NZ578475A - Napadisylate salt of a muscarinic m3 antagonist - Google Patents

Napadisylate salt of a muscarinic m3 antagonist

Info

Publication number
NZ578475A
NZ578475A NZ578475A NZ57847508A NZ578475A NZ 578475 A NZ578475 A NZ 578475A NZ 578475 A NZ578475 A NZ 578475A NZ 57847508 A NZ57847508 A NZ 57847508A NZ 578475 A NZ578475 A NZ 578475A
Authority
NZ
New Zealand
Prior art keywords
phenyl
oxazol
cyclohexyl
chloro
salt
Prior art date
Application number
NZ578475A
Other languages
English (en)
Inventor
Barbara Giuseppina Avitabile
David O'sullivan
Richard James Bull
Original Assignee
Pulmagen Therapeutics Synergy
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB0702416.9A external-priority patent/GB0702416D0/en
Priority claimed from GBGB0702385.6A external-priority patent/GB0702385D0/en
Application filed by Pulmagen Therapeutics Synergy, Astrazeneca Ab filed Critical Pulmagen Therapeutics Synergy
Publication of NZ578475A publication Critical patent/NZ578475A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/10—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D263/12—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with radicals containing only hydrogen and carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/32—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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  • General Chemical & Material Sciences (AREA)
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  • Pulmonology (AREA)
  • Biomedical Technology (AREA)
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  • Physical Education & Sports Medicine (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Oncology (AREA)
  • Neurosurgery (AREA)
  • Endocrinology (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Communicable Diseases (AREA)
  • Rheumatology (AREA)
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  • Reproductive Health (AREA)
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NZ578475A 2007-02-07 2008-02-06 Napadisylate salt of a muscarinic m3 antagonist NZ578475A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0702416.9A GB0702416D0 (en) 2007-02-07 2007-02-07 New combination
GBGB0702385.6A GB0702385D0 (en) 2007-02-07 2007-02-07 New combination
PCT/GB2008/000434 WO2008096149A2 (en) 2007-02-07 2008-02-06 Napadisylate salt of a muscarinic m3 antagonist

Publications (1)

Publication Number Publication Date
NZ578475A true NZ578475A (en) 2011-05-27

Family

ID=39485211

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ578475A NZ578475A (en) 2007-02-07 2008-02-06 Napadisylate salt of a muscarinic m3 antagonist

Country Status (13)

Country Link
US (1) US7846955B2 (OSRAM)
EP (1) EP2118078A2 (OSRAM)
JP (1) JP5373634B2 (OSRAM)
KR (1) KR20090119757A (OSRAM)
AU (1) AU2008212673B2 (OSRAM)
BR (1) BRPI0807004A2 (OSRAM)
CA (1) CA2675629A1 (OSRAM)
EC (1) ECSP099566A (OSRAM)
IL (1) IL199909A0 (OSRAM)
MX (1) MX2009008364A (OSRAM)
NZ (1) NZ578475A (OSRAM)
RU (1) RU2459810C2 (OSRAM)
WO (1) WO2008096149A2 (OSRAM)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0516313D0 (en) * 2005-08-08 2005-09-14 Argenta Discovery Ltd Azole derivatives and their uses
TW200825084A (en) 2006-11-14 2008-06-16 Astrazeneca Ab New compounds 521
NZ589091A (en) 2008-05-13 2011-07-29 Astrazeneca Ab Quinuclidine derivatives as muscarinic m3 receptor antagonists
TW201036957A (en) 2009-02-20 2010-10-16 Astrazeneca Ab Novel salt 628
ES2725784T3 (es) 2011-07-20 2019-09-27 Univ Brigham Young Compuestos de ceragenina hidrófobos y dispositivos que incorporan al mismo
US11524015B2 (en) 2013-03-15 2022-12-13 Brigham Young University Methods for treating inflammation, autoimmune disorders and pain
CN110420211A (zh) 2013-03-15 2019-11-08 布莱阿姆青年大学 治疗炎症、自身免疫性疾病和疼痛的方法
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MX2009008364A (es) 2009-08-20
AU2008212673B2 (en) 2011-04-28
CA2675629A1 (en) 2008-08-14
ECSP099566A (es) 2009-12-28
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EP2118078A2 (en) 2009-11-18
US20100093816A1 (en) 2010-04-15
US7846955B2 (en) 2010-12-07
KR20090119757A (ko) 2009-11-19
BRPI0807004A2 (pt) 2014-04-15
WO2008096149A2 (en) 2008-08-14
AU2008212673A1 (en) 2008-08-14
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