PL1828125T3 - Pochodne arylopiperazyny i ich zastosowanie jako liganty selektywne receptora D3 dopaminy - Google Patents
Pochodne arylopiperazyny i ich zastosowanie jako liganty selektywne receptora D3 dopaminyInfo
- Publication number
- PL1828125T3 PL1828125T3 PL05822892T PL05822892T PL1828125T3 PL 1828125 T3 PL1828125 T3 PL 1828125T3 PL 05822892 T PL05822892 T PL 05822892T PL 05822892 T PL05822892 T PL 05822892T PL 1828125 T3 PL1828125 T3 PL 1828125T3
- Authority
- PL
- Poland
- Prior art keywords
- nrr
- alkylene
- polyfluoro
- alkyl
- dopamine
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/44—Iso-indoles; Hydrogenated iso-indoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Veterinary Medicine (AREA)
- Psychology (AREA)
- Addiction (AREA)
- Psychiatry (AREA)
- Gynecology & Obstetrics (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0412763A FR2878524B1 (fr) | 2004-12-01 | 2004-12-01 | Nouveaux derives d'arylpiperazine |
EP05822892A EP1828125B1 (fr) | 2004-12-01 | 2005-11-29 | Derives d'arylpiperazine et leur utilisation comme ligands selectifs du recepteur d3 de la dopamine |
PCT/FR2005/002964 WO2006058993A1 (fr) | 2004-12-01 | 2005-11-29 | Derives d’arylpiperazine et leur utilisation comme ligands selectifs du recepteur d3 de la dopamine |
Publications (1)
Publication Number | Publication Date |
---|---|
PL1828125T3 true PL1828125T3 (pl) | 2008-09-30 |
Family
ID=34951009
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PL05822892T PL1828125T3 (pl) | 2004-12-01 | 2005-11-29 | Pochodne arylopiperazyny i ich zastosowanie jako liganty selektywne receptora D3 dopaminy |
Country Status (12)
Country | Link |
---|---|
US (1) | US20080214542A1 (pl) |
EP (1) | EP1828125B1 (pl) |
AT (1) | ATE391711T1 (pl) |
DE (1) | DE602005006018T2 (pl) |
DK (1) | DK1828125T3 (pl) |
ES (1) | ES2302254T3 (pl) |
FR (1) | FR2878524B1 (pl) |
HR (1) | HRP20080187T3 (pl) |
PL (1) | PL1828125T3 (pl) |
PT (1) | PT1828125E (pl) |
SI (1) | SI1828125T1 (pl) |
WO (1) | WO2006058993A1 (pl) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU2006204522A1 (en) * | 2005-01-03 | 2006-07-13 | Universita Degli Studi Di Siena | Aryl piperazine derivatives for the treatment of neuropsychiatric disorders |
EP1870405A1 (en) * | 2006-06-22 | 2007-12-26 | Bioprojet | Carbonylated (Aza)cyclohexanes as dopamine D3 receptor ligands |
EP2238125A1 (en) * | 2008-02-01 | 2010-10-13 | NeuroSearch A/S | Novel aryl piperazine derivatives useful as modulators of dopamine and serotonin receptors |
EP2257531A1 (en) * | 2008-03-14 | 2010-12-08 | NeuroSearch A/S | Novel quinolinylamide derivatives useful as modulators of dopamine and serotonin receptors |
EP2354136B1 (en) | 2008-10-10 | 2016-02-24 | Institute Of Pharmacology And Toxicology Academy Of Military Medical Sciences P.L.A. China | Novel dopamine d3 receptor ligands and preparation and medical uses of the same |
US9227944B2 (en) | 2008-10-10 | 2016-01-05 | Institute Of Pharmacology And Toxicology Academy Of Military Science P.L.A. China | Dopamine D3 receptor ligands and preparation and medical uses of the same |
WO2014079504A1 (en) * | 2012-11-22 | 2014-05-30 | Biofordrug S.R.L. | Polycyclic ligands of 5-ht7 receptor and use thereof |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5523299A (en) * | 1992-08-06 | 1996-06-04 | Smithkline Beecham Plc | 5-(2-oxyphenyl)-pyrrole derivatives as dopamine D3 receptor antagonists |
US5523229A (en) * | 1994-03-22 | 1996-06-04 | Trustees Of The University Of Pennsylvania | Antibodies specific for oncofetal fibronectin |
WO2001049679A1 (en) * | 1999-12-30 | 2001-07-12 | H. Lundbeck A/S | 4-phenyl-1-piperazinyl, -piperidinyl and -tetrahydropyridyl derivatives |
EP1474399A1 (en) * | 2002-02-13 | 2004-11-10 | Glaxo Group Limited | Benzenesulfonamide derivatives as antipsychotic agents |
US20040204422A1 (en) * | 2003-04-14 | 2004-10-14 | Abbott Gmbh & Co. Kg. | N-[(Piperazinyl)hetaryl]arylsulfonamide compounds |
-
2004
- 2004-12-01 FR FR0412763A patent/FR2878524B1/fr not_active Expired - Fee Related
-
2005
- 2005-11-29 AT AT05822892T patent/ATE391711T1/de not_active IP Right Cessation
- 2005-11-29 EP EP05822892A patent/EP1828125B1/fr active Active
- 2005-11-29 SI SI200530267T patent/SI1828125T1/sl unknown
- 2005-11-29 PL PL05822892T patent/PL1828125T3/pl unknown
- 2005-11-29 US US11/720,526 patent/US20080214542A1/en not_active Abandoned
- 2005-11-29 DK DK05822892T patent/DK1828125T3/da active
- 2005-11-29 WO PCT/FR2005/002964 patent/WO2006058993A1/fr active Application Filing
- 2005-11-29 ES ES05822892T patent/ES2302254T3/es active Active
- 2005-11-29 DE DE602005006018T patent/DE602005006018T2/de not_active Expired - Fee Related
- 2005-11-29 PT PT05822892T patent/PT1828125E/pt unknown
-
2008
- 2008-04-23 HR HR20080187T patent/HRP20080187T3/xx unknown
Also Published As
Publication number | Publication date |
---|---|
WO2006058993A1 (fr) | 2006-06-08 |
DE602005006018D1 (de) | 2008-05-21 |
DE602005006018T2 (de) | 2008-07-10 |
FR2878524B1 (fr) | 2007-01-19 |
EP1828125A1 (fr) | 2007-09-05 |
EP1828125B1 (fr) | 2008-04-09 |
DK1828125T3 (da) | 2008-08-04 |
ATE391711T1 (de) | 2008-04-15 |
US20080214542A1 (en) | 2008-09-04 |
SI1828125T1 (sl) | 2008-08-31 |
ES2302254T3 (es) | 2008-07-01 |
PT1828125E (pt) | 2008-08-22 |
FR2878524A1 (fr) | 2006-06-02 |
HRP20080187T3 (en) | 2008-05-31 |
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