PH12014501625A1 - Novel 6-triazolopyridazinesulfanyl benzothiazole and benzimidazole derivatives, method for production thereof and application as medicaments and pharmaceutical compositions and novel use as met inhibitors - Google Patents

Novel 6-triazolopyridazinesulfanyl benzothiazole and benzimidazole derivatives, method for production thereof and application as medicaments and pharmaceutical compositions and novel use as met inhibitors

Info

Publication number
PH12014501625A1
PH12014501625A1 PH12014501625A PH12014501625A PH12014501625A1 PH 12014501625 A1 PH12014501625 A1 PH 12014501625A1 PH 12014501625 A PH12014501625 A PH 12014501625A PH 12014501625 A PH12014501625 A PH 12014501625A PH 12014501625 A1 PH12014501625 A1 PH 12014501625A1
Authority
PH
Philippines
Prior art keywords
phenyl
novel
medicaments
triazolopyridazinesulfanyl
benzothiazole
Prior art date
Application number
PH12014501625A
Other languages
English (en)
Inventor
Albert Eva
Bacque Eric
Nemecek Conception
Ugolini Antonio
Wentzler Sylvie
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/FR2008/001172 external-priority patent/WO2009056692A2/fr
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of PH12014501625A1 publication Critical patent/PH12014501625A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
PH12014501625A 2007-08-09 2014-07-15 Novel 6-triazolopyridazinesulfanyl benzothiazole and benzimidazole derivatives, method for production thereof and application as medicaments and pharmaceutical compositions and novel use as met inhibitors PH12014501625A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0705789A FR2919870B1 (fr) 2007-08-09 2007-08-09 Nouveaux derives de 6-triazolopyridazine-sulfanyl benzothiazole et benzothiazole et benzimidazole, procede, compositions pharmaceutiques et nouvelle utilisation comme inhibiteurs de cmet
PCT/FR2008/001172 WO2009056692A2 (fr) 2007-08-09 2008-08-06 Nouveaux derives de 6-triazolopyridazine-sulfanyl benzothiazole et benzimidazole, leur procede de preparation, leur application a titre de medicaments, compositions pharmaceutiques et nouvelle utilisation notamment comme inhibiteurs de met

Publications (1)

Publication Number Publication Date
PH12014501625A1 true PH12014501625A1 (en) 2016-01-18

Family

ID=39304792

Family Applications (1)

Application Number Title Priority Date Filing Date
PH12014501625A PH12014501625A1 (en) 2007-08-09 2014-07-15 Novel 6-triazolopyridazinesulfanyl benzothiazole and benzimidazole derivatives, method for production thereof and application as medicaments and pharmaceutical compositions and novel use as met inhibitors

Country Status (3)

Country Link
FR (1) FR2919870B1 (fr)
HN (1) HN2010000295A (fr)
PH (1) PH12014501625A1 (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102388048B (zh) 2009-02-10 2014-07-30 阿斯利康(瑞典)有限公司 三唑并[4,3-b]哒嗪衍生物及其用于前列腺癌的用途

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20080080584A (ko) * 2005-11-30 2008-09-04 버텍스 파마슈티칼스 인코포레이티드 c-Met의 억제제 및 이의 용도
UA98297C2 (en) * 2005-12-21 2012-05-10 Янссен Фармацевтика, Н.В. Triazolopyridazines as tyrosine kinase modulators
EP2032578A2 (fr) * 2006-05-30 2009-03-11 Pfizer Products Incorporated Dérivés de la triazolopyridazine
PE20121506A1 (es) * 2006-07-14 2012-11-26 Amgen Inc Compuestos triazolopiridinas como inhibidores de c-met

Also Published As

Publication number Publication date
HN2010000295A (es) 2013-04-22
FR2919870B1 (fr) 2014-05-16
FR2919870A1 (fr) 2009-02-13

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