PL3894424T3 - Sól mesylanowa związku aminolupanowego o działaniu hamującym dojrzewanie hiv - Google Patents

Sól mesylanowa związku aminolupanowego o działaniu hamującym dojrzewanie hiv

Info

Publication number
PL3894424T3
PL3894424T3 PL19823817.2T PL19823817T PL3894424T3 PL 3894424 T3 PL3894424 T3 PL 3894424T3 PL 19823817 T PL19823817 T PL 19823817T PL 3894424 T3 PL3894424 T3 PL 3894424T3
Authority
PL
Poland
Prior art keywords
lupane
amino
compound
inhibitory activity
mesylate salt
Prior art date
Application number
PL19823817.2T
Other languages
English (en)
Inventor
Amy WOODS
Original Assignee
VIIV Healthcare UK(No.4) Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by VIIV Healthcare UK(No.4) Limited filed Critical VIIV Healthcare UK(No.4) Limited
Publication of PL3894424T3 publication Critical patent/PL3894424T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J63/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • C07J63/008Expansion of ring D by one atom, e.g. D homo steroids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)
  • AIDS & HIV (AREA)
  • General Chemical & Material Sciences (AREA)
  • Molecular Biology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
PL19823817.2T 2018-12-10 2019-12-09 Sól mesylanowa związku aminolupanowego o działaniu hamującym dojrzewanie hiv PL3894424T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862777432P 2018-12-10 2018-12-10
US201962874557P 2019-07-16 2019-07-16
PCT/IB2019/060564 WO2020121161A1 (en) 2018-12-10 2019-12-09 Mesylate salt of an amino-lupane compound with hiv maturation inhibitory activity

Publications (1)

Publication Number Publication Date
PL3894424T3 true PL3894424T3 (pl) 2023-05-02

Family

ID=68944386

Family Applications (1)

Application Number Title Priority Date Filing Date
PL19823817.2T PL3894424T3 (pl) 2018-12-10 2019-12-09 Sól mesylanowa związku aminolupanowego o działaniu hamującym dojrzewanie hiv

Country Status (16)

Country Link
US (1) US20220024970A1 (pl)
EP (1) EP3894424B1 (pl)
JP (1) JP2022510475A (pl)
CY (1) CY1125952T1 (pl)
DK (1) DK3894424T3 (pl)
ES (1) ES2938486T3 (pl)
FI (1) FI3894424T3 (pl)
HR (1) HRP20230208T1 (pl)
HU (1) HUE061184T2 (pl)
LT (1) LT3894424T (pl)
PL (1) PL3894424T3 (pl)
PT (1) PT3894424T (pl)
RS (1) RS64113B1 (pl)
SI (1) SI3894424T1 (pl)
SM (1) SMT202300049T1 (pl)
WO (1) WO2020121161A1 (pl)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SK9742002A3 (en) * 2000-01-07 2003-02-04 Transform Pharmaceuticals Inc High-throughput formation, identification, and analysis of diverse solid-forms
WO2014184553A1 (en) * 2013-05-15 2014-11-20 Cipla Limited Pharmaceutical antiretroviral compositions
NZ724644A (en) 2014-04-11 2023-07-28 Viiv Healthcare Uk No 4 Ltd Triterpenoids with hiv maturation inhibitory activity, substituted in position 3 by a non-aromatic ring carrying a haloalkyl substituent

Also Published As

Publication number Publication date
JP2022510475A (ja) 2022-01-26
EP3894424A1 (en) 2021-10-20
WO2020121161A1 (en) 2020-06-18
US20220024970A1 (en) 2022-01-27
SI3894424T1 (sl) 2023-04-28
HRP20230208T1 (hr) 2023-04-14
PT3894424T (pt) 2023-02-28
RS64113B1 (sr) 2023-04-28
ES2938486T3 (es) 2023-04-11
CY1125952T1 (el) 2024-09-20
HUE061184T2 (hu) 2023-05-28
SMT202300049T1 (it) 2023-03-17
FI3894424T3 (fi) 2023-04-25
EP3894424B1 (en) 2023-01-25
LT3894424T (lt) 2023-03-10
DK3894424T3 (da) 2023-03-06

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