PL2547683T3 - Sposób wytwarzania Sitagliptyny - Google Patents

Sposób wytwarzania Sitagliptyny

Info

Publication number
PL2547683T3
PL2547683T3 PL11718244T PL11718244T PL2547683T3 PL 2547683 T3 PL2547683 T3 PL 2547683T3 PL 11718244 T PL11718244 T PL 11718244T PL 11718244 T PL11718244 T PL 11718244T PL 2547683 T3 PL2547683 T3 PL 2547683T3
Authority
PL
Poland
Prior art keywords
preparing sitagliptin
sitagliptin
preparing
Prior art date
Application number
PL11718244T
Other languages
English (en)
Inventor
Jindrich Richter
Josef Jirman
Original Assignee
Zentiva Ks
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zentiva Ks filed Critical Zentiva Ks
Publication of PL2547683T3 publication Critical patent/PL2547683T3/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • General Chemical & Material Sciences (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Endocrinology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Catalysts (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
PL11718244T 2010-03-16 2011-03-15 Sposób wytwarzania Sitagliptyny PL2547683T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CZ20100198A CZ303113B6 (cs) 2010-03-16 2010-03-16 Zpusob prípravy sitagliptinu
PCT/CZ2011/000021 WO2011113399A1 (en) 2010-03-16 2011-03-15 Method of preparing sitagliptin
EP11718244.4A EP2547683B1 (en) 2010-03-16 2011-03-15 Method of preparing sitagliptin

Publications (1)

Publication Number Publication Date
PL2547683T3 true PL2547683T3 (pl) 2014-07-31

Family

ID=44168403

Family Applications (1)

Application Number Title Priority Date Filing Date
PL11718244T PL2547683T3 (pl) 2010-03-16 2011-03-15 Sposób wytwarzania Sitagliptyny

Country Status (7)

Country Link
EP (1) EP2547683B1 (pl)
BR (1) BR112012021591A2 (pl)
CZ (1) CZ303113B6 (pl)
EA (1) EA201290899A1 (pl)
ES (1) ES2457740T3 (pl)
PL (1) PL2547683T3 (pl)
WO (1) WO2011113399A1 (pl)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2674432A1 (en) 2012-06-14 2013-12-18 LEK Pharmaceuticals d.d. New synthetic route for the preparation of ß aminobutyryl substituted 5,6,7,8-tetrahydro[1,4]diazolo[4,3-alpha]pyrazin-7-yl compounds
US20150353564A1 (en) * 2013-01-22 2015-12-10 Apotex Technologies Inc. Processes for the Preparation of Chiral Beta Amino Acid Derivatives Using Asymmetric Hydrogenation Catalysts
CN103232455A (zh) * 2013-05-14 2013-08-07 聊城九州和谷生物科技有限公司 一种西他列汀的工业化生产方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5874629A (en) * 1996-06-12 1999-02-23 Merck & Co., Inc. Chiral bisphosphines
UA74912C2 (en) 2001-07-06 2006-02-15 Merck & Co Inc Beta-aminotetrahydroimidazo-(1,2-a)-pyrazines and tetratriazolo-(4,3-a)-pyrazines as inhibitors of dipeptylpeptidase for the treatment or prevention of diabetes
AR043515A1 (es) 2003-03-19 2005-08-03 Merck & Co Inc Procedimiento para preparar derivados quirales beta aminoacidos mediante hidrogenacion asimetrica
US7214813B2 (en) * 2003-05-30 2007-05-08 The Penn State Research Foundation Preparation of chiral cyclic amino acids and derivatives
GB0316439D0 (en) * 2003-07-15 2003-08-20 Johnson Matthey Plc Catalysts
TW200602293A (en) * 2004-04-05 2006-01-16 Merck & Co Inc Process for the preparation of enantiomerically enriched beta amino acid derivatives
AR052879A1 (es) 2005-01-24 2007-04-11 Merck & Co Inc Procedimiento para preparar derivados de beta aminoacidos quirales por hidrogenacion asimetrica

Also Published As

Publication number Publication date
EP2547683A1 (en) 2013-01-23
CZ2010198A3 (cs) 2011-09-29
BR112012021591A2 (pt) 2018-02-06
EP2547683B1 (en) 2014-02-19
WO2011113399A1 (en) 2011-09-22
ES2457740T3 (es) 2014-04-29
CZ303113B6 (cs) 2012-04-11
EA201290899A1 (ru) 2013-02-28

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