PL2678333T3 - Ulepszony sposób otrzymywania worykonazolu i jego produktów pośrednich - Google Patents

Ulepszony sposób otrzymywania worykonazolu i jego produktów pośrednich

Info

Publication number
PL2678333T3
PL2678333T3 PL12709178T PL12709178T PL2678333T3 PL 2678333 T3 PL2678333 T3 PL 2678333T3 PL 12709178 T PL12709178 T PL 12709178T PL 12709178 T PL12709178 T PL 12709178T PL 2678333 T3 PL2678333 T3 PL 2678333T3
Authority
PL
Poland
Prior art keywords
voriconazole
intermediates
preparation
improved process
improved
Prior art date
Application number
PL12709178T
Other languages
English (en)
Inventor
Nitin Maheshwari
Roshan Ramesh Medhane
Mohan Prasad
Sudershan Kumar Arora
Original Assignee
Ranbaxy Laboratories Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ranbaxy Laboratories Ltd filed Critical Ranbaxy Laboratories Ltd
Publication of PL2678333T3 publication Critical patent/PL2678333T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PL12709178T 2011-02-21 2012-02-21 Ulepszony sposób otrzymywania worykonazolu i jego produktów pośrednich PL2678333T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IN433DE2011 2011-02-21
PCT/IB2012/050791 WO2012114273A1 (en) 2011-02-21 2012-02-21 An improved process for the preparation of voriconazole and intermediates thereof
EP12709178.3A EP2678333B1 (en) 2011-02-21 2012-02-21 An improved process for the preparation of voriconazole and intermediates thereof

Publications (1)

Publication Number Publication Date
PL2678333T3 true PL2678333T3 (pl) 2015-08-31

Family

ID=46720174

Family Applications (1)

Application Number Title Priority Date Filing Date
PL12709178T PL2678333T3 (pl) 2011-02-21 2012-02-21 Ulepszony sposób otrzymywania worykonazolu i jego produktów pośrednich

Country Status (7)

Country Link
US (1) US20140350252A1 (pl)
EP (1) EP2678333B1 (pl)
AU (1) AU2012221788A1 (pl)
CA (1) CA2827379A1 (pl)
PL (1) PL2678333T3 (pl)
WO (1) WO2012114273A1 (pl)
ZA (1) ZA201306212B (pl)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102898419A (zh) * 2012-11-15 2013-01-30 南京海陵中药制药工艺技术研究有限公司 一种制备伏立康唑中间体ⅰ的方法
CN105277629A (zh) * 2014-06-12 2016-01-27 陕西合成药业股份有限公司 一种分离分析伏立康唑磷酸酯或其药用盐异构体的hplc方法
CN105699498B (zh) * 2014-11-25 2020-06-12 陕西合成药业股份有限公司 一种分离分析伏立康唑磷酸酯或其药用盐有关物质的hplc方法
CN105503834B (zh) * 2015-12-23 2021-03-05 浙江华海药业股份有限公司 一种伏立康唑中间体的合成方法
CN111704606A (zh) * 2020-06-11 2020-09-25 广东隆赋药业股份有限公司 一种伏立康唑中间体的制备方法
CN112079819B (zh) * 2020-09-24 2022-06-17 南京易亨制药有限公司 一种改进的伏立康唑消旋体制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8819308D0 (en) 1988-08-13 1988-09-14 Pfizer Ltd Triazole antifungal agents
GB9002375D0 (en) 1990-02-02 1990-04-04 Pfizer Ltd Triazole antifungal agents
GB9516121D0 (en) * 1995-08-05 1995-10-04 Pfizer Ltd Organometallic addition to ketones

Also Published As

Publication number Publication date
EP2678333B1 (en) 2015-04-08
EP2678333A1 (en) 2014-01-01
ZA201306212B (en) 2014-04-30
WO2012114273A1 (en) 2012-08-30
CA2827379A1 (en) 2012-08-30
AU2012221788A1 (en) 2013-09-05
US20140350252A1 (en) 2014-11-27

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