PT88990A - Processo para a preparacao de novos acidos aza-cicloalquil-alcano-difosfonicos - Google Patents
Processo para a preparacao de novos acidos aza-cicloalquil-alcano-difosfonicosInfo
- Publication number
- PT88990A PT88990A PT88990A PT8899088A PT88990A PT 88990 A PT88990 A PT 88990A PT 88990 A PT88990 A PT 88990A PT 8899088 A PT8899088 A PT 8899088A PT 88990 A PT88990 A PT 88990A
- Authority
- PT
- Portugal
- Prior art keywords
- diphosphones
- cicloalquil
- alcano
- aza
- preparation
- Prior art date
Links
- 239000002253 acid Substances 0.000 title 1
- 150000007513 acids Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/5532—Seven-(or more) membered rings
- C07F9/5535—Seven-(or more) membered rings condensed with carbocyclic rings or ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
- A61P3/14—Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/576—Six-membered rings
- C07F9/5765—Six-membered rings condensed with carbocyclic rings or carbocyclic ring systems
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Diabetes (AREA)
- Engineering & Computer Science (AREA)
- Endocrinology (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH443587 | 1987-11-13 |
Publications (1)
Publication Number | Publication Date |
---|---|
PT88990A true PT88990A (pt) | 1989-11-30 |
Family
ID=4276083
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT88990A PT88990A (pt) | 1987-11-13 | 1988-11-11 | Processo para a preparacao de novos acidos aza-cicloalquil-alcano-difosfonicos |
Country Status (6)
Country | Link |
---|---|
US (1) | US4929606A (pt) |
EP (1) | EP0317505A1 (pt) |
JP (1) | JPH01160993A (pt) |
AU (1) | AU2503688A (pt) |
DK (1) | DK632088A (pt) |
PT (1) | PT88990A (pt) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3822650A1 (de) * | 1988-07-05 | 1990-02-01 | Boehringer Mannheim Gmbh | Neue diphosphonsaeurederivate, verfahren zu deren herstellung und diese verbindungen enthaltende arzneimittel |
US4990503A (en) * | 1988-08-12 | 1991-02-05 | Yamanouchi Pharmaceutical Co., Ltd. | Heterocyclic bisphosphonic acid derivatives |
DE3843481A1 (de) * | 1988-12-23 | 1990-06-28 | Boehringer Ingelheim Kg | Substituierte 3-azabicyclo/3.1.1/heptane, ihre herstellung und ihre verwendung |
MX21452A (es) * | 1989-07-07 | 1994-01-31 | Ciba Geigy Ag | Preparaciones farmaceuticas que se administran en forma topica. |
US5139786A (en) * | 1989-07-07 | 1992-08-18 | Ciba-Geigy Corporation | Topical formulations |
EP0510066A4 (en) * | 1990-01-12 | 1992-12-02 | Rhone-Poulenc Rorer International (Holdings) Inc. | 1-azetidyl and 1-hexamethylenimine alkyl or aryl bisphosphonic acids and their use as pharmacological agents |
US5270365A (en) * | 1991-12-17 | 1993-12-14 | Merck & Co., Inc. | Prevention and treatment of periodontal disease with alendronate |
JPH06298779A (ja) * | 1993-04-15 | 1994-10-25 | Hoechst Japan Ltd | ヘテロ環イミノビスメチレンビスホスホン酸誘導体 |
US5854227A (en) * | 1994-03-04 | 1998-12-29 | Hartmann; John F. | Therapeutic derivatives of diphosphonates |
EP1057488A4 (en) * | 1998-12-25 | 2003-10-22 | Toray Industries | INTERLEUKIN-6 PRODUCTION INHIBITORS |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3733270A (en) * | 1971-03-08 | 1973-05-15 | Monsanto Co | Methods of scale inhibition |
JPS54135724A (en) * | 1978-04-11 | 1979-10-22 | Nissan Chem Ind Ltd | Preparation of amino-methylenedisulfonic acid derivative |
SU1002300A1 (ru) * | 1981-10-29 | 1983-03-07 | Ордена Ленина институт элементоорганических соединений им.А.Н.Несмеянова | Способ получени @ -аминозамещенных- @ -оксипропилидендифосфоновых кислот |
DE3203308A1 (de) * | 1982-01-27 | 1983-07-28 | Schering Ag, 1000 Berlin Und 4619 Bergkamen | Diphosphonsaeure-derivate und diese enthaltende pharmazeutische praeparate |
DE3232997A1 (de) * | 1982-09-04 | 1984-03-08 | Henkel KGaA, 4000 Düsseldorf | Diphosphonsaeuren |
DE3428524A1 (de) * | 1984-08-02 | 1986-02-13 | Boehringer Mannheim Gmbh, 6800 Mannheim | Neue diphosphonsaeurederivate, verfahren zu deren herstellung und diese verbindungen enthaltende arzneimittel |
IL77243A (en) * | 1984-12-21 | 1996-11-14 | Procter & Gamble | Pharmaceutical compositions containing geminal diphosphonic acid compounds and certain such novel compounds |
DE3623397A1 (de) * | 1986-07-11 | 1988-01-14 | Boehringer Mannheim Gmbh | Neue diphosphonsaeurederivate, verfahren zu deren herstellung und diese verbindungen enthaltende arzneimittel |
DE3626058A1 (de) * | 1986-08-01 | 1988-02-11 | Boehringer Mannheim Gmbh | Neue diphosphonsaeurederivate, verfahren zu deren herstellung und diese verbindungen enthaltende arzneimittel |
DE3770787D1 (en) * | 1986-11-21 | 1991-07-18 | Ciba Geigy Ag | Aromatisch substituierte azacyclo-alkylalkandiphosphonsaeuren. |
-
1988
- 1988-11-03 EP EP88810751A patent/EP0317505A1/de not_active Withdrawn
- 1988-11-07 US US07/267,585 patent/US4929606A/en not_active Expired - Fee Related
- 1988-11-11 PT PT88990A patent/PT88990A/pt not_active Application Discontinuation
- 1988-11-11 AU AU25036/88A patent/AU2503688A/en not_active Abandoned
- 1988-11-11 DK DK632088A patent/DK632088A/da not_active Application Discontinuation
- 1988-11-12 JP JP63284858A patent/JPH01160993A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
AU2503688A (en) | 1989-05-25 |
JPH01160993A (ja) | 1989-06-23 |
DK632088A (da) | 1989-05-14 |
EP0317505A1 (de) | 1989-05-24 |
US4929606A (en) | 1990-05-29 |
DK632088D0 (da) | 1988-11-11 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC3A | Refusal |
Effective date: 19921126 |