PL3823623T3 - Podstawiony związek aminopirymidynowy do zastosowania w metodzie leczenia i zapobiegania stwardnieniu rozsianemu - Google Patents

Podstawiony związek aminopirymidynowy do zastosowania w metodzie leczenia i zapobiegania stwardnieniu rozsianemu

Info

Publication number
PL3823623T3
PL3823623T3 PL19768898.9T PL19768898T PL3823623T3 PL 3823623 T3 PL3823623 T3 PL 3823623T3 PL 19768898 T PL19768898 T PL 19768898T PL 3823623 T3 PL3823623 T3 PL 3823623T3
Authority
PL
Poland
Prior art keywords
treatment
multiple sclerosis
preventing multiple
aminopyrimidine compound
substituted aminopyrimidine
Prior art date
Application number
PL19768898.9T
Other languages
English (en)
Inventor
Martin DYROFF
David Mitchell
Orestis Papasouliotis
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of PL3823623T3 publication Critical patent/PL3823623T3/pl

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
PL19768898.9T 2018-07-20 2019-07-19 Podstawiony związek aminopirymidynowy do zastosowania w metodzie leczenia i zapobiegania stwardnieniu rozsianemu PL3823623T3 (pl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201862700977P 2018-07-20 2018-07-20
US201862730184P 2018-09-12 2018-09-12
US201962839273P 2019-04-26 2019-04-26
PCT/IB2019/056198 WO2020016850A1 (en) 2018-07-20 2019-07-19 A substituted amino-pyrimidine compound for use in a method for treatment and prevention of multiple sclerosis

Publications (1)

Publication Number Publication Date
PL3823623T3 true PL3823623T3 (pl) 2025-03-24

Family

ID=67953828

Family Applications (1)

Application Number Title Priority Date Filing Date
PL19768898.9T PL3823623T3 (pl) 2018-07-20 2019-07-19 Podstawiony związek aminopirymidynowy do zastosowania w metodzie leczenia i zapobiegania stwardnieniu rozsianemu

Country Status (22)

Country Link
US (1) US12251382B2 (pl)
EP (1) EP3823623B1 (pl)
JP (1) JP7724151B2 (pl)
KR (1) KR20210034623A (pl)
CN (1) CN112437665A (pl)
AU (2) AU2019306828A1 (pl)
BR (1) BR112021000893A2 (pl)
CA (1) CA3106772A1 (pl)
DK (1) DK3823623T3 (pl)
ES (1) ES3009670T3 (pl)
FI (1) FI3823623T3 (pl)
HR (1) HRP20241737T1 (pl)
HU (1) HUE069840T2 (pl)
IL (1) IL280197A (pl)
MX (1) MX2021000094A (pl)
PL (1) PL3823623T3 (pl)
PT (1) PT3823623T (pl)
SG (1) SG11202100518TA (pl)
TW (1) TWI879737B (pl)
UA (1) UA127744C2 (pl)
WO (1) WO2020016850A1 (pl)
ZA (1) ZA202101118B (pl)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2021173740A1 (en) * 2020-02-28 2021-09-02 Genentech, Inc. Methods of treating primary progressive multiple sclerosis using an inhibitor of bruton's tyrosine kinase
CN117320712A (zh) 2021-05-14 2023-12-29 罗索肿瘤学公司 布鲁顿酪氨酸激酶抑制剂的共晶型
US20240327379A1 (en) * 2021-07-15 2024-10-03 Sandoz Ag Mandelate form of 1-(4-(((6-amino-5-(4-phenoxyphenyl)pyrimidin-4-yl)amino)methyl)piperidin-1-yl)prop-2-en-1-one
JP2025520698A (ja) 2022-06-24 2025-07-03 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツング 自己免疫疾患および炎症性疾患のための処置レジメン

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10060388A1 (de) * 2000-12-05 2002-06-06 Merck Patent Gmbh Verwendung von Pyrazolo [4,3-d]pyrimidinen
WO2011156900A2 (en) * 2010-06-17 2011-12-22 Waratah Pharmaceuticals Inc. Compounds, compositions and methods for treatment of multiple sclerosis
SG10201604682VA (en) * 2011-06-10 2016-07-28 Merck Patent Gmbh Compositions and methods for the production of pyrimidine and pyridine compounds with btk inhibitory activity
WO2013106535A1 (en) * 2012-01-10 2013-07-18 Nimbus Iris, Inc. Irak inhibitors and uses thereof
AR090885A1 (es) * 2012-05-02 2014-12-10 Teva Pharma Uso de laquinimod en alta dosis para el tratamiento de la esclerosis multiple
HRP20231547T1 (hr) 2015-11-17 2024-03-15 Merck Patent Gmbh Postupci liječenja multiple skleroze primjenom spojeva pirimidina i piridina s aktivnošću inhibicije btk
US10464923B2 (en) * 2017-02-27 2019-11-05 Merck Patent Gmbh Crystalline forms of 1-(4-{[6-amino-5-(4-phenoxy-phenyl)-pyrimidin-4-ylamino]-methyl}-piperidin-1-yl)-propenone

Also Published As

Publication number Publication date
UA127744C2 (uk) 2023-12-20
ES3009670T3 (en) 2025-03-31
BR112021000893A2 (pt) 2021-04-13
CA3106772A1 (en) 2020-01-23
CN112437665A (zh) 2021-03-02
IL280197A (en) 2021-03-01
US20210260060A1 (en) 2021-08-26
DK3823623T3 (da) 2025-01-02
WO2020016850A1 (en) 2020-01-23
SG11202100518TA (en) 2021-02-25
EP3823623A1 (en) 2021-05-26
AU2025203171A1 (en) 2025-05-22
TWI879737B (zh) 2025-04-11
US12251382B2 (en) 2025-03-18
HUE069840T2 (hu) 2025-04-28
ZA202101118B (en) 2025-06-25
JP7724151B2 (ja) 2025-08-15
TW202019425A (zh) 2020-06-01
EP3823623B1 (en) 2024-10-09
HRP20241737T1 (hr) 2025-02-28
AU2019306828A1 (en) 2021-03-11
JP2021532104A (ja) 2021-11-25
FI3823623T3 (fi) 2025-01-09
PT3823623T (pt) 2025-01-06
MX2021000094A (es) 2021-03-25
KR20210034623A (ko) 2021-03-30

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