PL2491045T3 - Pochodne 2-okso-1-pirolidynyloimidazotiadiazolu - Google Patents

Pochodne 2-okso-1-pirolidynyloimidazotiadiazolu

Info

Publication number
PL2491045T3
PL2491045T3 PL10781818T PL10781818T PL2491045T3 PL 2491045 T3 PL2491045 T3 PL 2491045T3 PL 10781818 T PL10781818 T PL 10781818T PL 10781818 T PL10781818 T PL 10781818T PL 2491045 T3 PL2491045 T3 PL 2491045T3
Authority
PL
Poland
Prior art keywords
oxo
imidazothiadiazole derivatives
pyrrolidinyl
pyrrolidinyl imidazothiadiazole
derivatives
Prior art date
Application number
PL10781818T
Other languages
English (en)
Polish (pl)
Inventor
Yannick Quesnel
Laurent Turet
Joël Mercier
Original Assignee
Ucb Biopharma Sprl
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42034570&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL2491045(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ucb Biopharma Sprl filed Critical Ucb Biopharma Sprl
Publication of PL2491045T3 publication Critical patent/PL2491045T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/433Thidiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
PL10781818T 2009-10-23 2010-10-21 Pochodne 2-okso-1-pirolidynyloimidazotiadiazolu PL2491045T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP09173912 2009-10-23
EP10781818.9A EP2491045B1 (en) 2009-10-23 2010-10-21 2-oxo-1-pyrrolidinyl imidazothiadiazole derivatives
PCT/EP2010/006434 WO2011047860A1 (en) 2009-10-23 2010-10-21 2-oxo-1-pyrrolidinyl imidazothiadiazole derivatives

Publications (1)

Publication Number Publication Date
PL2491045T3 true PL2491045T3 (pl) 2016-06-30

Family

ID=42034570

Family Applications (1)

Application Number Title Priority Date Filing Date
PL10781818T PL2491045T3 (pl) 2009-10-23 2010-10-21 Pochodne 2-okso-1-pirolidynyloimidazotiadiazolu

Country Status (30)

Country Link
US (1) US8822508B2 (forum.php)
EP (1) EP2491045B1 (forum.php)
JP (1) JP5808020B2 (forum.php)
KR (1) KR20120102058A (forum.php)
CN (1) CN102574869A (forum.php)
AR (1) AR078722A1 (forum.php)
AU (1) AU2010310100B2 (forum.php)
BR (1) BR112012009310B8 (forum.php)
CA (1) CA2778194C (forum.php)
CL (1) CL2012001031A1 (forum.php)
CY (1) CY1117288T1 (forum.php)
DK (1) DK2491045T3 (forum.php)
EA (1) EA201200616A1 (forum.php)
ES (1) ES2565515T3 (forum.php)
HR (1) HRP20160263T1 (forum.php)
HU (1) HUE028668T2 (forum.php)
IL (1) IL218696A0 (forum.php)
IN (1) IN2012DN02793A (forum.php)
MA (1) MA33679B1 (forum.php)
ME (1) ME02355B (forum.php)
MX (1) MX347070B (forum.php)
PE (1) PE20121562A1 (forum.php)
PH (1) PH12012500570A1 (forum.php)
PL (1) PL2491045T3 (forum.php)
RS (1) RS54595B1 (forum.php)
SI (1) SI2491045T1 (forum.php)
SM (1) SMT201600076B (forum.php)
TN (1) TN2012000147A1 (forum.php)
TW (1) TW201118103A (forum.php)
WO (1) WO2011047860A1 (forum.php)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8957218B2 (en) * 2011-04-18 2015-02-17 Ucb Pharma S.A. 2-oxo-1-imidazolidinyl imidazothiadiazole derivatives
US9581654B2 (en) 2013-02-12 2017-02-28 Johnson Controls Technology Company Vehicle battery monitoring system
PT3096790T (pt) 2014-01-21 2019-10-15 Janssen Pharmaceutica Nv Combinações compreendendo moduladores alostéricos positivos ou agonistas ortostéricos do recetor glutamatérgico metabotrópico do subtipo 2 e seu uso
EP3827830A1 (en) 2014-01-21 2021-06-02 Janssen Pharmaceutica NV Combinations comprising positive allosteric modulators or orthosteric agonists of metabotropic glutamatergic receptor subtype 2 and their use
CN110869374B (zh) * 2017-07-10 2022-08-30 Ucb生物制药有限责任公司 2-氧代-1,3-噁唑烷基咪唑并噻二唑衍生物
MA49558A (fr) 2017-07-10 2021-05-05 UCB Biopharma SRL Dérivativés de 2-oxo-1-imidazolidinyl imidazothiadiazole
CN107827870B (zh) * 2017-10-24 2019-11-08 江苏仁明生物科技有限公司 一种正电子药物[18f]fpmmp及其制备方法与中间体
EA202091403A1 (ru) * 2017-12-12 2020-10-14 Юсб Байофарма Срл Производные 2-оксо-1-пирролидинилимидазотиадиазола
US11286266B2 (en) 2018-05-08 2022-03-29 UCB Biopharma SRL 1-imidazothiadiazolo-2H-pyrrol-5-one derivatives
CN113549052B (zh) * 2021-07-09 2022-09-02 首都医科大学脑重大疾病研究中心(北京脑重大疾病研究院) 4-苯基-1-(吡啶-4-基甲基)吡咯烷-2-酮衍生物及其制备方法和应用
WO2025132331A1 (en) 2023-12-21 2025-06-26 UCB Biopharma SRL Compounds for treatment of a hyperkinetic movement disorder
CN119606962B (zh) * 2025-02-17 2025-05-02 中国人民解放军总医院第三医学中心 padsevonil在制备治疗TFE3重排性肾细胞癌的药物中的应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8412358D0 (en) 1984-05-15 1984-06-20 Ucb Sa Pharmaceutical composition
GB8412357D0 (en) 1984-05-15 1984-06-20 Ucb Sa Pharmaceutical composition
GB0004297D0 (en) 2000-02-23 2000-04-12 Ucb Sa 2-oxo-1 pyrrolidine derivatives process for preparing them and their uses
ES2323313T3 (es) 2003-12-02 2009-07-13 Ucb Pharma, S.A. Derivados de imidazol, procedimientos para prepararlos y sus usos.
EP2308867A3 (en) * 2005-06-01 2011-10-19 UCB Pharma S.A. 2-oxo-1-pyrrolidine deriatives, processes for preparing them and their uses

Also Published As

Publication number Publication date
EA201200616A1 (ru) 2012-12-28
HRP20160263T1 (hr) 2016-04-08
BR112012009310B8 (pt) 2021-05-25
BR112012009310A2 (pt) 2016-06-07
ME02355B (me) 2016-06-20
MA33679B1 (fr) 2012-10-01
AU2010310100B2 (en) 2015-09-10
AU2010310100A1 (en) 2012-05-17
IL218696A0 (en) 2012-05-31
CA2778194A1 (en) 2011-04-28
DK2491045T3 (en) 2016-03-14
ES2565515T3 (es) 2016-04-05
CA2778194C (en) 2016-07-12
US20120245208A1 (en) 2012-09-27
CY1117288T1 (el) 2017-04-26
US8822508B2 (en) 2014-09-02
TN2012000147A1 (en) 2013-09-19
JP5808020B2 (ja) 2015-11-10
EP2491045B1 (en) 2015-12-23
AR078722A1 (es) 2011-11-30
MX347070B (es) 2017-04-11
RS54595B1 (en) 2016-08-31
SMT201600076B (it) 2016-04-29
PH12012500570A1 (en) 2012-10-22
EP2491045A1 (en) 2012-08-29
TW201118103A (en) 2011-06-01
MX2012003839A (es) 2012-05-08
CL2012001031A1 (es) 2012-09-14
HUE028668T2 (en) 2016-12-28
JP2013508321A (ja) 2013-03-07
CN102574869A (zh) 2012-07-11
BR112012009310B1 (pt) 2021-01-12
SI2491045T1 (sl) 2016-04-29
KR20120102058A (ko) 2012-09-17
PE20121562A1 (es) 2012-11-30
WO2011047860A1 (en) 2011-04-28
IN2012DN02793A (forum.php) 2015-07-24

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