PT84441B - Process for preparing benzylpyrimidine derivatives and compositions containing them - Google Patents

Process for preparing benzylpyrimidine derivatives and compositions containing them

Info

Publication number
PT84441B
PT84441B PT84441A PT8444187A PT84441B PT 84441 B PT84441 B PT 84441B PT 84441 A PT84441 A PT 84441A PT 8444187 A PT8444187 A PT 8444187A PT 84441 B PT84441 B PT 84441B
Authority
PT
Portugal
Prior art keywords
preparing
compositions containing
benzylpyrimidine derivatives
benzylpyrimidine
derivatives
Prior art date
Application number
PT84441A
Other languages
English (en)
Other versions
PT84441A (en
Inventor
Louis Giral
Michele Calas
Marc Puygrenier
Original Assignee
Rousselot Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rousselot Co filed Critical Rousselot Co
Publication of PT84441A publication Critical patent/PT84441A/pt
Publication of PT84441B publication Critical patent/PT84441B/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • C07D239/49—Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT84441A 1986-03-13 1987-03-11 Process for preparing benzylpyrimidine derivatives and compositions containing them PT84441B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8603602A FR2595697B1 (fr) 1986-03-13 1986-03-13 Derives de benzyl-pyrimidine, leur procede de preparation ainsi que les compositions en contenant

Publications (2)

Publication Number Publication Date
PT84441A PT84441A (en) 1987-04-01
PT84441B true PT84441B (en) 1989-03-22

Family

ID=9333094

Family Applications (1)

Application Number Title Priority Date Filing Date
PT84441A PT84441B (en) 1986-03-13 1987-03-11 Process for preparing benzylpyrimidine derivatives and compositions containing them

Country Status (4)

Country Link
EP (1) EP0237516A1 (pt)
JP (1) JPS6399061A (pt)
FR (1) FR2595697B1 (pt)
PT (1) PT84441B (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4206528A1 (de) * 1992-03-02 1993-09-09 Bayer Ag Cyanalken-derivate, verfahren zu ihrer herstellung und ihre verwendung als mikrobizid fuer den materialschutz
PT863882E (pt) 1995-10-17 2002-07-31 Janssen Pharmaceutica Nv Pirimidinas e triazinas amino-substituidas
KR100822530B1 (ko) 2004-03-05 2008-04-16 에프. 호프만-라 로슈 아게 Ｐ2ｘ3 및 ｐ2ｘ2/3 길항물질로서의 다이아미노피리미딘
JP4850913B2 (ja) 2005-09-01 2012-01-11 エフ．ホフマン−ラ ロシュ アーゲー Ｐ２ｘ３及びｐ２ｘ２／３調節因子としてのジアミノピリジン
CN101253159B (zh) 2005-09-01 2011-12-07 弗·哈夫曼-拉罗切有限公司 作为p2x3和p2x2/3调节剂的二氨基嘧啶类化合物
EP1924564B1 (en) 2005-09-01 2016-11-09 F.Hoffmann-La Roche Ag Diaminopyrimidines as p2x3 and p2x2/3 modulators
CN104529911B (zh) * 2014-12-31 2017-06-23 华中农业大学 一种氚标记艾地普林的制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1204678B (de) * 1958-04-18 1965-11-11 Wellcome Found Verfahren zur Herstellung von in 5'-oder 6'-Stellung bromsubstituierten 2, 4-Diamino-5-benzylpyrimidinen
FR1292920A (fr) * 1959-04-18 1962-05-11 Wellcome Found Dérivés de la pyrimidine et leur préparation
US3485840A (en) * 1964-11-12 1969-12-23 Hoffmann La Roche 2,4-diamino - 5 - (2',4',5'-substituted benzyl) pyrimidines,intermediates and processes

Also Published As

Publication number Publication date
FR2595697B1 (fr) 1988-07-08
EP0237516A1 (fr) 1987-09-16
FR2595697A1 (fr) 1987-09-18
PT84441A (en) 1987-04-01
JPS6399061A (ja) 1988-04-30

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