PT1444206E - Compostas de benzo[b]azepin-2-ona substituida como analgesicos - Google Patents
Compostas de benzo[b]azepin-2-ona substituida como analgesicosInfo
- Publication number
- PT1444206E PT1444206E PT02781280T PT02781280T PT1444206E PT 1444206 E PT1444206 E PT 1444206E PT 02781280 T PT02781280 T PT 02781280T PT 02781280 T PT02781280 T PT 02781280T PT 1444206 E PT1444206 E PT 1444206E
- Authority
- PT
- Portugal
- Prior art keywords
- azepin
- ona
- analgesics
- replaced
- benzo compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
- C07D223/14—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D223/16—Benzazepines; Hydrogenated benzazepines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P23/00—Anaesthetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Immunology (AREA)
- Rheumatology (AREA)
- Pulmonology (AREA)
- Dermatology (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10153348A DE10153348A1 (de) | 2001-10-29 | 2001-10-29 | Substituierte Benzo(b)azepin-2-on-Verbindungen |
Publications (1)
Publication Number | Publication Date |
---|---|
PT1444206E true PT1444206E (pt) | 2006-07-31 |
Family
ID=7704098
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT02781280T PT1444206E (pt) | 2001-10-29 | 2002-10-23 | Compostas de benzo[b]azepin-2-ona substituida como analgesicos |
Country Status (15)
Country | Link |
---|---|
US (1) | US7041662B2 (pt) |
EP (1) | EP1444206B1 (pt) |
JP (1) | JP2005511570A (pt) |
AR (1) | AR037124A1 (pt) |
AT (1) | ATE320418T1 (pt) |
CA (1) | CA2464191A1 (pt) |
CY (1) | CY1105039T1 (pt) |
DE (2) | DE10153348A1 (pt) |
DK (1) | DK1444206T3 (pt) |
ES (1) | ES2260487T3 (pt) |
HU (1) | HUP0401762A2 (pt) |
PE (1) | PE20030614A1 (pt) |
PL (1) | PL369852A1 (pt) |
PT (1) | PT1444206E (pt) |
WO (1) | WO2003037873A1 (pt) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BRPI0511049A (pt) * | 2004-05-12 | 2007-11-27 | Bayer Cropscience Gmbh | regulação do crescimento de plantas |
EA012602B1 (ru) * | 2004-05-12 | 2009-10-30 | Байер Кропсайенс Аг | Регулирование роста растений |
SE531698C2 (sv) | 2007-07-12 | 2009-07-07 | Respiratorius Ab | Nya bronkdilaterande a,b-omättade amider |
AU2016297024B2 (en) | 2015-07-22 | 2021-03-04 | Enanta Pharmaceuticals, Inc. | Benzodiazepine derivatives as RSV inhibitors |
WO2020190935A1 (en) | 2019-03-18 | 2020-09-24 | Enanta Pharmaceuticals, Inc. | Benzodiazepine derivatives as rsv inhibitors |
CN112759545B (zh) * | 2019-11-06 | 2022-12-13 | 复旦大学 | 3-(二甲氨基甲基)哌啶-4-醇类衍生物及其制备方法和药物用途 |
CN112759546B (zh) * | 2019-11-06 | 2022-08-26 | 复旦大学 | 3-(二甲氨基甲基)哌啶-4-醇衍生物及其制备方法和药物用途 |
CN112759587B (zh) * | 2019-11-06 | 2022-12-30 | 复旦大学 | 3-(二甲氨基甲基)哌啶-4-醇类衍生物及其制备方法和药物用途 |
WO2021088758A1 (zh) * | 2019-11-06 | 2021-05-14 | 复旦大学 | 一类阿片受体激动剂及其制备方法和药物用途 |
CN112759544B (zh) * | 2019-11-06 | 2022-08-26 | 复旦大学 | 3-(二甲氨基甲基)哌啶-4-醇衍生物制备方法和药物用途 |
WO2022086840A1 (en) | 2020-10-19 | 2022-04-28 | Enanta Pharmaceuticals, Inc. | Heterocyclic compounds as anti-viral agents |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3475414A (en) * | 1966-12-05 | 1969-10-28 | Miles Lab | Tetrahydro-1-benzazepin-2(1h)-one derivatives |
TW213901B (pt) * | 1992-01-27 | 1993-10-01 | Pfizer | |
DE19525137C2 (de) * | 1995-07-11 | 2003-02-27 | Gruenenthal Gmbh | 6-Dimethylaminomethyl-1-phenyl-cyclohexanverbin -dungen als Zwischenprodukte zur Herstellung pharmazeutischer Wirkstoffe |
-
2001
- 2001-10-29 DE DE10153348A patent/DE10153348A1/de not_active Withdrawn
-
2002
- 2002-10-23 DK DK02781280T patent/DK1444206T3/da active
- 2002-10-23 EP EP02781280A patent/EP1444206B1/de not_active Expired - Lifetime
- 2002-10-23 HU HU0401762A patent/HUP0401762A2/hu unknown
- 2002-10-23 PT PT02781280T patent/PT1444206E/pt unknown
- 2002-10-23 JP JP2003540155A patent/JP2005511570A/ja active Pending
- 2002-10-23 ES ES02781280T patent/ES2260487T3/es not_active Expired - Lifetime
- 2002-10-23 DE DE50206096T patent/DE50206096D1/de not_active Expired - Fee Related
- 2002-10-23 PL PL02369852A patent/PL369852A1/xx not_active Application Discontinuation
- 2002-10-23 AT AT02781280T patent/ATE320418T1/de not_active IP Right Cessation
- 2002-10-23 WO PCT/EP2002/011830 patent/WO2003037873A1/de active IP Right Grant
- 2002-10-23 CA CA002464191A patent/CA2464191A1/en not_active Abandoned
- 2002-10-28 PE PE2002001056A patent/PE20030614A1/es not_active Application Discontinuation
- 2002-10-29 AR ARP020104098A patent/AR037124A1/es unknown
-
2004
- 2004-04-14 US US10/824,244 patent/US7041662B2/en not_active Expired - Fee Related
-
2006
- 2006-05-31 CY CY20061100687T patent/CY1105039T1/el unknown
Also Published As
Publication number | Publication date |
---|---|
ATE320418T1 (de) | 2006-04-15 |
HUP0401762A2 (hu) | 2004-12-28 |
US20040224938A1 (en) | 2004-11-11 |
PL369852A1 (en) | 2005-05-02 |
CA2464191A1 (en) | 2003-05-08 |
AR037124A1 (es) | 2004-10-20 |
US7041662B2 (en) | 2006-05-09 |
PE20030614A1 (es) | 2003-07-26 |
CY1105039T1 (el) | 2010-03-03 |
EP1444206A1 (de) | 2004-08-11 |
WO2003037873A1 (de) | 2003-05-08 |
EP1444206B1 (de) | 2006-03-15 |
DK1444206T3 (da) | 2006-07-24 |
ES2260487T3 (es) | 2006-11-01 |
JP2005511570A (ja) | 2005-04-28 |
DE10153348A1 (de) | 2003-05-08 |
DE50206096D1 (de) | 2006-05-11 |
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