OA10239A - Distamycin a derivatives as anti-malarial agents - Google Patents
Distamycin a derivatives as anti-malarial agents Download PDFInfo
- Publication number
- OA10239A OA10239A OA60725A OA60725A OA10239A OA 10239 A OA10239 A OA 10239A OA 60725 A OA60725 A OA 60725A OA 60725 A OA60725 A OA 60725A OA 10239 A OA10239 A OA 10239A
- Authority
- OA
- OAPI
- Prior art keywords
- formula
- compounds
- above defined
- case
- group
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ITFI930083A IT1263089B (it) | 1993-04-26 | 1993-04-26 | Composti pirrol-amidinici, processi di preparazione e composizioni farmaceutiche che li contengono. |
Publications (1)
Publication Number | Publication Date |
---|---|
OA10239A true OA10239A (en) | 1997-10-07 |
Family
ID=11350437
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
OA60725A OA10239A (en) | 1993-04-26 | 1995-10-24 | Distamycin a derivatives as anti-malarial agents |
Country Status (9)
Country | Link |
---|---|
US (1) | US5670534A (it) |
EP (1) | EP0698011A1 (it) |
CN (1) | CN1125437A (it) |
AU (1) | AU6646394A (it) |
BR (1) | BR9406509A (it) |
CA (1) | CA2161552A1 (it) |
IT (1) | IT1263089B (it) |
OA (1) | OA10239A (it) |
WO (1) | WO1994025436A1 (it) |
Families Citing this family (23)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9416005D0 (en) * | 1994-08-08 | 1994-09-28 | Erba Carlo Spa | Peptidic compounds analogous to distamycin a and process for their preparation |
AU734715B2 (en) | 1996-02-26 | 2001-06-21 | California Institute Of Technology | Improved polyamides for binding in the minor groove of double stranded DNA |
AU6757698A (en) | 1996-02-26 | 1998-10-30 | California Institute Of Technology | Stereochemical control of the dna binding affinity, sequence specificity, and orientation-preference of chiral hairpin polyamides in the minor groove |
US6090947A (en) | 1996-02-26 | 2000-07-18 | California Institute Of Technology | Method for the synthesis of pyrrole and imidazole carboxamides on a solid support |
US6506906B1 (en) | 1996-02-26 | 2003-01-14 | California Institute Of Technology | Preparation and use of bifunctional molecules having DNA sequence binding specificity |
US6635417B1 (en) | 1996-07-31 | 2003-10-21 | California Institute Of Technology | Complex formation between DSDNA and oligomer of cyclic heterocycles |
US6555692B1 (en) | 1996-02-26 | 2003-04-29 | California Institute Of Technology | Preparation and use of bifunctional molecules having DNA sequence binding specificity |
US6143901A (en) * | 1996-07-31 | 2000-11-07 | Genesoft, Inc. | Complex formation between dsDNA and pyrrole imidazole polyamides |
US5998140A (en) * | 1996-07-31 | 1999-12-07 | The Scripps Research Institute | Complex formation between dsDNA and oligomer of cyclic heterocycles |
JP2003529609A (ja) | 2000-03-16 | 2003-10-07 | ジーンソフト インコーポレイティッド | 核酸結合部分を含む荷電した化合物およびその利用法 |
US7078536B2 (en) * | 2001-03-14 | 2006-07-18 | Genesoft Pharmaceuticals, Inc. | Charged compounds comprising a nucleic acid binding moiety and uses therefor |
WO2002101007A2 (en) * | 2001-06-13 | 2002-12-19 | Genesoft Pharmaceuticals, Inc | Antipathogenic benzamide compounds |
JP2005505508A (ja) * | 2001-06-13 | 2005-02-24 | ジーンソフト ファーマシューティカルズ インコーポレイテッド | 抗感染活性を有するベンゾチオフェン化合物 |
ITTO20010633A1 (it) | 2001-07-02 | 2003-01-02 | Univ Ferrara | Nuovo impiego di poliammidi eterocicliche e benzoeterocicliche strutturalmente correlate all'antibiotico naturale distamicina a. |
WO2004012736A1 (en) | 2002-08-02 | 2004-02-12 | Genesoft Pharmaceuticals, Inc. | Biaryl compounds having anti-infective activity |
EP1562931A2 (en) * | 2002-10-25 | 2005-08-17 | Genesoft Pharmaceuticals, Inc. | Anti-infective biaryl compounds |
JP2006509027A (ja) | 2002-12-10 | 2006-03-16 | オーシェント ファーマシューティカルズ コーポレーション | (ピロールカルボキサミド)−(ベンズアミド)−(イミダゾールカルボキサミド)モチーフを有する抗菌化合物 |
ITMI20031015A1 (it) * | 2003-05-20 | 2004-11-21 | Naxospharma S R L | Poli-(amminopirrolcarbossammidi) per uso nella profilassi e nel trattamento delle endoparassitosi animali e loro composizioni con ciclodestrine. |
ITMI20031111A1 (it) * | 2003-06-03 | 2004-12-04 | Naxospharma Srl | Processo per la sintesi della distramicina e analoghi poli-4-(1-metilpirrolo)-2-carbossiammidici. |
US7094791B2 (en) * | 2003-07-31 | 2006-08-22 | Avalon Pharmaceuticals, Inc. | Derivatives of 3-hydroxy-pyrrole-2,4-dicarboxylic acid and uses thereof |
SG155222A1 (en) * | 2004-08-13 | 2009-09-30 | Genentech Inc | Thiazole based inhibitors of atp-utilizing enzymes |
GB0619325D0 (en) * | 2006-09-30 | 2006-11-08 | Univ Strathclyde | New compounds |
US8494795B2 (en) * | 2008-05-05 | 2013-07-23 | Schweitzer Engineering Laboratories Inc | Apparatus and method for estimating synchronized phasors at predetermined times referenced to a common time standard in an electrical system |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1243389B (it) * | 1990-11-22 | 1994-06-10 | Menarini Farma Ind | Derivati poliaminopirrolcarbossiamidici, processi di preparazione e composizioni farmaceutiche che li contengono. |
IT1262921B (it) * | 1992-01-10 | 1996-07-22 | Federico Arcamone | Agenti antitumorali analoghi di oligopeptidi pirrol-amidinici retroversi processi di preparazione e prodotti farmaceutici che li contengono |
-
1993
- 1993-04-26 IT ITFI930083A patent/IT1263089B/it active IP Right Grant
-
1994
- 1994-04-21 AU AU66463/94A patent/AU6646394A/en not_active Abandoned
- 1994-04-21 EP EP94915076A patent/EP0698011A1/en not_active Withdrawn
- 1994-04-21 CA CA002161552A patent/CA2161552A1/en not_active Abandoned
- 1994-04-21 BR BR9406509A patent/BR9406509A/pt not_active Application Discontinuation
- 1994-04-21 CN CN94192517A patent/CN1125437A/zh active Pending
- 1994-04-21 US US08/549,737 patent/US5670534A/en not_active Expired - Fee Related
- 1994-04-21 WO PCT/EP1994/001235 patent/WO1994025436A1/en not_active Application Discontinuation
-
1995
- 1995-10-24 OA OA60725A patent/OA10239A/en unknown
Also Published As
Publication number | Publication date |
---|---|
ITFI930083A0 (it) | 1993-04-26 |
AU6646394A (en) | 1994-11-21 |
US5670534A (en) | 1997-09-23 |
CA2161552A1 (en) | 1994-11-10 |
EP0698011A1 (en) | 1996-02-28 |
WO1994025436A1 (en) | 1994-11-10 |
BR9406509A (pt) | 1996-01-09 |
CN1125437A (zh) | 1996-06-26 |
IT1263089B (it) | 1996-07-24 |
ITFI930083A1 (it) | 1994-10-26 |
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