PA8793901A1 - Uso de gestágenos en combinación con (6s)-5-metiltetrahidrofolato para la terapia la endometriosis con simultánea reducción de los efectos colaterales terapéuticos, así como reducción del riesgo de malformaciones congénitas al comenzar un embarazo - Google Patents

Uso de gestágenos en combinación con (6s)-5-metiltetrahidrofolato para la terapia la endometriosis con simultánea reducción de los efectos colaterales terapéuticos, así como reducción del riesgo de malformaciones congénitas al comenzar un embarazo

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Publication number
PA8793901A1
PA8793901A1 PA20088793901A PA8793901A PA8793901A1 PA 8793901 A1 PA8793901 A1 PA 8793901A1 PA 20088793901 A PA20088793901 A PA 20088793901A PA 8793901 A PA8793901 A PA 8793901A PA 8793901 A1 PA8793901 A1 PA 8793901A1
Authority
PA
Panama
Prior art keywords
beginning
reduction
risk
therapy
combination
Prior art date
Application number
PA20088793901A
Other languages
English (en)
Inventor
Seitz Christian
Wasserfall Annemarie
Diefenbach Konstanze
Zimmermann Holger
King Kristina
Original Assignee
Bayer Schering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38846909&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PA8793901(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag
Publication of PA8793901A1 publication Critical patent/PA8793901A1/es

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/02Drugs for genital or sexual disorders; Contraceptives for disorders of the vagina
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/12Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18Feminine contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/02Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/34Gestagens

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Diabetes (AREA)
  • Gynecology & Obstetrics (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)

Abstract

SE USAN GESTAGENOS ANTIANDROGENICOS EN UNA UNIDAD DE DOSIS DIARIA QUE EQUIVALE A COMO MAXIMO EL DOBLE DE LA DOSIS INHIBIDORA DE LA OVULACION EN COMBINACION CON (6S) -5-METILTETRAHIDROFOLATO PARA OBTENER PREPARADOS FARMACEUTICOS PARA LA TERAPIA DE ENDOMETRIOSIS CON SIMULTANEA REDUCCION DE LOS EFECTOS COLATERALES TERAPEUTICOS, TALES COMO LA INFLUENCIA NEGATIVA SOBRE LA DENSIDAD OSEA/EL METABOLISMO OSEO Y EL RIESGO DE OSTEOPOROSIS, ASI COMO, EN EL CASO DE INICIADO UN EMBARAZO, LA REDUCCION DEL RIESGO DE MALFORMACIONES CONGENITAS, COMO DEFECTOS DEL TUBO NEURAL, FISURAS PALATINA, DE LABIOS Y MANDIBULA, Y COMPLICACIONES EN EL EMBARAZO, TALES COMO DESPRENDIMIENTO DE PLACENTA Y ABORTO. LA INVENCION ES APROPIADA PARA USAR A LARGO PLAZO.
PA20088793901A 2007-08-24 2008-08-22 Uso de gestágenos en combinación con (6s)-5-metiltetrahidrofolato para la terapia la endometriosis con simultánea reducción de los efectos colaterales terapéuticos, así como reducción del riesgo de malformaciones congénitas al comenzar un embarazo PA8793901A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP07016642A EP2027855A1 (de) 2007-08-24 2007-08-24 Verwendung von Gestagenen in Kombination mit (6S)5-Methyltetrahydrofolat zur Therapie der Endometriose mit gleichzeitiger Verminderung von Therapie-Nebenwirkungen sowie der Verminderung des Risikos angeborener Fehlbildungen bei Eintritt einer Gravidität

Publications (1)

Publication Number Publication Date
PA8793901A1 true PA8793901A1 (es) 2009-04-23

Family

ID=38846909

Family Applications (1)

Application Number Title Priority Date Filing Date
PA20088793901A PA8793901A1 (es) 2007-08-24 2008-08-22 Uso de gestágenos en combinación con (6s)-5-metiltetrahidrofolato para la terapia la endometriosis con simultánea reducción de los efectos colaterales terapéuticos, así como reducción del riesgo de malformaciones congénitas al comenzar un embarazo

Country Status (17)

Country Link
EP (2) EP2027855A1 (es)
JP (1) JP2010536808A (es)
KR (1) KR20100047872A (es)
CN (1) CN101784271A (es)
AR (1) AR070023A1 (es)
AU (1) AU2008291406A1 (es)
BR (1) BRPI0815756A2 (es)
CA (1) CA2696030A1 (es)
CL (1) CL2008002485A1 (es)
EA (1) EA201000338A1 (es)
MX (1) MX2010002190A (es)
PA (1) PA8793901A1 (es)
PE (1) PE20090608A1 (es)
TW (1) TW200930377A (es)
UY (1) UY31306A1 (es)
WO (1) WO2009027003A1 (es)
ZA (1) ZA201002035B (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101874806A (zh) * 2009-04-29 2010-11-03 北京本草天源药物研究院 一种地诺孕素固体制剂
CN108379226B (zh) * 2018-05-28 2019-11-29 上海市计划生育科学研究所 氯地孕酮自微乳组合物、其制备方法及应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH693255A5 (de) 1997-06-13 2003-05-15 Eprova Ag Verwendung von Tetrahydrofolaten in der natürlichenstereoisomeren Form zur Herstellung einer pharmazeutischenZubereitung geeignet zur Beeinflussung des Homocystein-Spiegels.
JP4418105B2 (ja) 1997-12-26 2010-02-17 持田製薬株式会社 ジエノゲストを有効成分とする血管新生抑制剤
CH693905A5 (de) 1999-04-15 2004-04-15 Eprova Ag Stabile kristalline Salze von 5-Methyltetrahydrofolsäure.
US20050032741A1 (en) * 2003-08-06 2005-02-10 Balaji Venkataraman Vitamin Compositions
DE102005034498A1 (de) * 2005-07-20 2007-01-25 Grünenthal GmbH Orale Kontrazeption mit Trimegeston
DE102005053771A1 (de) * 2005-11-09 2007-05-10 Grünenthal GmbH Darreichform zur hormonalen Kontrazeption

Also Published As

Publication number Publication date
UY31306A1 (es) 2008-11-28
KR20100047872A (ko) 2010-05-10
BRPI0815756A2 (pt) 2015-02-18
MX2010002190A (es) 2010-03-17
AR070023A1 (es) 2010-03-10
CL2008002485A1 (es) 2009-11-20
CA2696030A1 (en) 2009-03-05
EP2027855A1 (de) 2009-02-25
JP2010536808A (ja) 2010-12-02
TW200930377A (en) 2009-07-16
CN101784271A (zh) 2010-07-21
ZA201002035B (en) 2012-09-26
WO2009027003A1 (de) 2009-03-05
EA201000338A1 (ru) 2010-08-30
AU2008291406A1 (en) 2009-03-05
EP2194978A1 (de) 2010-06-16
PE20090608A1 (es) 2009-06-12

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