PT80246B - METHOD FOR PREPARING NEW CEFALOSPORIN DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM - Google Patents

METHOD FOR PREPARING NEW CEFALOSPORIN DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Info

Publication number
PT80246B
PT80246B PT80246A PT8024685A PT80246B PT 80246 B PT80246 B PT 80246B PT 80246 A PT80246 A PT 80246A PT 8024685 A PT8024685 A PT 8024685A PT 80246 B PT80246 B PT 80246B
Authority
PT
Portugal
Prior art keywords
pharmaceutical compositions
compositions containing
preparing new
cefalosporin
derivatives
Prior art date
Application number
PT80246A
Other languages
Portuguese (pt)
Other versions
PT80246A (en
Inventor
Takayuki Naito
Jun Okumura
Masahisa Oka
Haruhiro Yamashita
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of PT80246A publication Critical patent/PT80246A/en
Publication of PT80246B publication Critical patent/PT80246B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D285/00Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01Five-membered rings
    • C07D285/02Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/081,2,4-Thiadiazoles; Hydrogenated 1,2,4-thiadiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/78Separation; Purification; Stabilisation; Use of additives
    • C07C45/79Separation; Purification; Stabilisation; Use of additives by solid-liquid treatment; by chemisorption

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
PT80246A 1984-04-09 1985-04-04 METHOD FOR PREPARING NEW CEFALOSPORIN DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM PT80246B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US59794184A 1984-04-09 1984-04-09

Publications (2)

Publication Number Publication Date
PT80246A PT80246A (en) 1985-05-01
PT80246B true PT80246B (en) 1987-10-20

Family

ID=24393575

Family Applications (1)

Application Number Title Priority Date Filing Date
PT80246A PT80246B (en) 1984-04-09 1985-04-04 METHOD FOR PREPARING NEW CEFALOSPORIN DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Country Status (31)

Country Link
JP (4) JPS615084A (en)
KR (1) KR870002166B1 (en)
AR (1) AR244694A1 (en)
AT (1) AT388735B (en)
AU (2) AU580990B2 (en)
BE (1) BE902148A (en)
CA (3) CA1276929C (en)
CH (1) CH669197A5 (en)
DD (3) DD249024A5 (en)
DE (1) DE3512225A1 (en)
DK (1) DK155985A (en)
ES (4) ES8607318A1 (en)
FI (1) FI84830C (en)
FR (1) FR2563832B1 (en)
GB (3) GB2157293B (en)
GR (1) GR850883B (en)
HU (2) HU193750B (en)
IE (2) IE58408B1 (en)
IL (1) IL74826A (en)
IT (1) IT1190353B (en)
LU (1) LU85840A1 (en)
MY (1) MY101940A (en)
NL (1) NL192925C (en)
NZ (1) NZ211659A (en)
OA (1) OA07985A (en)
PT (1) PT80246B (en)
RU (1) RU2056425C1 (en)
SE (4) SE466205B (en)
SU (4) SU1375140A3 (en)
YU (2) YU46151B (en)
ZA (1) ZA852236B (en)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS61145186A (en) * 1984-12-20 1986-07-02 Meiji Seika Kaisha Ltd Novel cephem compound and preparation thereof
US4708955A (en) * 1985-06-24 1987-11-24 Bristol-Myers Company 3-(substituted)propenyl-7-aminothiazol-ylcephalosporanic acids and esters thereof
DE3650157T2 (en) * 1985-12-26 1995-05-04 Eisai Co Ltd CEPHALOSPORINE COMPOUNDS.
AU614723B2 (en) * 1986-10-13 1991-09-12 Eisai Co. Ltd. 3-propenylcephem derivative
IL84128A (en) * 1986-10-13 1992-12-01 Eisai Co Ltd 3-propenylcephem derivatives, their preparation and pharmaceutical compositions containing them
JPH085897B2 (en) * 1986-11-06 1996-01-24 エーザイ株式会社 3-propenyl cephem derivative
FR2622585B1 (en) * 1987-11-03 1991-04-19 Roussel Uclaf NOVEL CEPHALOSPORINS COMPRISING IN POSITION 3 A SUBSTITUTED VINYL RADICAL, THEIR PREPARATION PROCESS, THEIR APPLICATION AS MEDICAMENTS, THE COMPOSITIONS CONTAINING THEM AND THE NEW INTERMEDIATES OBTAINED
JPH0699449B2 (en) * 1988-03-16 1994-12-07 エーザイ株式会社 Synthetic intermediate of cephem derivative
EP0612751A3 (en) * 1988-03-16 1994-09-21 Eisai Co Ltd Compounds for the preparation of cephem derivatives.
FR2655042B1 (en) * 1989-11-29 1994-01-21 Adir Cie NOVEL SUBSTITUTED BENZOTHIAZOLINONES, PROCESS FOR THEIR PREPARATION AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.
FR2663332B1 (en) * 1990-06-15 1997-11-07 Roussel Uclaf NOVEL CEPHALOSPORINS COMPRISING IN POSITION 3 A RADICAL PROPENYL SUBSTITUTED BY A QUATERNARY AMMONIUM, THEIR PREPARATION PROCESS, THEIR APPLICATION AS MEDICAMENTS, THE COMPOSITIONS CONTAINING THEM AND THE NEW INTERMEDIATES OBTAINED.
US5126336A (en) * 1990-08-23 1992-06-30 Bristol-Myers Squibb Company Antibiotic c-3 catechol-substituted cephalosporin compounds, compositions and method of use thereof
AT396108B (en) * 1991-08-21 1993-06-25 Biochemie Gmbh NEW PROCESS AND NEW INTERMEDIATE PRODUCTS FOR THE PRODUCTION OF 7-AMINOCEPHALOSPORANIC ACID DERIVATIVES
JPH0741484A (en) * 1993-07-29 1995-02-10 Katayama Seiyakushiyo:Kk Cephem compound and antimicrobial agent
US5661144A (en) * 1994-08-16 1997-08-26 Meiji Seika Kabushiki Kaisha Cephem derivatives with 3-substituted bis heterocycles
PL345266A1 (en) 1998-06-22 2001-12-03 Hoffmann La Roche Propenyl cephalosporin derivatives
EP1666483B1 (en) 2003-09-09 2011-08-17 Nippon Chemical Industrial Company Limited Process for producing 3-chloromethyl-3-cephem derivative

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1342241A (en) * 1970-01-23 1974-01-03 Glaxo Lab Ltd Cephalosporin compounds
US4390534A (en) * 1978-12-29 1983-06-28 Fujisawa Pharmaceutical Co., Ltd. Cephem and cepham compounds
EP0025017A1 (en) * 1979-08-28 1981-03-11 Ciba-Geigy Ag Polyazathia compounds, process for their preparation, pharmaceutical preparations containing such compounds and use of the latter
US4409214A (en) * 1979-11-19 1983-10-11 Fujisawa Pharmaceutical, Co., Ltd. 7-Acylamino-3-vinylcephalosporanic acid derivatives and processes for the preparation thereof
GR75644B (en) * 1980-06-18 1984-08-02 Fujisawa Pharmaceutical Co
GR78245B (en) * 1980-09-12 1984-09-26 Ciba Geigy Ag
US4521413A (en) * 1981-09-14 1985-06-04 Fujisawa Pharmaceutical Co., Ltd. Cephem compounds
US4486586A (en) * 1983-02-10 1984-12-04 Bristol-Myers Company Cephalosporin derivatives

Also Published As

Publication number Publication date
SE470260B (en) 1993-12-20
FI84830C (en) 1992-01-27
GB8721347D0 (en) 1987-10-14
SE8901225D0 (en) 1989-04-06
BE902148A (en) 1985-10-09
IE58403B1 (en) 1993-09-22
ZA852236B (en) 1985-11-27
IT1190353B (en) 1988-02-16
DE3512225A1 (en) 1985-10-17
NL192925B (en) 1998-01-05
YU118987A (en) 1988-10-31
PT80246A (en) 1985-05-01
SE8501680D0 (en) 1985-04-03
YU46213B (en) 1993-05-28
NL192925C (en) 1998-05-07
DD249024A5 (en) 1987-08-26
RU2056425C1 (en) 1996-03-20
JPH0350754B2 (en) 1991-08-02
HU193750B (en) 1987-11-30
NZ211659A (en) 1988-11-29
ES542013A0 (en) 1986-06-16
DD251752A5 (en) 1987-11-25
ES8800949A1 (en) 1987-12-01
KR870002166B1 (en) 1987-12-14
SE8901224D0 (en) 1989-04-06
SE8901226L (en) 1989-04-06
SE8501680L (en) 1985-10-10
LU85840A1 (en) 1985-12-16
ES551550A0 (en) 1987-06-01
GB2194789B (en) 1988-10-12
KR850007424A (en) 1985-12-04
JPH0351716B2 (en) 1991-08-07
FI84830B (en) 1991-10-15
AU580990B2 (en) 1989-02-09
DD236735A5 (en) 1986-06-18
GB2157293B (en) 1988-10-05
SE470259B (en) 1993-12-20
JPH0262557B2 (en) 1990-12-26
AR244694A1 (en) 1993-11-30
IE58408B1 (en) 1993-09-22
OA07985A (en) 1987-01-31
ES557060A0 (en) 1987-12-01
GR850883B (en) 1985-11-25
ES8607318A1 (en) 1986-06-16
NL8501002A (en) 1985-11-01
FR2563832B1 (en) 1989-08-18
MY101940A (en) 1992-02-15
GB8721346D0 (en) 1987-10-14
JPS615084A (en) 1986-01-10
SU1436882A3 (en) 1988-11-07
GB8508846D0 (en) 1985-05-09
IE850866L (en) 1985-10-09
ES551551A0 (en) 1987-07-01
FI851379L (en) 1985-10-10
GB2194790A (en) 1988-03-16
SE505256C2 (en) 1997-07-21
GB2194790B (en) 1988-10-05
YU46151B (en) 1993-05-28
IT8520267A0 (en) 1985-04-05
HU204277B (en) 1991-12-30
AU610278B2 (en) 1991-05-16
IL74826A0 (en) 1985-07-31
CH669197A5 (en) 1989-02-28
IL74826A (en) 1990-01-18
SU1367858A3 (en) 1988-01-15
AU2504188A (en) 1989-03-02
GB2194789A (en) 1988-03-16
GB2157293A (en) 1985-10-23
SE8901225L (en) 1989-04-06
SE466205B (en) 1992-01-13
SE8901226D0 (en) 1989-04-06
FI851379A0 (en) 1985-04-04
JPH0357106B2 (en) 1991-08-30
FR2563832A1 (en) 1985-11-08
AT388735B (en) 1989-08-25
JPS61143390A (en) 1986-07-01
CA1276929C (en) 1990-11-27
HUT37622A (en) 1986-01-23
CA1340638C (en) 1999-07-06
SU1375140A3 (en) 1988-02-15
SE8901224L (en) 1989-04-06
YU60085A (en) 1987-12-31
JPS61143387A (en) 1986-07-01
DE3512225C2 (en) 1990-02-22
ATA103985A (en) 1989-01-15
ES8706694A1 (en) 1987-07-01
CA1340672C (en) 1999-07-20
JPS61143391A (en) 1986-07-01
SU1487814A3 (en) 1989-06-15
AU4086285A (en) 1985-10-17
DK155985A (en) 1985-10-10
ES8706155A1 (en) 1987-06-01
DK155985D0 (en) 1985-04-03

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