SI3894424T1 - Mezilatna sol amino-lupanske spojine z zaviralno aktivnostjo dozorevanja HIV-a - Google Patents

Mezilatna sol amino-lupanske spojine z zaviralno aktivnostjo dozorevanja HIV-a

Info

Publication number
SI3894424T1
SI3894424T1 SI201930452T SI201930452T SI3894424T1 SI 3894424 T1 SI3894424 T1 SI 3894424T1 SI 201930452 T SI201930452 T SI 201930452T SI 201930452 T SI201930452 T SI 201930452T SI 3894424 T1 SI3894424 T1 SI 3894424T1
Authority
SI
Slovenia
Prior art keywords
lupane
amino
compound
inhibitory activity
mesylate salt
Prior art date
Application number
SI201930452T
Other languages
English (en)
Inventor
Amy Woods
Original Assignee
Viiv Healthcare Uk (No. 4) Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Viiv Healthcare Uk (No. 4) Limited filed Critical Viiv Healthcare Uk (No. 4) Limited
Publication of SI3894424T1 publication Critical patent/SI3894424T1/sl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J63/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • C07J63/008Expansion of ring D by one atom, e.g. D homo steroids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • AIDS & HIV (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
SI201930452T 2018-12-10 2019-12-09 Mezilatna sol amino-lupanske spojine z zaviralno aktivnostjo dozorevanja HIV-a SI3894424T1 (sl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201862777432P 2018-12-10 2018-12-10
US201962874557P 2019-07-16 2019-07-16
EP19823817.2A EP3894424B1 (en) 2018-12-10 2019-12-09 Mesylate salt of an amino-lupane compound with hiv maturation inhibitory activity
PCT/IB2019/060564 WO2020121161A1 (en) 2018-12-10 2019-12-09 Mesylate salt of an amino-lupane compound with hiv maturation inhibitory activity

Publications (1)

Publication Number Publication Date
SI3894424T1 true SI3894424T1 (sl) 2023-04-28

Family

ID=68944386

Family Applications (1)

Application Number Title Priority Date Filing Date
SI201930452T SI3894424T1 (sl) 2018-12-10 2019-12-09 Mezilatna sol amino-lupanske spojine z zaviralno aktivnostjo dozorevanja HIV-a

Country Status (14)

Country Link
US (1) US20220024970A1 (sl)
EP (1) EP3894424B1 (sl)
JP (1) JP2022510475A (sl)
DK (1) DK3894424T3 (sl)
ES (1) ES2938486T3 (sl)
FI (1) FI3894424T3 (sl)
HR (1) HRP20230208T1 (sl)
HU (1) HUE061184T2 (sl)
LT (1) LT3894424T (sl)
PL (1) PL3894424T3 (sl)
PT (1) PT3894424T (sl)
RS (1) RS64113B1 (sl)
SI (1) SI3894424T1 (sl)
WO (1) WO2020121161A1 (sl)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN2013MU01749A (sl) * 2013-05-15 2015-06-26 Cipla Ltd
CA2944778C (en) 2014-04-11 2022-06-14 ViiV Healthcare UK (No.4) Limited Triterpenoids with hiv maturation inhibitory activity

Also Published As

Publication number Publication date
LT3894424T (lt) 2023-03-10
DK3894424T3 (da) 2023-03-06
ES2938486T3 (es) 2023-04-11
EP3894424B1 (en) 2023-01-25
FI3894424T3 (fi) 2023-04-25
JP2022510475A (ja) 2022-01-26
PL3894424T3 (pl) 2023-05-02
EP3894424A1 (en) 2021-10-20
HRP20230208T1 (hr) 2023-04-14
PT3894424T (pt) 2023-02-28
WO2020121161A1 (en) 2020-06-18
RS64113B1 (sr) 2023-04-28
HUE061184T2 (hu) 2023-05-28
US20220024970A1 (en) 2022-01-27

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