RU2017115188A3 - - Google Patents

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Publication number
RU2017115188A3
RU2017115188A3 RU2017115188A RU2017115188A RU2017115188A3 RU 2017115188 A3 RU2017115188 A3 RU 2017115188A3 RU 2017115188 A RU2017115188 A RU 2017115188A RU 2017115188 A RU2017115188 A RU 2017115188A RU 2017115188 A3 RU2017115188 A3 RU 2017115188A3
Authority
RU
Russia
Application number
RU2017115188A
Other languages
Russian (ru)
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RU2017115188A (ru
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of RU2017115188A publication Critical patent/RU2017115188A/ru
Publication of RU2017115188A3 publication Critical patent/RU2017115188A3/ru

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02Boron compounds
    • C07F5/025Boronic and borinic acid compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/69Boron compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Dermatology (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
RU2017115188A 2014-10-01 2015-10-01 Производные бороновой кислоты RU2017115188A (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP14003392.9 2014-10-01
EP14003392 2014-10-01
PCT/EP2015/002008 WO2016050359A1 (en) 2014-10-01 2015-10-01 Boronic acid derivatives

Publications (2)

Publication Number Publication Date
RU2017115188A RU2017115188A (ru) 2018-11-06
RU2017115188A3 true RU2017115188A3 (enExample) 2019-03-29

Family

ID=51690789

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2017115188A RU2017115188A (ru) 2014-10-01 2015-10-01 Производные бороновой кислоты

Country Status (14)

Country Link
US (1) US10294246B2 (enExample)
EP (1) EP3201207B1 (enExample)
JP (1) JP6835711B2 (enExample)
KR (1) KR102450583B1 (enExample)
CN (1) CN107001390B (enExample)
AU (1) AU2015327346B2 (enExample)
BR (1) BR112017006420A2 (enExample)
CA (1) CA2963205A1 (enExample)
ES (1) ES2873000T3 (enExample)
IL (1) IL251301B (enExample)
MX (1) MX370336B (enExample)
RU (1) RU2017115188A (enExample)
SG (1) SG11201702623TA (enExample)
WO (1) WO2016050359A1 (enExample)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2015327411B2 (en) 2014-10-01 2020-01-02 Merck Patent Gmbh Boronic acid derivatives
CA2963198A1 (en) 2014-10-01 2016-04-07 Merck Patent Gmbh Boronic acid derivatives
JP6662865B2 (ja) 2014-10-01 2020-03-11 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツングMerck Patent Gesellschaft mit beschraenkter Haftung ボロン酸誘導体
WO2019038250A1 (en) 2017-08-24 2019-02-28 Merck Patent Gmbh Boronic acid derivatives
CN112469480A (zh) * 2018-07-26 2021-03-09 默克专利股份公司 硼酸衍生物
CN113135943A (zh) * 2020-01-19 2021-07-20 首药控股(北京)有限公司 硼酸衍生物
CN113135944A (zh) * 2020-01-19 2021-07-20 首药控股(北京)有限公司 硼酸衍生物
US20250340577A1 (en) * 2021-03-02 2025-11-06 Case Western Reserve University Beta-lactomase inhibitors and uses thereof
WO2022243155A1 (en) * 2021-05-19 2022-11-24 Syngenta Crop Protection Ag Weed control method
IL310390A (en) 2021-07-29 2024-03-01 Merck Patent Gmbh Crystalline forms of [(1r)-2-(1-benzofuran-3-yl)-1-{[(1s,2r,4r)-7- oxabicyclo[2.2.1]heptan-2-yl]formamido}ethyl]boronic acid, adducts thereof, and processes to obtain
KR20240090392A (ko) * 2021-10-14 2024-06-21 쇼우야오 홀딩스 (베이징) 코., 엘티디. 보론산 유도체
WO2023232830A1 (en) 2022-06-02 2023-12-07 Merck Patent Gmbh Boronic acid adducts

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL111175A0 (en) * 1993-10-07 1994-12-29 Du Pont Merck Pharma Electrophilic peptide analogs as inhibitors of trypsin-like serine proteases and pharmaceutical compositions containing them
EP1196436A2 (en) * 1999-07-07 2002-04-17 Bristol-Myers Squibb Pharma Company Peptide boronic acid inhibitors of hepatitis c virus protease
US7271186B1 (en) 2002-12-09 2007-09-18 Northwestern University Nanomolar β-lactamase inhibitors
EA201000774A1 (ru) * 2007-11-13 2010-12-30 Новартис Интернэшнл Фармасьютикл Лтд. Ингибиторы бета-лактамазы
AR075090A1 (es) * 2008-09-29 2011-03-09 Millennium Pharm Inc Derivados de acido 1-amino-2-ciclobutiletilboronico inhibidores de proteosoma,utiles como agentes anticancerigenos, y composiciones farmaceuticas que los comprenden.
SG10201605152SA (en) * 2011-12-22 2016-08-30 Ares Trading Sa Alpha-amino boronic acid derivatives, selective immunoproteasome inhibitors
AU2015327411B2 (en) 2014-10-01 2020-01-02 Merck Patent Gmbh Boronic acid derivatives
CA2963198A1 (en) 2014-10-01 2016-04-07 Merck Patent Gmbh Boronic acid derivatives
JP6662865B2 (ja) 2014-10-01 2020-03-11 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツングMerck Patent Gesellschaft mit beschraenkter Haftung ボロン酸誘導体

Also Published As

Publication number Publication date
JP2017536335A (ja) 2017-12-07
MX2017004046A (es) 2017-06-19
CN107001390B (zh) 2020-11-27
SG11201702623TA (en) 2017-04-27
US10294246B2 (en) 2019-05-21
CN107001390A (zh) 2017-08-01
MX370336B (es) 2019-12-10
WO2016050359A1 (en) 2016-04-07
JP6835711B2 (ja) 2021-02-24
IL251301B (en) 2022-02-01
AU2015327346A1 (en) 2017-05-18
RU2017115188A (ru) 2018-11-06
EP3201207B1 (en) 2021-02-24
BR112017006420A2 (pt) 2017-12-19
ES2873000T3 (es) 2021-11-03
AU2015327346B2 (en) 2019-12-05
KR20170062517A (ko) 2017-06-07
KR102450583B1 (ko) 2022-10-04
IL251301A0 (en) 2017-05-29
US20180105539A1 (en) 2018-04-19
EP3201207A1 (en) 2017-08-09
CA2963205A1 (en) 2016-04-07

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Legal Events

Date Code Title Description
FA92 Acknowledgement of application withdrawn (lack of supplementary materials submitted)

Effective date: 20190919