PT89998A - Processo para a preparacao de 4-pentafluorofenoxipiperidinas 1--substituidas e de uma composicao farmaceutica que os contem - Google Patents

Processo para a preparacao de 4-pentafluorofenoxipiperidinas 1--substituidas e de uma composicao farmaceutica que os contem

Info

Publication number
PT89998A
PT89998A PT89998A PT8999889A PT89998A PT 89998 A PT89998 A PT 89998A PT 89998 A PT89998 A PT 89998A PT 8999889 A PT8999889 A PT 8999889A PT 89998 A PT89998 A PT 89998A
Authority
PT
Portugal
Prior art keywords
pentafluorofenoxipiperidines
substituted
preparing
pharmaceutical composition
pharmaceutical
Prior art date
Application number
PT89998A
Other languages
English (en)
Inventor
Grover Cleveland Helsley
Larry Davis
Gordom Edward Olsen
Original Assignee
Hoechst Roussel Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma
Publication of PT89998A publication Critical patent/PT89998A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40Oxygen atoms
    • C07D211/44Oxygen atoms attached in position 4
    • C07D211/46Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Psychiatry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT89998A 1988-03-14 1989-03-13 Processo para a preparacao de 4-pentafluorofenoxipiperidinas 1--substituidas e de uma composicao farmaceutica que os contem PT89998A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US16793588A 1988-03-14 1988-03-14

Publications (1)

Publication Number Publication Date
PT89998A true PT89998A (pt) 1989-11-10

Family

ID=22609420

Family Applications (1)

Application Number Title Priority Date Filing Date
PT89998A PT89998A (pt) 1988-03-14 1989-03-13 Processo para a preparacao de 4-pentafluorofenoxipiperidinas 1--substituidas e de uma composicao farmaceutica que os contem

Country Status (4)

Country Link
EP (1) EP0333028A1 (pt)
JP (1) JPH01275557A (pt)
DK (1) DK121089A (pt)
PT (1) PT89998A (pt)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1280699A (en) * 1968-12-23 1972-07-05 Robins Co Inc A H 0-substituted-4-phenoxypiperidines
US4518713A (en) * 1984-04-13 1985-05-21 Hoechst-Roussel Pharmaceuticals Inc. Analgesic substituted-1-aminoalkylamino-4-aryloxypiperidines

Also Published As

Publication number Publication date
EP0333028A1 (en) 1989-09-20
JPH01275557A (ja) 1989-11-06
DK121089D0 (da) 1989-03-13
DK121089A (da) 1989-09-15

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Legal Events

Date Code Title Description
FC3A Refusal

Effective date: 19940421