PT846686E - Derivados de 1-fenil-pirazole e suas utilizacoes como agentes parasiticidas - Google Patents

Derivados de 1-fenil-pirazole e suas utilizacoes como agentes parasiticidas

Info

Publication number
PT846686E
PT846686E PT97309229T PT97309229T PT846686E PT 846686 E PT846686 E PT 846686E PT 97309229 T PT97309229 T PT 97309229T PT 97309229 T PT97309229 T PT 97309229T PT 846686 E PT846686 E PT 846686E
Authority
PT
Portugal
Prior art keywords
optionally substituted
halogen atoms
halogen
alkyl optionally
phenyl
Prior art date
Application number
PT97309229T
Other languages
English (en)
Inventor
Bernard Joseph Banks
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of PT846686E publication Critical patent/PT846686E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
PT97309229T 1996-11-30 1997-11-17 Derivados de 1-fenil-pirazole e suas utilizacoes como agentes parasiticidas PT846686E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9625045.1A GB9625045D0 (en) 1996-11-30 1996-11-30 Parasiticidal compounds

Publications (1)

Publication Number Publication Date
PT846686E true PT846686E (pt) 2002-05-31

Family

ID=10803815

Family Applications (1)

Application Number Title Priority Date Filing Date
PT97309229T PT846686E (pt) 1996-11-30 1997-11-17 Derivados de 1-fenil-pirazole e suas utilizacoes como agentes parasiticidas

Country Status (9)

Country Link
EP (1) EP0846686B1 (pt)
JP (1) JP3083278B2 (pt)
AT (1) ATE211735T1 (pt)
CA (1) CA2223237C (pt)
DE (1) DE69709532T2 (pt)
DK (1) DK0846686T3 (pt)
ES (1) ES2166954T3 (pt)
GB (1) GB9625045D0 (pt)
PT (1) PT846686E (pt)

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US6979686B1 (en) 2001-12-07 2005-12-27 Pharmacia Corporation Substituted pyrazoles as p38 kinase inhibitors
US6514977B1 (en) * 1997-05-22 2003-02-04 G.D. Searle & Company Substituted pyrazoles as p38 kinase inhibitors
EP1019394A1 (en) 1997-05-22 2000-07-19 G.D. Searle & Co. PYRAZOLE DERIVATIVES AS p38 KINASE INHIBITORS
GB9801851D0 (en) * 1998-01-29 1998-03-25 Pfizer Ltd Parasiticidal agents
ES2359973T3 (es) * 1998-03-19 2011-05-30 MERCK SHARP & DOHME CORP. Composiciones poliméricas líquidas para la liberación controlada de sustancias bioactivas.
GB9810354D0 (en) * 1998-05-14 1998-07-15 Pfizer Ltd Heterocycles
AR021608A1 (es) * 1998-12-11 2002-07-31 Merial Ltd Represion de artropodos en animales
US6531501B1 (en) 1998-12-11 2003-03-11 Aventis Cropscience, S.A. Control of arthropods in animals
AU765492B2 (en) 1998-12-25 2003-09-18 Teikoku Hormone Mfg. Co., Ltd. Aminopyrazole derivatives
US6506784B1 (en) 1999-07-01 2003-01-14 3-Dimensional Pharmaceuticals, Inc. Use of 1,3-substituted pyrazol-5-yl sulfonates as pesticides
US6409988B1 (en) 1999-07-01 2002-06-25 3-Dimensional Pharmaceuticals, Inc. Radiolabeled 1-aryl pyrazoles, the synthesis thereof and the use thereof as pest GABA receptor ligands
GB9916052D0 (en) * 1999-07-08 1999-09-08 Pfizer Ltd Anthelmintic compositions
JP2001031509A (ja) * 1999-07-15 2001-02-06 Nippon Bayer Agrochem Co Ltd チエニル−ピラゾール類の有害生物防除剤としての利用
US6518266B1 (en) 1999-07-22 2003-02-11 3-Dimensional Pharmaceuticals 1- Aryl-3-thioalkyl pyrazoles, the synthesis thereof and the use thereof as insecticides
WO2001025241A2 (en) 1999-10-06 2001-04-12 3-Dimensional Pharmaceuticals, Inc. Fused 1-(2,6-dichloro-4-trifluoromethylphenyl)-pyrazoles, the synthesis thereof and the use thereof as pesticides
MXPA02005511A (es) 1999-12-02 2004-09-10 Aventis Cropscience Sa Control de artropodos en animales.
GB0016787D0 (en) * 2000-07-07 2000-08-30 Pfizer Ltd Compounds useful in therapy
IL163790A0 (en) 2002-03-05 2005-12-18 Bayer Cropscience Sa 5-Substituted-alkylaminopyrazole derivatives as pesticides
CA2508474C (en) 2002-12-03 2011-04-26 Bayer Cropscience S.A. Pesticidal sulphonylaminopyrazoles
AU2003288038B2 (en) 2002-12-03 2009-04-23 Boehringer Ingelheim Animal Health USA Inc. Pesticidal 5- (acylamino) pyrazole derivatives
WO2005023773A1 (en) * 2003-09-04 2005-03-17 Pfizer Limited Process for the preparation of substituted aryl pyrazoles
GB0413970D0 (en) * 2004-06-22 2004-07-28 Syngenta Participations Ag Chemical compounds
CA2611979A1 (en) * 2005-06-15 2006-12-21 Pfizer Limited Substituted arylpyrazoles
US8362086B2 (en) 2005-08-19 2013-01-29 Merial Limited Long acting injectable formulations
PL2035390T3 (pl) 2006-07-05 2016-06-30 Merial Inc Związki będące pochodnymi 1-arylo-5-alkilopirazolu, sposoby ich wytwarzania i zastosowania
DE102006061538A1 (de) 2006-12-27 2008-07-03 Bayer Healthcare Ag Kombinationsprodukt zur Bekämpfung von Parasiten an Tieren
DE102006061537A1 (de) 2006-12-27 2008-07-03 Bayer Healthcare Ag Mittel zur Bekämpfung von Parasiten an Tieren
JP2011530548A (ja) 2008-08-14 2011-12-22 バイエル・クロップサイエンス・アーゲー 殺虫性4−フェニル−1h−ピラゾール類
US9173728B2 (en) 2008-11-19 2015-11-03 Merial Inc. Multi-cavity container having offset indentures for dispensing fluids
WO2010059529A2 (en) 2008-11-19 2010-05-27 Merial Limited Compositions comprising an aryl pyrazole and/or a formamidine, methods and uses thereof
CA2769385C (en) 2009-07-30 2017-10-17 Merial Limited Insecticidal 4-amino-thieno[2,3-d]-pyrimidine compounds and methods of their use
UA108641C2 (uk) 2010-04-02 2015-05-25 Паразитицидна композиція, яка містить чотири активних агенти, та спосіб її застосування
CN104023720B (zh) 2011-11-17 2016-10-26 梅里亚有限公司 包含芳基吡唑和取代咪唑的组合物,其方法和用途
JO3626B1 (ar) 2012-02-23 2020-08-27 Merial Inc تركيبات موضعية تحتوي على فيبرونيل و بيرميثرين و طرق استخدامها
TWI579274B (zh) 2012-04-20 2017-04-21 龍馬躍公司 製備1-芳基-5-烷基吡唑化合物的改良方法
UY35428A (es) 2013-03-15 2014-10-31 Monsanto Technology Llc ?azoles n-,c-disustituidos y composiciones y métodos para controlar plagas de nematodos?.
NZ731446A (en) 2014-10-31 2018-09-28 Boehringer Ingelheim Animal Health Usa Inc Parasiticidal composition comprising fipronil
CN107108514A (zh) * 2015-01-13 2017-08-29 先正达参股股份有限公司 具有含硫取代基的杀有害生物活性杂环衍生物
SI3395801T1 (sl) * 2015-12-16 2021-08-31 Nippon Soda Co., Ltd. Arilazolna spojina in sredstvo za zatiranje škodljivcev
CN106117145A (zh) * 2016-07-12 2016-11-16 潍坊鑫诺化工有限公司 5‑氨基‑1‑(2,6‑二氯‑4‑三氟甲基苯基)‑3‑氰基吡唑的制备方法
AR112672A1 (es) 2017-08-11 2019-11-27 Syngenta Participations Ag Derivados de tiofeno activos como plaguicidas

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1054655B (it) * 1975-08-27 1981-11-30 Lepetit Spa Derivati condensati del l isochinolina
FR2326421A1 (fr) * 1975-09-30 1977-04-29 Ugine Kuhlmann Nouveaux trifluoromethyl-3-aryl-4 amino-5 pyrazoles et leur application comme bases diazotables pour la synthese de matieres colorantes
YU47834B (sr) * 1989-08-10 1996-01-09 Schering Agrochemical Limited Azolni pesticid
AU1191292A (en) * 1991-02-11 1992-09-07 Schering Agrochemicals Limited Imidazole pesticides
HUT69739A (en) * 1992-03-26 1995-09-28 Dowelanco Process for producing n-heterocyclic nitroanilines and fungicides containing the compounds

Also Published As

Publication number Publication date
ES2166954T3 (es) 2002-05-01
CA2223237A1 (en) 1998-05-30
ATE211735T1 (de) 2002-01-15
EP0846686B1 (en) 2002-01-09
JP3083278B2 (ja) 2000-09-04
DE69709532D1 (de) 2002-02-14
CA2223237C (en) 2002-08-06
GB9625045D0 (en) 1997-01-22
EP0846686A1 (en) 1998-06-10
DK0846686T3 (da) 2002-03-25
JPH10182614A (ja) 1998-07-07
DE69709532T2 (de) 2002-10-31

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