PT80375A - Process for preparing n,3-disubstituted 2-oxindole-1-carboxamides useful as analgesic and antiinflammatory agents - Google Patents

Process for preparing n,3-disubstituted 2-oxindole-1-carboxamides useful as analgesic and antiinflammatory agents

Info

Publication number
PT80375A
PT80375A PT80375A PT8037585A PT80375A PT 80375 A PT80375 A PT 80375A PT 80375 A PT80375 A PT 80375A PT 8037585 A PT8037585 A PT 8037585A PT 80375 A PT80375 A PT 80375A
Authority
PT
Portugal
Prior art keywords
oxindole
disubstituted
analgesic
preparing
antiinflammatory agents
Prior art date
Application number
PT80375A
Other languages
Portuguese (pt)
Other versions
PT80375B (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of PT80375A publication Critical patent/PT80375A/en
Publication of PT80375B publication Critical patent/PT80375B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/18Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/30Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/32Oxygen atoms
    • C07D209/34Oxygen atoms in position 2
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56Ring systems containing three or more rings
    • C07D209/58[b]- or [c]-condensed
    • C07D209/60Naphtho [b] pyrroles; Hydrogenated naphtho [b] pyrroles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56Ring systems containing three or more rings
    • C07D209/58[b]- or [c]-condensed
    • C07D209/70[b]- or [c]-condensed containing carbocyclic rings other than six-membered
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
PT80375A 1984-05-04 1985-04-30 N-3-DISSUBSTITUATED, UTEIS 2-OXIDOLE-1-CARBOXAMIDES AS ANALGESIC AND ANTI-INFLAMMATORY AGENTS PT80375B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US60735684A 1984-05-04 1984-05-04

Publications (2)

Publication Number Publication Date
PT80375A true PT80375A (en) 1985-05-01
PT80375B PT80375B (en) 1987-09-30

Family

ID=24431933

Family Applications (1)

Application Number Title Priority Date Filing Date
PT80375A PT80375B (en) 1984-05-04 1985-04-30 N-3-DISSUBSTITUATED, UTEIS 2-OXIDOLE-1-CARBOXAMIDES AS ANALGESIC AND ANTI-INFLAMMATORY AGENTS

Country Status (25)

Country Link
JP (1) JPS60243068A (en)
KR (1) KR870000497B1 (en)
AR (1) AR241159A1 (en)
BG (2) BG60208B2 (en)
CS (1) CS252828B2 (en)
DD (1) DD232916A5 (en)
EG (1) EG17193A (en)
ES (2) ES8609248A1 (en)
FI (1) FI80016C (en)
HU (1) HU196057B (en)
IE (1) IE851103L (en)
IN (1) IN161509B (en)
MA (1) MA20424A1 (en)
MW (1) MW1685A1 (en)
MX (1) MX5839A (en)
NO (1) NO163132C (en)
OA (1) OA08098A (en)
PL (2) PL145416B1 (en)
PT (1) PT80375B (en)
RO (2) RO91141B (en)
RU (1) RU2017729C1 (en)
SU (1) SU1468413A3 (en)
YU (1) YU44998B (en)
ZA (1) ZA853324B (en)
ZW (1) ZW7885A1 (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5047554A (en) * 1989-04-18 1991-09-10 Pfizer Inc. 3-substituted-2-oxindole derivatives
IL95880A (en) * 1989-10-13 1995-12-31 Pfizer Use of 3-substituted-2-oxindole derivatives for the preparation of a pharmaceutical preparation for inhibiting interleukin-1 biosynthesis

Also Published As

Publication number Publication date
KR850008154A (en) 1985-12-13
NO163132B (en) 1990-01-02
ZA853324B (en) 1986-12-30
ES542813A0 (en) 1986-07-16
CS252828B2 (en) 1987-10-15
ES8609248A1 (en) 1986-07-16
YU73085A (en) 1988-04-30
FI851756L (en) 1985-11-05
IE851103L (en) 1985-11-04
DD232916A5 (en) 1986-02-12
ES8707182A1 (en) 1987-07-16
JPS60243068A (en) 1985-12-03
RO91141B (en) 1987-07-03
PL257892A1 (en) 1986-10-07
IN161509B (en) 1987-12-19
MX5839A (en) 1993-11-01
JPH0335315B2 (en) 1991-05-27
PL147508B1 (en) 1989-06-30
NO851774L (en) 1985-11-05
KR870000497B1 (en) 1987-03-12
RO91141A (en) 1987-06-30
ZW7885A1 (en) 1985-07-24
YU44998B (en) 1991-06-30
NO163132C (en) 1990-04-11
RO94455B (en) 1988-07-01
BG60208B2 (en) 1993-12-30
SU1468413A3 (en) 1989-03-23
FI80016C (en) 1990-04-10
RU2017729C1 (en) 1994-08-15
CS320285A2 (en) 1987-03-12
MW1685A1 (en) 1986-09-10
OA08098A (en) 1987-03-31
PL253203A1 (en) 1986-06-17
RO94455A (en) 1988-06-30
EG17193A (en) 1990-08-30
HUT37754A (en) 1986-02-28
AR241159A1 (en) 1991-12-30
MA20424A1 (en) 1985-12-31
ES551275A0 (en) 1987-07-16
HU196057B (en) 1988-09-28
BG60207B2 (en) 1993-12-30
PL145416B1 (en) 1988-09-30
AR241159A2 (en) 1991-12-30
PT80375B (en) 1987-09-30
FI80016B (en) 1989-12-29
FI851756A0 (en) 1985-05-03

Similar Documents

Publication Publication Date Title
HUT39161A (en) Process for preparing 2-pyridon-derivatives and pharmaceuticals comprising the same
DE3560511D1 (en) Pleuromutilin derivatives, process for their preparation and their use
GB2159520B (en) 1, 24-dihydroxy- 22-vitamin d3 and process for preparing same
YU18085A (en) Process for obtaining 1,3-disubstituted 2-oxindoles
HUT47956A (en) Process for producing 2,3-disubstituted izoxazolidines and pharmaceuticals comprising same
PT81393A (en) Process for preparing oxindole antiinflammatory agents
EP0186628A3 (en) Pentaerythritdiphosphites, process for their preparation and their use as stabilizers
DE3662275D1 (en) Copper-chromium-titanium-silicon alloy, process for its production and its use
EP0228701A3 (en) 2-iodo-perfluoro-2-methylathanes, process for their production and their application
DE3665875D1 (en) Crystalline polyester-imides, process for production thereof, and use thereof
CS690485A2 (en) Process for preparing aminoalcohols
ZA85655B (en) Hydantoin derivatives,process for producing the same and medicine containing the same
EP0153732A3 (en) Polybutadiene and process for preparing the same
YU18185A (en) Process for preparing new 1,3,2-dioxaborinanes
ZA851190B (en) Pleuromutilin derivatives,process for their preparation and their use
PT80375A (en) Process for preparing n,3-disubstituted 2-oxindole-1-carboxamides useful as analgesic and antiinflammatory agents
HUT39442A (en) Process for preparing 1,3-disubstituted tetrahydro-pyridines
PT81140A (en) Process for preparing analgesic and antiinflammatory 1,3-diacyl-2-oxindole compounds
HUT42270A (en) Composition containing bromo-dichloro-imidazol derivatives as active agents and process for producing the active agents
HUT41233A (en) Insekticide, acaricide and nematocide compositions containing new benzoyl-phenyl-urea derivatives and process for producing the active agents
PT80104A (en) Process for preparing 1,2,4-triazacycloalkadiene derivatives
HUT37591A (en) Process for preparing /1,3-dioxi-1,3-propane-diil/-diimino/ -bis-benzoic acid and its derivatives
DE3561058D1 (en) Hydroxy-thia-alcanes, process for their preparation and their uses
GB2176188B (en) Process for producing 2,6-naphthalenediol and 2,6-diacetoxynaphthalene
PT79926B (en) Process for preparing 1,3-disubstituted 2-oxindoles useful as analgesic and anti-inflammatory agents