RU2022109286A3 - - Google Patents

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Publication number
RU2022109286A3
RU2022109286A3 RU2022109286A RU2022109286A RU2022109286A3 RU 2022109286 A3 RU2022109286 A3 RU 2022109286A3 RU 2022109286 A RU2022109286 A RU 2022109286A RU 2022109286 A RU2022109286 A RU 2022109286A RU 2022109286 A3 RU2022109286 A3 RU 2022109286A3
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RU
Russia
Application number
RU2022109286A
Other languages
Russian (ru)
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RU2022109286A (ru
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Publication date
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Publication of RU2022109286A publication Critical patent/RU2022109286A/ru
Publication of RU2022109286A3 publication Critical patent/RU2022109286A3/ru

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RU2022109286A 2017-10-10 2018-10-04 Кристаллическая форма гидрата свободного основания лорлатиниба RU2022109286A (ru)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201762570326P 2017-10-10 2017-10-10
US62/570,326 2017-10-10
US201862727734P 2018-09-06 2018-09-06
US62/727,734 2018-09-06

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
RU2020113141A Division RU2845218C2 (ru) 2017-10-10 2018-10-04 Кристаллическая форма гидрата свободного основания лорлатиниба

Publications (2)

Publication Number Publication Date
RU2022109286A RU2022109286A (ru) 2022-05-06
RU2022109286A3 true RU2022109286A3 (enExample) 2026-03-10

Family

ID=64049474

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2022109286A RU2022109286A (ru) 2017-10-10 2018-10-04 Кристаллическая форма гидрата свободного основания лорлатиниба

Country Status (21)

Country Link
US (1) US11299500B2 (enExample)
EP (1) EP3694863B1 (enExample)
JP (1) JP7153069B2 (enExample)
KR (1) KR102424621B1 (enExample)
CN (1) CN111201235B (enExample)
AU (1) AU2018349259B2 (enExample)
CA (1) CA3077508C (enExample)
CY (1) CY1126141T1 (enExample)
DK (1) DK3694863T3 (enExample)
ES (1) ES2952985T3 (enExample)
FI (1) FI3694863T3 (enExample)
HU (1) HUE062926T2 (enExample)
MX (1) MX2020003373A (enExample)
PL (1) PL3694863T3 (enExample)
PT (1) PT3694863T (enExample)
RU (1) RU2022109286A (enExample)
SG (1) SG11202002445SA (enExample)
SI (1) SI3694863T1 (enExample)
TW (1) TWI775960B (enExample)
WO (1) WO2019073347A1 (enExample)
ZA (1) ZA202001661B (enExample)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG10201913200XA (en) 2015-07-31 2020-03-30 Pfizer Crystalline form of lorlatinib free base
CA3019905C (en) 2016-04-08 2022-08-23 Pfizer Inc. Crystalline forms of lorlatinib maleate
WO2019209633A1 (en) * 2018-04-23 2019-10-31 Pliva Hrvatska D.O.O. Solid state forms of lorlatinib and their preparation
US12391708B2 (en) 2019-07-18 2025-08-19 Tapi Croatia Industries Ltd Crystalline Lorlatinib : fumaric acid and solid state form thereof
CN112321604A (zh) * 2019-08-05 2021-02-05 华东理工大学 大环类jak2抑制剂及其应用
EP4041396A1 (en) 2019-10-10 2022-08-17 Sandoz AG Polymorph of lorlatinib
CN112824417A (zh) * 2019-11-21 2021-05-21 上海天慈国际药业有限公司 一种劳拉替尼的制备方法
TW202146017A (zh) 2020-03-05 2021-12-16 美商輝瑞股份有限公司 間變性淋巴瘤激酶抑制劑及周期蛋白依賴型激酶抑制劑之組合
CN111362967B (zh) * 2020-04-28 2021-09-07 南京雷正医药科技有限公司 苯并氧杂二氮杂十四碳烯衍生物及其用途

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2796967C (en) 2010-05-04 2015-12-01 Pfizer Inc. Heterocyclic derivatives as alk inhibitors
JP5808818B2 (ja) 2010-11-25 2015-11-10 ラツィオファーム・ゲーエムベーハー アファチニブの新規塩及び多形形態
PE20141639A1 (es) * 2011-06-08 2014-11-08 Biogen Idec Inc Proceso para preparar fumarato de dimetilo de alta pureza y cristalino
CA2863892C (en) * 2012-03-06 2016-08-30 Pfizer Inc. Macrocyclic derivatives for the treatment of proliferative diseases
CA2916605C (en) 2013-06-28 2018-04-24 Pfizer Inc. Solid forms of a macrocyclic kinase inhibitor
EP3183256A4 (en) * 2014-08-20 2018-05-30 Teligene Ltd. Substituted macrocycles useful as kinases inhibitors and methods of use thereof
WO2016026423A1 (en) * 2014-08-20 2016-02-25 Teligene Ltd Substituted macrocycles useful as kinases inhibitors and methods of use thereof
SG10201913200XA (en) 2015-07-31 2020-03-30 Pfizer Crystalline form of lorlatinib free base
CA3019905C (en) 2016-04-08 2022-08-23 Pfizer Inc. Crystalline forms of lorlatinib maleate

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