RU92016289A - Новые 2-сахаринилметил гетероциклические карбоксилаты, полезные для использования в качестве ингибиторов протеолитических ферментов, их композиции и способ их применения - Google Patents

Новые 2-сахаринилметил гетероциклические карбоксилаты, полезные для использования в качестве ингибиторов протеолитических ферментов, их композиции и способ их применения

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Publication number
RU92016289A
RU92016289A RU92016289/33A RU92016289A RU92016289A RU 92016289 A RU92016289 A RU 92016289A RU 92016289/33 A RU92016289/33 A RU 92016289/33A RU 92016289 A RU92016289 A RU 92016289A RU 92016289 A RU92016289 A RU 92016289A
Authority
RU
Russia
Prior art keywords
saccharinilmethyl
inhibitors
useful
composition
new
Prior art date
Application number
RU92016289/33A
Other languages
English (en)
Other versions
RU2078081C1 (ru
Inventor
Поль Данлэп Ричард
Джон Хласта Деннец
Чиманлал Десай Ранджит
Гамильтон Лэйтимер Ли
Сабраманьям Чакрапани
Джозеф Курт Джон
Райс Белл Мэлкольм
Кьюмар Вирендра
Original Assignee
Стерлинг Уинтроп Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Стерлинг Уинтроп Инк. filed Critical Стерлинг Уинтроп Инк.
Publication of RU92016289A publication Critical patent/RU92016289A/ru
Application granted granted Critical
Publication of RU2078081C1 publication Critical patent/RU2078081C1/ru

Links

Claims (1)

  1. Изобретение относится к высокопроизводительному способу оптически активных замещенных 1,4-диолов, обладающих высокой степенью энантиомерной чистоты. Предлагаемый способ включает в себя электролитическое сочетание оптически активные β-оксикарбоновых кислот с высокой степенью энантиомерной чистоты.
RU9292016289A 1991-12-30 1992-12-29 2-сахаринилметилгетероциклические карбоксилаты или кислотно-аддитивные соли этих соединений основного характера или основно-аддитивные соли этих соединений кислотного характера, и фармацевтическая композиция, ингибирующая активность протеолитических ферментов RU2078081C1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US81662191A 1991-12-30 1991-12-30
US816621 1991-12-30

Publications (2)

Publication Number Publication Date
RU92016289A true RU92016289A (ru) 1995-06-19
RU2078081C1 RU2078081C1 (ru) 1997-04-27

Family

ID=25221159

Family Applications (1)

Application Number Title Priority Date Filing Date
RU9292016289A RU2078081C1 (ru) 1991-12-30 1992-12-29 2-сахаринилметилгетероциклические карбоксилаты или кислотно-аддитивные соли этих соединений основного характера или основно-аддитивные соли этих соединений кислотного характера, и фармацевтическая композиция, ингибирующая активность протеолитических ферментов

Country Status (18)

Country Link
US (5) US5376653A (ru)
EP (1) EP0550111B1 (ru)
JP (1) JPH05255287A (ru)
AT (1) ATE178899T1 (ru)
AU (1) AU653279B2 (ru)
CA (1) CA2086346A1 (ru)
CZ (1) CZ386892A3 (ru)
DE (1) DE69228923D1 (ru)
FI (1) FI925947A (ru)
HU (2) HUT65735A (ru)
IL (1) IL104260A0 (ru)
MX (1) MX9207611A (ru)
NO (1) NO301882B1 (ru)
NZ (1) NZ245587A (ru)
RU (1) RU2078081C1 (ru)
SG (1) SG50076A1 (ru)
SK (1) SK16599A3 (ru)
TW (1) TW223633B (ru)

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