RO70892A - PROCEDURE FOR THE PREPARATION OF 3,4-DIMETHOXY-N- (3- (4-METHOXYPHENYL) -1-METHYL-N-PROPYL) PENETYLAMINE - Google Patents

PROCEDURE FOR THE PREPARATION OF 3,4-DIMETHOXY-N- (3- (4-METHOXYPHENYL) -1-METHYL-N-PROPYL) PENETYLAMINE

Info

Publication number
RO70892A
RO70892A RO7383749A RO8374973A RO70892A RO 70892 A RO70892 A RO 70892A RO 7383749 A RO7383749 A RO 7383749A RO 8374973 A RO8374973 A RO 8374973A RO 70892 A RO70892 A RO 70892A
Authority
RO
Romania
Prior art keywords
penetylamine
dimethoxy
methoxyphenyl
propyl
methyl
Prior art date
Application number
RO7383749A
Other languages
French (fr)
Romanian (ro)
Inventor
Ronald R Tuttle
Jack Mills
Original Assignee
Eli Lilly And Co,Us
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22918877&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=RO70892(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Eli Lilly And Co,Us filed Critical Eli Lilly And Co,Us
Publication of RO70892A publication Critical patent/RO70892A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00Compounds containing amino groups bound to a carbon skeleton
    • C07C211/01Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms
    • C07C211/26Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing at least one six-membered aromatic ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/45Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by condensation
    • C07C45/46Friedel-Crafts reactions

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Cardiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
RO7383749A 1972-04-12 1973-04-12 PROCEDURE FOR THE PREPARATION OF 3,4-DIMETHOXY-N- (3- (4-METHOXYPHENYL) -1-METHYL-N-PROPYL) PENETYLAMINE RO70892A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US24346672A 1972-04-12 1972-04-12

Publications (1)

Publication Number Publication Date
RO70892A true RO70892A (en) 1982-02-26

Family

ID=22918877

Family Applications (2)

Application Number Title Priority Date Filing Date
RO7374457A RO65105A (en) 1972-04-12 1973-04-12 PROCEDURE FOR PREPARATION OF DOPAMIN DERIVATIVES
RO7383749A RO70892A (en) 1972-04-12 1973-04-12 PROCEDURE FOR THE PREPARATION OF 3,4-DIMETHOXY-N- (3- (4-METHOXYPHENYL) -1-METHYL-N-PROPYL) PENETYLAMINE

Family Applications Before (1)

Application Number Title Priority Date Filing Date
RO7374457A RO65105A (en) 1972-04-12 1973-04-12 PROCEDURE FOR PREPARATION OF DOPAMIN DERIVATIVES

Country Status (31)

Country Link
JP (2) JPS5825656B2 (en)
KR (1) KR790000113B1 (en)
AR (1) AR203822A1 (en)
AT (1) AT323719B (en)
AU (1) AU472734B2 (en)
BE (1) BE798051A (en)
BG (1) BG23001A3 (en)
CA (1) CA1018188A (en)
CH (2) CH569691A5 (en)
CS (2) CS190406B2 (en)
CY (1) CY963A (en)
DD (1) DD107670B3 (en)
DE (1) DE2317710C2 (en)
DK (1) DK142750C (en)
ES (1) ES413639A1 (en)
FR (1) FR2182947B1 (en)
GB (1) GB1392674A (en)
HK (1) HK50178A (en)
HU (2) HU166213B (en)
IE (1) IE37511B1 (en)
IL (1) IL42016A (en)
KE (1) KE2870A (en)
MY (1) MY7800381A (en)
NL (1) NL174459C (en)
PH (1) PH11041A (en)
PL (2) PL90695B1 (en)
RO (2) RO65105A (en)
SE (1) SE399064B (en)
SU (1) SU496719A3 (en)
YU (2) YU36483B (en)
ZA (1) ZA732136B (en)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH585693A5 (en) * 1974-02-08 1977-03-15 Ciba Geigy Ag
US4342692A (en) * 1980-10-20 1982-08-03 Usv Pharmaceutical Corporation Pyrrolidines
NO822514L (en) * 1981-07-22 1983-01-24 Syntex Inc PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVITY 2,5-SUBSTITUTED PYRROLIDE INGREDIENTS
JPS6061523A (en) * 1983-09-16 1985-04-09 Shionogi & Co Ltd Oral dobutamine pharmaceutical
ZA881076B (en) * 1987-02-24 1989-10-25 Lilly Co Eli Dobutamine salts
JPH0383364U (en) * 1989-12-18 1991-08-23
WO1992020645A1 (en) * 1991-05-20 1992-11-26 Tsumura & Co. Phellodendrine analogs and allergy type iv suppressor containing the same as active ingredient
ATE155125T1 (en) * 1993-04-13 1997-07-15 Duphar Int Res PRODUCTION OF DOBUTAMIN COMPOUNDS
EP0620208B1 (en) * 1993-04-13 1997-07-09 Duphar International Research B.V Production of dobutamine compounds
DK1546088T3 (en) 2002-10-03 2015-03-30 Novaremed Ltd RELATIONSHIPS FOR USING THE TREATMENT OF AUTO-IMMUNE DISEASES, IMMUNOALLERGIC DISEASES AND ORGAN OR TISSUE TRANSPLANT AID
AU2005225239B2 (en) 2002-10-03 2012-06-14 Novaremed Ltd Compounds for treating AIDS and other diseases
GB0804213D0 (en) 2008-03-06 2008-04-16 New Era Biotech Ltd A method of printing or preventing pain
BR112012002246A2 (en) 2009-07-31 2019-09-24 Cognition Therapeutics Inc acceptable pharmaceutical compound, compound or salt thereof, pharmaceutical composition, method for inhibiting, treating and / or reducing cognitive decline and / or akzhmer's disease in a patient
US8802734B2 (en) 2009-09-09 2014-08-12 Novaremed Limited Method of treating or preventing pain
HK1202248A1 (en) * 2011-08-25 2015-09-25 考格尼申治疗股份有限公司 Compositions and methods for treating neurodegenerative disease
DK3099296T3 (en) 2014-01-31 2019-04-15 Cognition Therapeutics Inc ISO-INDOLINE DERIVATIVES, COMPOSITIONS AND METHODS FOR TREATING NEURODEGENERATIVE DISEASE
KR102614814B1 (en) 2017-05-15 2023-12-20 카그니션 테라퓨틱스, 인코퍼레이티드 Composition for treating neurodegenerative diseases
CN114524734B (en) * 2021-12-27 2024-04-26 嘉实(湖南)医药科技有限公司 Preparation method of dobutamine hydrochloride
CN117326958B (en) * 2023-09-21 2025-07-11 锦州奥鸿药业有限责任公司 A preparation method of high-purity dobutamine hydrochloride

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2276619A (en) * 1942-03-17 N-phentlaliphatic-dihtoroxyphentnl

Also Published As

Publication number Publication date
DD107670B3 (en) 1988-04-06
CH569691A5 (en) 1975-11-28
CY963A (en) 1978-12-22
BG23001A3 (en) 1977-05-20
HK50178A (en) 1978-09-15
DK142750B (en) 1981-01-12
AU472734B2 (en) 1976-06-03
CS190448B2 (en) 1979-05-31
KR790000113B1 (en) 1979-03-20
ZA732136B (en) 1974-03-27
HU166213B (en) 1975-02-28
FR2182947A1 (en) 1973-12-14
IL42016A0 (en) 1973-06-29
AR203822A1 (en) 1975-10-31
PH11041A (en) 1977-10-25
NL174459B (en) 1984-01-16
YU37113B (en) 1984-08-31
DD107670A5 (en) 1974-08-12
YU36483B (en) 1984-02-29
AU5438573A (en) 1974-10-17
NL7305097A (en) 1973-10-16
GB1392674A (en) 1975-04-30
JPS497237A (en) 1974-01-22
CA1018188A (en) 1977-09-27
PL90695B1 (en) 1977-01-31
DE2317710A1 (en) 1973-10-18
YU97673A (en) 1982-02-25
DK142750C (en) 1981-08-17
SE399064B (en) 1978-01-30
SU496719A3 (en) 1975-12-25
MY7800381A (en) 1978-12-31
JPS58131945A (en) 1983-08-06
JPS6221343B2 (en) 1987-05-12
JPS5825656B2 (en) 1983-05-28
BE798051A (en) 1973-10-11
CH580563A5 (en) 1976-10-15
NL174459C (en) 1984-06-18
RO65105A (en) 1980-01-15
DE2317710C2 (en) 1983-08-04
IE37511B1 (en) 1977-08-03
IL42016A (en) 1976-05-31
YU321279A (en) 1983-04-27
HU167597B (en) 1975-11-28
FR2182947B1 (en) 1976-07-02
ES413639A1 (en) 1976-01-16
CS190406B2 (en) 1979-05-31
AT323719B (en) 1975-07-25
PL94207B1 (en) 1977-07-30
KE2870A (en) 1978-09-01

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