PT88022A - Processo para a preparacao de 5-aril-11-substituido-5h,11h-pirrolo-{2,1-c}{1,4}benzoxazepinas - Google Patents

Processo para a preparacao de 5-aril-11-substituido-5h,11h-pirrolo-{2,1-c}{1,4}benzoxazepinas

Info

Publication number
PT88022A
PT88022A PT88022A PT8802288A PT88022A PT 88022 A PT88022 A PT 88022A PT 88022 A PT88022 A PT 88022A PT 8802288 A PT8802288 A PT 8802288A PT 88022 A PT88022 A PT 88022A
Authority
PT
Portugal
Prior art keywords
benzoxazepins
pyrrolo
aryl
substituted
preparation
Prior art date
Application number
PT88022A
Other languages
English (en)
Inventor
Richard Charles Effland
Kevin James Kapples
Original Assignee
Hoechst Roussel Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma
Publication of PT88022A publication Critical patent/PT88022A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
PT88022A 1987-07-20 1988-07-19 Processo para a preparacao de 5-aril-11-substituido-5h,11h-pirrolo-{2,1-c}{1,4}benzoxazepinas PT88022A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/075,463 US4794110A (en) 1987-07-20 1987-07-20 5-Aryl-11-substituted-5H,11H-pyrrolo[2,1-c][1,4]benzoxazepined as analgesic and hypotensive agents

Publications (1)

Publication Number Publication Date
PT88022A true PT88022A (pt) 1989-06-30

Family

ID=22125924

Family Applications (1)

Application Number Title Priority Date Filing Date
PT88022A PT88022A (pt) 1987-07-20 1988-07-19 Processo para a preparacao de 5-aril-11-substituido-5h,11h-pirrolo-{2,1-c}{1,4}benzoxazepinas

Country Status (5)

Country Link
US (1) US4794110A (pt)
EP (1) EP0300356A1 (pt)
JP (1) JPS6440486A (pt)
DK (1) DK401988A (pt)
PT (1) PT88022A (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5015637A (en) * 1990-05-25 1991-05-14 Hoechst-Roussel Pharmaceutical Inc. Pyrido[3,4-b]pyrrolo[1,2-e][1,4,5]oxadiazepines
CA2450073C (en) 2001-07-25 2017-08-29 Biomarin Pharmaceutical Inc. Compositions and methods for modulating blood-brain barrier transport
EP2392258B1 (en) 2005-04-28 2014-10-08 Proteus Digital Health, Inc. Pharma-informatics system
KR20090071598A (ko) 2006-09-18 2009-07-01 랩터 파마슈티컬 인코포레이티드 수용체 결합 단백질(rap)-접합체 투여에 의한 간 질환의 치료
GB0711776D0 (en) * 2007-06-18 2007-07-25 Syngenta Participations Ag Substituted aromatic heterocyclic compounds as fungicides
EP2398500B1 (en) 2009-02-20 2019-03-13 2-BBB Medicines B.V. Glutathione-based drug delivery system
MY163048A (en) 2009-05-06 2017-08-15 Laboratory Skin Care Inc Dermal delivery compositions comprising active agent-calcium phosphate particle complexes and methods of using the same
US20120077778A1 (en) 2010-09-29 2012-03-29 Andrea Bourdelais Ladder-Frame Polyether Conjugates

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4045448A (en) * 1976-02-26 1977-08-30 American Hoechst Corporation Pyrrolo[2,1-c][1,4]benzoxazepine and benzoxazocine derivatives
US4169094A (en) * 1977-01-19 1979-09-25 American Hoechst Corporation Process for preparing aminoalkylpyrrolobenzoxazalkanes
US4681879A (en) * 1983-11-07 1987-07-21 Hoechst-Roussel Pharmaceuticals Inc. 11-substituted 5H,11H-pyrrolo[2,1-c][1,4]benzoxazepines as antipsychotic and analgesic agents
US4608374A (en) * 1983-11-07 1986-08-26 Hoechst-Roussel Pharmaceuticals Inc. 11-substituted 5H,11H-pyrrolo[2,1-c][1,4]benzoxazepines as antipsychotic and analgesic agents

Also Published As

Publication number Publication date
DK401988A (da) 1989-01-21
EP0300356A1 (en) 1989-01-25
JPS6440486A (en) 1989-02-10
DK401988D0 (da) 1988-07-19
US4794110A (en) 1988-12-27

Similar Documents

Publication Publication Date Title
BR8803759A (pt) Processo para a preparacao de 2,2,6,6-tetrametil-4-piperidilaminas
BR8902297A (pt) Processo para a preparacao de 1,1,1,2-tetrafluoretano
PT94059A (pt) Processo para a preparacao de copolimetros hidrossoluveis, de n-vinilamidas
PT84316B (pt) Processo para a preparacao de cicloalcano {1,2 -b} indole-sulfamidas
PT89705B (pt) Processo para a preparacao de 2', 3'-didesoxi-2', 2'-difluoronucleosidos
BR8802484A (pt) Processo para a preparacao de isocianatos
BR9003345A (pt) Processo para a preparacao de 1,1,1,2-tetrafluoretano
PT90293A (pt) Processo para a preparacao de macrolidos
PT91895A (pt) Processo para a preparacao de 9h-purinas substituidas
BR8906327A (pt) Processo para a preparacao de organoclorossilanos
PT90854A (pt) Processo para a preparacao de 1-aril-2-naftoilaminas
PT89039A (pt) Processo para a preparacao de l-ramnose
PT89056A (pt) Processo para a preparacao de hidroxilaminas substituidas
BR8803678A (pt) Processo para a preparacao de polieteramidas
BR8205514A (pt) Processo para a preparacao de 1,2-dicloroetano
PT84459B (pt) Processo para a preparacao de derivados de ciclopropano 1,1-dissubstituidos
BR8804414A (pt) Processo para a producao de dos 2,2,4-monoesteres tri-substitui-insaturados
PT93736A (pt) Processo para a preparacao de n,n'-ditrimetoxi-benzoil-piperazinas 2- substituidas
BR8806351A (pt) Processo para a preparacao de fenil-ureias
BR8903367A (pt) Processo para a preparacao de organoclorossilanos
PT88022A (pt) Processo para a preparacao de 5-aril-11-substituido-5h,11h-pirrolo-{2,1-c}{1,4}benzoxazepinas
BR8902030A (pt) Processo para a preparacao de n-fosfonometilglicina
BR9003346A (pt) Processo para a preparacao de 1,2-dicloro-1,1,2-trifluoretano
BR9101662A (pt) Processo para a producao de 1,4-butanodiol
BR8500540A (pt) Processo para a preparacao de 1,3,2-dioxaborinanos

Legal Events

Date Code Title Description
FC3A Refusal

Effective date: 19941109