PE20010041A1 - Derivados de 1-aminoetilindol, su preparacion y su aplicacion en terapeutica - Google Patents
Derivados de 1-aminoetilindol, su preparacion y su aplicacion en terapeuticaInfo
- Publication number
- PE20010041A1 PE20010041A1 PE2000000344A PE0003442000A PE20010041A1 PE 20010041 A1 PE20010041 A1 PE 20010041A1 PE 2000000344 A PE2000000344 A PE 2000000344A PE 0003442000 A PE0003442000 A PE 0003442000A PE 20010041 A1 PE20010041 A1 PE 20010041A1
- Authority
- PE
- Peru
- Prior art keywords
- alkyl
- aminoethylindol
- derivatives
- fluoroalkyl
- hydroxyethyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Urology & Nephrology (AREA)
- Otolaryngology (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
Abstract
SE REFIERE A DERIVADOS DE 1-AMINOETILINDOL DE FORMULA I, DONDE: A ES H, HALOGENO, HIDROXI; B Y D SON H, ALQUILO C1-C3; R1 ES H, ALQUILO C1-C4, FLUOROALQUILO C1-C2, PERFLUOROALQUILO C1-C2; R2 ES H, HALOGENO, ALQUILO C1-C6, CICLOALQUILO C3-C6, FLUOROALQUILO C1-C2, PERFLUOROALQUILO, FENILO; R3 Y R4 SON H, HALOGENO, ALQUILO C1-C6; R5 Y R6 SON H, ALQUILO C1-C6, FLUOROALQUILO C1-C2; R5 Y R6 JUNTOS SON ALQUILENO C2-C7. SON COMPUESTOS PREFERIDOS 2-METILINDOL-4-(1-DIETILAMINO-2-HIDROXIETIL)INDOL, 1(N)-METIL-2-ETILINDOL-4-(1-DIETILAMINO-2-HIDROXIETIL)INDOL, 1(N)-METIL-2-FENIL-4-(1-DIETILAMINO-2-HIDROXIETIL)INDOL, ENTRE OTROS. SE REFIERE TAMBIEN A UN PROCEDIMIENTO PARA LA PREPARACION. LOS DERIVADOS DE 1-AMINOETILINDOL DE FORMULA I TIENEN ACCION CONTRACTIL SOBRE LOS MUSCULOS LISOS URETRALES Y ARTERIALES Y PUEDEN SER UTILES PARA EL TRATAMIENTO DE INCONTINENCIA URINARIA DE ESFUERZO, INSUFICIENCIA VENOSA, MIGRANA, TRASTORNOS GASTROINTESTINALES
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9904577A FR2792316B1 (fr) | 1999-04-13 | 1999-04-13 | Derives de 1-aminoethylindole, leur preparation et leur application en therapeutique |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PE20010041A1 true PE20010041A1 (es) | 2001-04-12 |
Family
ID=9544316
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PE2000000344A PE20010041A1 (es) | 1999-04-13 | 2000-04-13 | Derivados de 1-aminoetilindol, su preparacion y su aplicacion en terapeutica |
Country Status (7)
| Country | Link |
|---|---|
| AR (1) | AR023451A1 (es) |
| AU (1) | AU3971400A (es) |
| CO (1) | CO5180549A1 (es) |
| FR (1) | FR2792316B1 (es) |
| PE (1) | PE20010041A1 (es) |
| UY (1) | UY26102A1 (es) |
| WO (1) | WO2000061554A1 (es) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR077405A1 (es) | 2009-07-10 | 2011-08-24 | Sanofi Aventis | Derivados del indol inhibidores de hsp90, composiciones que los contienen y utilizacion de los mismos para el tratamiento del cancer |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2752839B1 (fr) * | 1996-08-29 | 1998-10-09 | Synthelabo | Derives de benzofurane, leur preparation et leur application en therapeutique |
| FR2752840A1 (fr) * | 1996-08-29 | 1998-03-06 | Synthelabo | Derives de benzothiophene, leur preparation et leur application en therapeutique |
-
1999
- 1999-04-13 FR FR9904577A patent/FR2792316B1/fr not_active Expired - Fee Related
-
2000
- 2000-04-10 UY UY26102A patent/UY26102A1/es not_active Application Discontinuation
- 2000-04-11 WO PCT/FR2000/000922 patent/WO2000061554A1/fr active Application Filing
- 2000-04-11 CO CO00026489A patent/CO5180549A1/es not_active Application Discontinuation
- 2000-04-11 AU AU39714/00A patent/AU3971400A/en not_active Abandoned
- 2000-04-12 AR ARP000101669A patent/AR023451A1/es unknown
- 2000-04-13 PE PE2000000344A patent/PE20010041A1/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| AR023451A1 (es) | 2002-09-04 |
| UY26102A1 (es) | 2000-10-31 |
| WO2000061554A1 (fr) | 2000-10-19 |
| FR2792316B1 (fr) | 2001-06-22 |
| AU3971400A (en) | 2000-11-14 |
| CO5180549A1 (es) | 2002-07-30 |
| FR2792316A1 (fr) | 2000-10-20 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |