHETIC EFFECT - Google Patents

PROCEDURE FOR THE PREPARATION OF 2-ALKYL-2-DIALKYLAMINO-2, '6'-ACETOXYLIDIDES WITH LOCAL AESTHETIC EFFECT

Info

Publication number
SE393374B
SE393374B SE7115656A SE1565671A SE393374B SE 393374 B SE393374 B SE 393374B SE 7115656 A SE7115656 A SE 7115656A SE 1565671 A SE1565671 A SE 1565671A SE 393374 B SE393374 B SE 393374B
Authority
SE
Sweden
Prior art keywords
acetoxylidides
dialkylamino
alkyl
procedure
preparation
Prior art date
Application number
SE7115656A
Other languages
Swedish (sv)
Inventor
H J F Adams
G H Kronberg
B H Takman
Original Assignee
Astra Pharma Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astra Pharma Prod filed Critical Astra Pharma Prod
Publication of SE393374B publication Critical patent/SE393374B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C53/00Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen
    • C07C53/38Acyl halides
    • C07C53/46Acyl halides containing halogen outside the carbonyl halide group
    • C07C53/50Acyl halides containing halogen outside the carbonyl halide group of acids containing three or more carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
SE7115656A 1970-12-22 1971-12-07 PROCEDURE FOR THE PREPARATION OF 2-ALKYL-2-DIALKYLAMINO-2, '6'-ACETOXYLIDIDES WITH LOCAL AESTHETIC EFFECT SE393374B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10077770A 1970-12-22 1970-12-22
US00164022A US3812147A (en) 1970-12-22 1971-07-19 Acylxylidide local anaesthetics

Publications (1)

Publication Number Publication Date
SE393374B true SE393374B (en) 1977-05-09

Family

ID=26797539

Family Applications (1)

Application Number Title Priority Date Filing Date
SE7115656A SE393374B (en) 1970-12-22 1971-12-07 PROCEDURE FOR THE PREPARATION OF 2-ALKYL-2-DIALKYLAMINO-2, '6'-ACETOXYLIDIDES WITH LOCAL AESTHETIC EFFECT

Country Status (23)

Country Link
US (1) US3812147A (en)
JP (1) JPS5644063B1 (en)
AR (1) AR193840A1 (en)
AT (1) AT319205B (en)
AU (1) AU468489B2 (en)
BE (1) BE776656A (en)
BR (1) BR7108466D0 (en)
CA (1) CA943966A (en)
DD (1) DD99779A5 (en)
DE (1) DE2162744C3 (en)
DK (1) DK139814B (en)
ES (2) ES398210A1 (en)
FI (1) FI55027C (en)
FR (1) FR2118985B1 (en)
GB (1) GB1369259A (en)
HU (1) HU163373B (en)
IE (1) IE35909B1 (en)
IT (1) IT1066334B (en)
NL (2) NL172149C (en)
NO (1) NO135934C (en)
PL (1) PL83097B1 (en)
SE (1) SE393374B (en)
SU (1) SU419023A3 (en)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4237068A (en) * 1971-07-28 1980-12-02 Astra Pharmaceutical Products, Inc. Primary aminoacylanilides
US3957996A (en) * 1971-12-08 1976-05-18 Astra Pharmaceutical Products, Inc. Pharmaceutical local anesthetic compositions
US3966934A (en) * 1971-12-08 1976-06-29 Astra Pharmaceutical Products, Inc. Synergistic local anesthetic compositions
US3975443A (en) * 1972-06-06 1976-08-17 Allen & Hanburys Limited 1-(3,4-dichlorobenzamidomethyl)-cyclohexyldimethylamine
JPS598269B2 (en) * 1975-08-22 1984-02-23 萬有製薬株式会社 Omega - aminoalkanesane arylamide
EP0062322A1 (en) * 1981-04-03 1982-10-13 The B.F. GOODRICH Company Improved process for synthesis of hindered amine stabilizers for polymeric materials
US4891058A (en) * 1988-07-18 1990-01-02 Ici Americas Inc. 1-alkyl-3-aryl imidazolidine-2,4-diones and herbicidal use
SE8900685D0 (en) * 1989-02-28 1989-02-28 Astra Ab NEW COMPOUNDS
US5153226A (en) * 1989-08-31 1992-10-06 Warner-Lambert Company Acat inhibitors for treating hypocholesterolemia
EP2101819B1 (en) 2006-11-20 2013-01-09 President and Fellows of Harvard College Methods, compositions, and kits for treating pain and pruritis
EP2995303A1 (en) 2009-07-10 2016-03-16 President and Fellows of Harvard College Permanently charged sodium and calcium channel blockers as anti-inflammatory agents
US11021443B2 (en) 2015-08-03 2021-06-01 President And Fellows Of Harvard College Charged ion channel blockers and methods for use
JP2022527690A (en) 2019-03-11 2022-06-03 ノシオン セラピューティクス,インコーポレイテッド Charged ion channel blockers and usage
US10780083B1 (en) 2019-03-11 2020-09-22 Nocion Therapeutics, Inc. Charged ion channel blockers and methods for use
WO2020185881A1 (en) 2019-03-11 2020-09-17 Nocion Therapeutics, Inc. Charged ion channel blockers and methods for use
BR112021017809A2 (en) 2019-03-11 2021-11-23 Nocion Therapeutics Inc Ester-substituted ion channel blockers and methods for use
US10786485B1 (en) 2019-03-11 2020-09-29 Nocion Therapeutics, Inc. Charged ion channel blockers and methods for use
WO2021091585A1 (en) 2019-11-06 2021-05-14 Nocion Therapeutics, Inc. Charged ion channel blockers and methods for use
WO2021091586A1 (en) 2019-11-06 2021-05-14 Nocion Therapeutics, Inc. Charged ion channel blockers and methods for use
MX2022011194A (en) 2020-03-11 2022-11-08 Nocion Therapeutics Inc Charged ion channel blockers and methods for use.

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1124837A (en) * 1966-06-03 1968-08-21 Wyeth John & Brother Ltd Substituted anilides

Also Published As

Publication number Publication date
NO135934B (en) 1977-03-21
IE35909L (en) 1972-06-22
NL172149C (en) 1983-07-18
JPS5644063B1 (en) 1981-10-16
CA943966A (en) 1974-03-19
IE35909B1 (en) 1976-06-23
IT1066334B (en) 1985-03-04
GB1369259A (en) 1974-10-23
DK139814C (en) 1979-10-01
DE2162744B2 (en) 1981-07-02
AU3709971A (en) 1973-06-28
AT319205B (en) 1974-12-10
BE776656A (en) 1972-06-14
FI55027C (en) 1979-05-10
AU468489B2 (en) 1976-01-15
BR7108466D0 (en) 1973-06-14
SU419023A3 (en) 1974-03-05
US3812147A (en) 1974-05-21
DE2162744C3 (en) 1982-04-15
DK139814B (en) 1979-04-23
PL83097B1 (en) 1975-12-31
NL8204126A (en) 1983-02-01
NO135934C (en) 1977-06-29
NL172149B (en) 1983-02-16
FI55027B (en) 1979-01-31
NL7117644A (en) 1972-06-26
DD99779A5 (en) 1973-08-20
AR193840A1 (en) 1973-05-31
FR2118985A1 (en) 1972-08-04
DE2162744A1 (en) 1972-07-06
ES425626A1 (en) 1976-06-16
FR2118985B1 (en) 1975-12-26
HU163373B (en) 1973-08-28
ES398210A1 (en) 1975-03-16

Similar Documents

Publication Publication Date Title
SE384211B (en) PROCEDURE FOR THE PREPARATION OF 2-SUBSTITUTED-4-AMINO-6,7,8-TRIALCOXIKINAZOLINES
SE393374B (en) PROCEDURE FOR THE PREPARATION OF 2-ALKYL-2-DIALKYLAMINO-2, '6'-ACETOXYLIDIDES WITH LOCAL AESTHETIC EFFECT
SE403286B (en) INTERMEDIATES FOR THE PREPARATION OF 1,4-HYDROXIMORFINAND DERIVATIVES
SE385885B (en) PROCEDURE FOR THE PREPARATION OF 4-AMINO-6-ARYLPYRIMIDINE DERIVATIVES
SE399427B (en) PROCEDURE FOR THE PREPARATION OF 2,4 DIAMINO-BENZYLPYRIMIDINES
SE384368B (en) PROCEDURE FOR THE PREPARATION OF 6-SUBSTITUTED - 4 - AMINO- 1,2 - DIHYDRO - 1 - HYDROXY - 2 - IMINOPYRIMIDINES
RO71354A (en) PROCEDURE FOR THE PREPARATION OF P-HALOPHENYL-2-PYRROLIDINONE
SE399701B (en) PROCEDURE FOR THE PREPARATION OF HYDROXYALKYLDIAMINE
SE390303B (en) PROCEDURE FOR THE PREPARATION OF ISOTIOCARBAMIDS WITH H? 712 BLOCKING EFFECT
FI54316B (en) ADJUSTMENT OF ADAMOSIN-5'-CARBONSYRADERIVAT WITH KRETSOMLOPPSVERKAN
SE394436B (en) PROCEDURE FOR THE PREPARATION OF 7-HALOGEN-LINCOMYCINES
SE380273B (en) PROCEDURE FOR THE PREPARATION OF THIOPYRIMIDINE DERIVATIVES
SE385011B (en) PROCEDURE FOR THE PREPARATION OF ALFA-LINCOSAMINIDES
SE389105B (en) PROCEDURE FOR THE PREPARATION OF CERTAIN STATED KETAZINES
SE388611B (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF 1,4-BENZODIAZEPONE DERIVATIVES
SE386175B (en) PROCEDURE FOR THE PREPARATION OF 1,4-BIS-ACYLPIPERAZINES
SE408418B (en) PROCEDURE FOR THE PREPARATION OF 5-FLUOR-PYRIMIDINES
SE390025B (en) PROCEDURE FOR THE PREPARATION OF 3 ALFA-HYDROXI-19-5 ALFA-PREGNAN-11,20-DION
SE380795B (en) PROCEDURE FOR THE PREPARATION OF THIOCARBAMIDS
SE383738B (en) PROCEDURE FOR THE PREPARATION OF SULFAMOYL BENZENESULPHONAMIDES WITH THERAPEUTIC PROPERTIES
SE382046B (en) PROCEDURE FOR THE PREPARATION OF 1-ARYLOXY-2-PROPANOL
SE389333B (en) PROCEDURE FOR THE PREPARATION OF ACCALIPOLYPHOSPHATE COMPLEX OF X-6-DESOXY-5-HYDROXITY SACYCLINE.
SE398878B (en) PROCEDURE FOR THE PREPARATION OF SUBSTITUTED 2,4-DIAMINO-5-BENZYLPYRIMIDINES
SE401366B (en) PROCEDURE FOR THE PREPARATION OF 2,6-METANO-3-BENSAZOCINES
RO70179A (en) PROCEDURE FOR THE PREPARATION OF IZOPRENE